eF-site ID 1oiy-A
PDB Code 1oiy
Chain A

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Title Structure of human Thr160-phospho CDK2/cyclin A complexed with a 6-cyclohexylmethyloxy-2-anilino-purine inhibitor
Classification KINASE
Compound CELL DIVISION PROTEIN KINASE 2
Source Homo sapiens (Human) (CGA2_HUMAN)
Sequence A:  SMENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLTE
GVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEF
LHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHR
VLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYXHE
VVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRAL
FPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPK
WARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALA
HPFFQDVTKPVPHL
Description


Functional site

1) chain A
residue 10
type
sequence I
description BINDING SITE FOR RESIDUE N41 A1298
source : AC2

2) chain A
residue 12
type
sequence E
description BINDING SITE FOR RESIDUE N41 A1298
source : AC2

3) chain A
residue 18
type
sequence V
description BINDING SITE FOR RESIDUE N41 A1298
source : AC2

4) chain A
residue 31
type
sequence A
description BINDING SITE FOR RESIDUE N41 A1298
source : AC2

5) chain A
residue 64
type
sequence V
description BINDING SITE FOR RESIDUE N41 A1298
source : AC2

6) chain A
residue 80
type
sequence F
description BINDING SITE FOR RESIDUE N41 A1298
source : AC2

7) chain A
residue 81
type
sequence E
description BINDING SITE FOR RESIDUE N41 A1298
source : AC2

8) chain A
residue 83
type
sequence L
description BINDING SITE FOR RESIDUE N41 A1298
source : AC2

9) chain A
residue 84
type
sequence H
description BINDING SITE FOR RESIDUE N41 A1298
source : AC2

10) chain A
residue 86
type
sequence D
description BINDING SITE FOR RESIDUE N41 A1298
source : AC2

11) chain A
residue 89
type
sequence K
description BINDING SITE FOR RESIDUE N41 A1298
source : AC2

12) chain A
residue 131
type
sequence Q
description BINDING SITE FOR RESIDUE N41 A1298
source : AC2

13) chain A
residue 132
type
sequence N
description BINDING SITE FOR RESIDUE N41 A1298
source : AC2

14) chain A
residue 134
type
sequence L
description BINDING SITE FOR RESIDUE N41 A1298
source : AC2

15) chain A
residue 10-33
type prosite
sequence IGEGTYGVVYKARNKLTGEVVALK
description PROTEIN_KINASE_ATP Protein kinases ATP-binding region signature. IGEGTYGVVYkArnkltgev..........VALK
source prosite : PS00107

16) chain A
residue 123-135
type prosite
sequence VLHRDLKPQNLLI
description PROTEIN_KINASE_ST Serine/Threonine protein kinases active-site signature. VlHrDLKpqNLLI
source prosite : PS00108


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