|
eF-site ID
|
1nl4-A |
PDB Code
|
1nl4 |
Chain
|
A |
|
click to enlarge
|
|
Title
|
Crystal Structure of Rat Farnesyl Transferase in Complex With A Potent Biphenyl Inhibitor |
Classification
|
TRANSFERASE |
Compound
|
Protein farnesyltransferase alpha subunit |
Source
|
Rattus norvegicus (Rat) (PFTB_RAT) |
|
Sequence
|
A: |
FLSLDSPTYVLYRDRAEWADIDPVPQNDGPSPVVQIIYSE
KFRDVYDYFRAVLQRDERSERAFKLTRDAIELNAANYTVW
HFRRVLLRSLQKDLQEEMNYITAIIEEQPKNYQVWHHRRV
LVEWLKDPSQELEFIADILNQDAKNYHAWQHRQWVIQEFR
LWDNELQYVDQLLKEDVRNNSVWNQRHFVISNTTGYSDRA
VLEREVQYTLEMIKLVPHNESAWNYLKGILQDRGLSRYPN
LLNQLLDLQPSHSSPYLIAFLVDIYEDMLENQCDNKEDIL
NKALELCEILAKEKDTIRKEYWRYIGRSLQSK
|
|
Description
|
|
Functional site
|
|
1)
|
chain |
A |
residue |
164 |
type |
|
sequence |
K
|
description |
BINDING SITE FOR RESIDUE HFP B 501
|
source |
: AC2
|
|
2)
|
chain |
A |
residue |
166 |
type |
|
sequence |
Y
|
description |
BINDING SITE FOR RESIDUE HFP B 501
|
source |
: AC2
|
|
3)
|
chain |
A |
residue |
166 |
type |
|
sequence |
Y
|
description |
BINDING SITE FOR RESIDUE FTL B 1
|
source |
: AC3
|
|
|
|