eF-site ID 1nl4-A
PDB Code 1nl4
Chain A

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Title Crystal Structure of Rat Farnesyl Transferase in Complex With A Potent Biphenyl Inhibitor
Classification TRANSFERASE
Compound Protein farnesyltransferase alpha subunit
Source Rattus norvegicus (Rat) (PFTB_RAT)
Sequence A:  FLSLDSPTYVLYRDRAEWADIDPVPQNDGPSPVVQIIYSE
KFRDVYDYFRAVLQRDERSERAFKLTRDAIELNAANYTVW
HFRRVLLRSLQKDLQEEMNYITAIIEEQPKNYQVWHHRRV
LVEWLKDPSQELEFIADILNQDAKNYHAWQHRQWVIQEFR
LWDNELQYVDQLLKEDVRNNSVWNQRHFVISNTTGYSDRA
VLEREVQYTLEMIKLVPHNESAWNYLKGILQDRGLSRYPN
LLNQLLDLQPSHSSPYLIAFLVDIYEDMLENQCDNKEDIL
NKALELCEILAKEKDTIRKEYWRYIGRSLQSK
Description


Functional site

1) chain A
residue 164
type
sequence K
description BINDING SITE FOR RESIDUE HFP B 501
source : AC2

2) chain A
residue 166
type
sequence Y
description BINDING SITE FOR RESIDUE HFP B 501
source : AC2

3) chain A
residue 166
type
sequence Y
description BINDING SITE FOR RESIDUE FTL B 1
source : AC3


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