eF-site ID 1yxt-A
PDB Code 1yxt
Chain A

click to enlarge
Title Crystal Structure of Kinase Pim1 in complex with AMPPNP
Classification TRANSFERASE
Compound Proto-oncogene serine/threonine-protein kinase Pim-1
Source Homo sapiens (Human) (PIM1_HUMAN)
Sequence A:  PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKD
RISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFER
PDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVL
EAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGAL
LKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILL
YDMVCGDIPFEHDEEIIRGQVFFRQRVSSECQHLIRWCLA
LRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHS
Description


Functional site

1) chain A
residue 44
type
sequence L
description BINDING SITE FOR RESIDUE ANP A 322
source : AC1

2) chain A
residue 46
type
sequence S
description BINDING SITE FOR RESIDUE ANP A 322
source : AC1

3) chain A
residue 48
type
sequence G
description BINDING SITE FOR RESIDUE ANP A 322
source : AC1

4) chain A
residue 49
type
sequence F
description BINDING SITE FOR RESIDUE ANP A 322
source : AC1

5) chain A
residue 50
type
sequence G
description BINDING SITE FOR RESIDUE ANP A 322
source : AC1

6) chain A
residue 52
type
sequence V
description BINDING SITE FOR RESIDUE ANP A 322
source : AC1

7) chain A
residue 65
type
sequence A
description BINDING SITE FOR RESIDUE ANP A 322
source : AC1

8) chain A
residue 67
type
sequence K
description BINDING SITE FOR RESIDUE ANP A 322
source : AC1

9) chain A
residue 104
type
sequence I
description BINDING SITE FOR RESIDUE ANP A 322
source : AC1

10) chain A
residue 121
type
sequence E
description BINDING SITE FOR RESIDUE ANP A 322
source : AC1

11) chain A
residue 128
type
sequence D
description BINDING SITE FOR RESIDUE ANP A 322
source : AC1

12) chain A
residue 167
type
sequence D
description BINDING SITE FOR RESIDUE ANP A 322
source : AC1

13) chain A
residue 171
type
sequence E
description BINDING SITE FOR RESIDUE ANP A 322
source : AC1

14) chain A
residue 172
type
sequence N
description BINDING SITE FOR RESIDUE ANP A 322
source : AC1

15) chain A
residue 174
type
sequence L
description BINDING SITE FOR RESIDUE ANP A 322
source : AC1

16) chain A
residue 185
type
sequence I
description BINDING SITE FOR RESIDUE ANP A 322
source : AC1

17) chain A
residue 186
type
sequence D
description BINDING SITE FOR RESIDUE ANP A 322
source : AC1

18) chain A
residue 44-67
type prosite
sequence LGSGGFGSVYSGIRVSDNLPVAIK
description PROTEIN_KINASE_ATP Protein kinases ATP-binding region signature. LGSGGFGSVYsGirvsdnlp..........VAIK
source prosite : PS00107

19) chain A
residue 163-175
type prosite
sequence VLHRDIKDENILI
description PROTEIN_KINASE_ST Serine/Threonine protein kinases active-site signature. VlHrDIKdeNILI
source prosite : PS00108


Display surface

Download
Links