|
eF-site ID
|
1oi9-D |
PDB Code
|
1oi9 |
Chain
|
D |
|
click to enlarge
|
|
Title
|
Structure of human Thr160-phospho CDK2/cyclin A complexed with a 6-cyclohexylmethyloxy-2-anilino-purine inhibitor |
Classification
|
KINASE |
Compound
|
CELL DIVISION PROTEIN KINASE 2 |
Source
|
Homo sapiens (Human) (CGA2_HUMAN) |
|
Sequence
|
D: |
YHEDIHTYLREMEVKCKPKVGYMKKQPDITNSMRAILVDW
LVEVGEEYKLQNETLHLAVNYIDRFLSSMSVLRGKLQLVG
TAAMLLASKFEEIYPPEVAEFVYITDDTYTKKQVLRMEHL
VLKVLTFDLAAPTVNQFLTQYFLHQQPANCKVESLAMFLG
ELSLIDADPYLKYLPSVIAGAAFHLALYTVTGQSWPESLI
RKTGYTLESLKPCLMDLHQTYLKAPQHAQQSIREKYKNSK
YHGVSLLNPPETL
|
|
Description
|
|
Functional site
|
|
1)
|
chain |
D |
residue |
189 |
type |
|
sequence |
M
|
description |
BINDING SITE FOR RESIDUE SGM D1193
|
source |
: AC5
|
|
2)
|
chain |
D |
residue |
192 |
type |
|
sequence |
K
|
description |
BINDING SITE FOR RESIDUE SGM D1193
|
source |
: AC5
|
|
3)
|
chain |
D |
residue |
193 |
type |
|
sequence |
C
|
description |
BINDING SITE FOR RESIDUE SGM D1193
|
source |
: AC5
|
|
4)
|
chain |
D |
residue |
241 |
type |
|
sequence |
R
|
description |
BINDING SITE FOR RESIDUE SGM D1193
|
source |
: AC5
|
|
5)
|
chain |
D |
residue |
305 |
type |
|
sequence |
D
|
description |
BINDING SITE FOR RESIDUE SGM D1193
|
source |
: AC5
|
|
|
|