eF-site ID 1okw-D
PDB Code 1okw
Chain D

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Title Cyclin A binding groove inhibitor Ac-Arg-Arg-Leu-Asn-(m-Cl-Phe)-NH2
Classification TRANSFERASE/TRANSFERASE INHIBITOR
Compound CELL DIVISION PROTEIN KINASE 2
Source Homo sapiens (Human) (1OKW)
Sequence D:  VPDYHEDIHTYLREMEVKCKPKVGYMKKQPDITNSMRAIL
VDWLVEVGEEYKLQNETLHLAVNYIDRFLSSMSVLRGKLQ
LVGTAAMLLASKFEEIYPPEVAEFVYITDDTYTKKQVLRM
EHLVLKVLTFDLAAPTVNQFLTQYFLHQQPANCKVESLAM
FLGELSLIDADPYLKYLPSVIAGAAFHLALYTVTGQSWPE
SLIRKTGYTLESLKPCLMDLHQTYLKAPQHAQQSIREKYK
NSKYHGVSLLNPPETLNL
Description


Functional site

1) chain D
residue 210
type
sequence M
description BINDING SITE FOR CHAIN F OF ACE-ARG-ARG-LEU-ASN-FCL-NH2
source : AC2

2) chain D
residue 217
type
sequence W
description BINDING SITE FOR CHAIN F OF ACE-ARG-ARG-LEU-ASN-FCL-NH2
source : AC2

3) chain D
residue 220
type
sequence E
description BINDING SITE FOR CHAIN F OF ACE-ARG-ARG-LEU-ASN-FCL-NH2
source : AC2

4) chain D
residue 254
type
sequence Q
description BINDING SITE FOR CHAIN F OF ACE-ARG-ARG-LEU-ASN-FCL-NH2
source : AC2

5) chain D
residue 281
type
sequence I
description BINDING SITE FOR CHAIN F OF ACE-ARG-ARG-LEU-ASN-FCL-NH2
source : AC2

6) chain D
residue 282
type
sequence T
description BINDING SITE FOR CHAIN F OF ACE-ARG-ARG-LEU-ASN-FCL-NH2
source : AC2

7) chain D
residue 285
type
sequence T
description BINDING SITE FOR CHAIN F OF ACE-ARG-ARG-LEU-ASN-FCL-NH2
source : AC2


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