eF-site ID 2aob-B
PDB Code 2aob
Chain B

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Title Crystal structures of a high-affinity macrocyclic peptide mimetic in complex with the Grb2 SH2 domain
Classification TRANSFERASE
Compound Growth factor receptor-bound protein 2
Source Homo sapiens (Human) (GRB2_HUMAN)
Sequence B:  PWFFGKIPRAKAEEMLSKQRHDGAFLIRESESAPGDFSLS
VKFGNDVQHFKVLRDGAGKYFLWVVKFNSLNELVDYHRST
SVSRNQQIFLRDI
Description


Functional site

1) chain B
residue 67
type
sequence R
description BINDING SITE FOR RESIDUE S1S B 1301
source : AC2

2) chain B
residue 86
type
sequence R
description BINDING SITE FOR RESIDUE S1S B 1301
source : AC2

3) chain B
residue 96
type
sequence S
description BINDING SITE FOR RESIDUE S1S B 1301
source : AC2

4) chain B
residue 106
type
sequence Q
description BINDING SITE FOR RESIDUE S1S B 1301
source : AC2

5) chain B
residue 107
type
sequence H
description BINDING SITE FOR RESIDUE S1S B 1301
source : AC2

6) chain B
residue 108
type
sequence F
description BINDING SITE FOR RESIDUE S1S B 1301
source : AC2

7) chain B
residue 109
type
sequence K
description BINDING SITE FOR RESIDUE S1S B 1301
source : AC2

8) chain B
residue 111
type
sequence L
description BINDING SITE FOR RESIDUE S1S B 1301
source : AC2

9) chain B
residue 120
type
sequence L
description BINDING SITE FOR RESIDUE S1S B 1301
source : AC2

10) chain B
residue 121
type
sequence W
description BINDING SITE FOR RESIDUE S1S B 1301
source : AC2

11) chain B
residue 121
type
sequence W
description BINDING SITE FOR RESIDUE S1S A 1401
source : AC3

12) chain B
residue 122
type
sequence V
description BINDING SITE FOR RESIDUE S1S A 1401
source : AC3

13) chain B
residue 124
type
sequence K
description BINDING SITE FOR RESIDUE S1S A 1401
source : AC3

14) chain B
residue 125
type
sequence F
description BINDING SITE FOR RESIDUE S1S A 1401
source : AC3

15) chain B
residue 130
type
sequence E
description BINDING SITE FOR RESIDUE S1S A 1401
source : AC3

16) chain B
residue 126
type
sequence N
description BINDING SITE FOR RESIDUE S1S A 1501
source : AC4

17) chain B
residue 127
type
sequence S
description BINDING SITE FOR RESIDUE S1S A 1601
source : AC5

18) chain B
residue 128
type
sequence L
description BINDING SITE FOR RESIDUE S1S A 1601
source : AC5

19) chain B
residue 126
type
sequence N
description BINDING SITE FOR RESIDUE S1S A 1701
source : AC6

20) chain B
residue 127
type
sequence S
description BINDING SITE FOR RESIDUE S1S A 1701
source : AC6

21) chain B
residue 142
type
sequence R
description BINDING SITE FOR RESIDUE S1S C 2201
source : AC7

22) chain B
residue 109
type
sequence K
description BINDING SITE FOR RESIDUE S1S C 2401
source : AC9

23) chain B
residue 111
type
sequence L
description BINDING SITE FOR RESIDUE S1S C 2401
source : AC9

24) chain B
residue 112
type
sequence R
description BINDING SITE FOR RESIDUE S1S C 2501
source : BC1

25) chain B
residue 109
type MOD_RES
sequence K
description N6-acetyllysine => ECO:0007744|PubMed:19608861
source Swiss-Prot : SWS_FT_FI1


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