|
eF-site ID
|
1jlg-B |
PDB Code
|
1jlg |
Chain
|
B |
|
click to enlarge
|
|
Title
|
CRYSTAL STRUCTURE OF Y188C MUTANT HIV-1 REVERSE TRANSCRIPTASE IN COMPLEX WITH UC-781 |
Classification
|
TRANSFERASE |
Compound
|
HIV-1 RT A-chain |
Source
|
Human immunodeficiency virus type 1 group M subtype B (isolate HXB2) (HIV-1) (POL_HV1H2) |
|
Sequence
|
B: |
ETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTEMEKEG
KISKIGPENPYNTPVFAIKKKDSTKWRKLVDFRELNKRTQ
DFWGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTA
FTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILE
PFRKQNPDIVIYQYMDDLCVGSDLEIGQHRTKIEELRQHL
LRWGELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWAS
QIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENRE
ILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKN
LKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPK
FKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQ
LEKEP
|
|
Description
|
|
Functional site
|
|
1)
|
chain |
B |
residue |
111 |
type |
BINDING |
sequence |
V
|
description |
BINDING => ECO:0000250
|
source |
Swiss-Prot : SWS_FT_FI1
|
|
2)
|
chain |
B |
residue |
186 |
type |
BINDING |
sequence |
D
|
description |
BINDING => ECO:0000250
|
source |
Swiss-Prot : SWS_FT_FI1
|
|
3)
|
chain |
B |
residue |
187 |
type |
BINDING |
sequence |
L
|
description |
BINDING => ECO:0000250
|
source |
Swiss-Prot : SWS_FT_FI1
|
|
4)
|
chain |
B |
residue |
402 |
type |
SITE |
sequence |
W
|
description |
Essential for RT p66/p51 heterodimerization => ECO:0000250
|
source |
Swiss-Prot : SWS_FT_FI3
|
|
5)
|
chain |
B |
residue |
415 |
type |
SITE |
sequence |
E
|
description |
Essential for RT p66/p51 heterodimerization => ECO:0000250
|
source |
Swiss-Prot : SWS_FT_FI3
|
|
|
|