eF-site ID 2c5v-C
PDB Code 2c5v
Chain C

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Title Differential Binding Of Inhibitors To Active And Inactive Cdk2 Provides Insights For Drug Design
Classification CELL CYCLE
Compound CELL DIVISION PROTEIN KINASE 2
Source Homo sapiens (Human) (2C5V)
Sequence C:  MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTE
TEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVF
EFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHS
HRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYT
HEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRR
ALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSF
PKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAA
LAHPFFQDVTKPVPHL
Description


Functional site

1) chain C
residue 10
type
sequence I
description BINDING SITE FOR RESIDUE CK4 C1297
source : AC2

2) chain C
residue 31
type
sequence A
description BINDING SITE FOR RESIDUE CK4 C1297
source : AC2

3) chain C
residue 33
type
sequence K
description BINDING SITE FOR RESIDUE CK4 C1297
source : AC2

4) chain C
residue 80
type
sequence F
description BINDING SITE FOR RESIDUE CK4 C1297
source : AC2

5) chain C
residue 81
type
sequence E
description BINDING SITE FOR RESIDUE CK4 C1297
source : AC2

6) chain C
residue 83
type
sequence L
description BINDING SITE FOR RESIDUE CK4 C1297
source : AC2

7) chain C
residue 84
type
sequence H
description BINDING SITE FOR RESIDUE CK4 C1297
source : AC2

8) chain C
residue 85
type
sequence Q
description BINDING SITE FOR RESIDUE CK4 C1297
source : AC2

9) chain C
residue 86
type
sequence D
description BINDING SITE FOR RESIDUE CK4 C1297
source : AC2

10) chain C
residue 89
type
sequence K
description BINDING SITE FOR RESIDUE CK4 C1297
source : AC2

11) chain C
residue 134
type
sequence L
description BINDING SITE FOR RESIDUE CK4 C1297
source : AC2

12) chain C
residue 145
type
sequence D
description BINDING SITE FOR RESIDUE CK4 C1297
source : AC2


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