eF-site ID 1okw-B
PDB Code 1okw
Chain B

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Title Cyclin A binding groove inhibitor Ac-Arg-Arg-Leu-Asn-(m-Cl-Phe)-NH2
Classification TRANSFERASE/TRANSFERASE INHIBITOR
Compound CELL DIVISION PROTEIN KINASE 2
Source null (1OKW)
Sequence B:  VPDYHEDIHTYLREMEVKCKPKVGYMKKQPDITNSMRAIL
VDWLVEVGEEYKLQNETLHLAVNYIDRFLSSMSVLRGKLQ
LVGTAAMLLASKFEEIYPPEVAEFVYITDDTYTKKQVLRM
EHLVLKVLTFDLAAPTVNQFLTQYFLHQQPANCKVESLAM
FLGELSLIDADPYLKYLPSVIAGAAFHLALYTVTGQSWPE
SLIRKTGYTLESLKPCLMDLHQTYLKAPQHAQQSIREKYK
NSKYHGVSLLNPPETLNL
Description


Functional site

1) chain B
residue 210
type
sequence M
description BINDING SITE FOR CHAIN E OF ACE-ARG-ARG-LEU-ASN-FCL-NH2
source : AC1

2) chain B
residue 213
type
sequence I
description BINDING SITE FOR CHAIN E OF ACE-ARG-ARG-LEU-ASN-FCL-NH2
source : AC1

3) chain B
residue 220
type
sequence E
description BINDING SITE FOR CHAIN E OF ACE-ARG-ARG-LEU-ASN-FCL-NH2
source : AC1

4) chain B
residue 253
type
sequence L
description BINDING SITE FOR CHAIN E OF ACE-ARG-ARG-LEU-ASN-FCL-NH2
source : AC1

5) chain B
residue 254
type
sequence Q
description BINDING SITE FOR CHAIN E OF ACE-ARG-ARG-LEU-ASN-FCL-NH2
source : AC1

6) chain B
residue 281
type
sequence I
description BINDING SITE FOR CHAIN E OF ACE-ARG-ARG-LEU-ASN-FCL-NH2
source : AC1

7) chain B
residue 282
type
sequence T
description BINDING SITE FOR CHAIN E OF ACE-ARG-ARG-LEU-ASN-FCL-NH2
source : AC1

8) chain B
residue 283
type
sequence D
description BINDING SITE FOR CHAIN E OF ACE-ARG-ARG-LEU-ASN-FCL-NH2
source : AC1

9) chain B
residue 285
type
sequence T
description BINDING SITE FOR CHAIN E OF ACE-ARG-ARG-LEU-ASN-FCL-NH2
source : AC1

10) chain B
residue 211-242
type prosite
sequence RAILVDWLVEVGEEYKLQNETLHLAVNYIDRF
description CYCLINS Cyclins signature. RaiLvdWLvevgeeykLqnetLhlAVnYIDRF
source prosite : PS00292


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