eF-site ID 2c4g-A
PDB Code 2c4g
Chain A

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Title STRUCTURE OF CDK2-CYCLIN A WITH PHA-533514
Classification TRANSFERASE
Compound CELL DIVISION PROTEIN KINASE 2
Source (CCNA2_HUMAN)
Sequence A:  PLVDMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIR
LDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKL
YLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLA
FCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPV
RTYTHEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEM
VTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDY
KPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRIS
AKAALAHPFFQDVTKPVPHLR
Description


Functional site

1) chain A
residue 256
type
sequence D
description BINDING SITE FOR RESIDUE SO4 A 305
source : AC1

2) chain A
residue 257
type
sequence E
description BINDING SITE FOR RESIDUE SO4 A 305
source : AC1

3) chain A
residue 260
type
sequence R
description BINDING SITE FOR RESIDUE SO4 A 305
source : AC1

4) chain A
residue 10
type
sequence I
description BINDING SITE FOR RESIDUE 514 A 306
source : AC3

5) chain A
residue 31
type
sequence A
description BINDING SITE FOR RESIDUE 514 A 306
source : AC3

6) chain A
residue 33
type
sequence K
description BINDING SITE FOR RESIDUE 514 A 306
source : AC3

7) chain A
residue 80
type
sequence F
description BINDING SITE FOR RESIDUE 514 A 306
source : AC3

8) chain A
residue 81
type
sequence E
description BINDING SITE FOR RESIDUE 514 A 306
source : AC3

9) chain A
residue 82
type
sequence F
description BINDING SITE FOR RESIDUE 514 A 306
source : AC3

10) chain A
residue 83
type
sequence L
description BINDING SITE FOR RESIDUE 514 A 306
source : AC3

11) chain A
residue 84
type
sequence H
description BINDING SITE FOR RESIDUE 514 A 306
source : AC3

12) chain A
residue 85
type
sequence Q
description BINDING SITE FOR RESIDUE 514 A 306
source : AC3

13) chain A
residue 86
type
sequence D
description BINDING SITE FOR RESIDUE 514 A 306
source : AC3

14) chain A
residue 89
type
sequence K
description BINDING SITE FOR RESIDUE 514 A 306
source : AC3

15) chain A
residue 134
type
sequence L
description BINDING SITE FOR RESIDUE 514 A 306
source : AC3

16) chain A
residue 10-33
type prosite
sequence IGEGTYGVVYKARNKLTGEVVALK
description PROTEIN_KINASE_ATP Protein kinases ATP-binding region signature. IGEGTYGVVYkArnkltgev..........VALK
source prosite : PS00107

17) chain A
residue 123-135
type prosite
sequence VLHRDLKPQNLLI
description PROTEIN_KINASE_ST Serine/Threonine protein kinases active-site signature. VlHrDLKpqNLLI
source prosite : PS00108


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