|
eF-site ID
|
1hrn-B |
PDB Code
|
1hrn |
Chain
|
B |
|
click to enlarge
|
|
Title
|
HIGH RESOLUTION CRYSTAL STRUCTURES OF RECOMBINANT HUMAN RENIN IN COMPLEX WITH POLYHYDROXYMONOAMIDE INHIBITORS |
Classification
|
HYDROLASE/HYDROLASE INHIBITOR |
Compound
|
RENIN |
Source
|
(RENI_HUMAN) |
|
Sequence
|
B: |
GNTTSSVILTNYMDTQYYGEIGIGTPPQTFKVVFDTGSSN
VWVPSSKCSRLYTACVYHKLFDASDSSSYKHNGTELTLRY
STGTVSGFLSQDIITVGGITVTQMFGEVTEMPALPFMLAE
FDGVVGMGFIEQAIGRVTPIFDNIISQGVLKEDVFSFYYN
RDSESLGGQIVLGGSDPQHYEGNFHYINLIKTGVWQIQMK
GVSVGSSTLLCEDGCLALVDTGASYISGSTSSIEKLMEAL
GAKKRLFDYVVKCNEGPTLPDISFHLGGKEYTLTSADYVF
QESYSSKKLCTLAIHAMDIPPPTGPTWALGATFIRKFYTE
FDRRNNRIGFALAR
|
|
Description
|
(1) |
RENIN COMPLEXED WITH POLYHYDROXYMONOAMIDE INHIBITOR BILA 980
|
|
Functional site
|
|
1)
|
chain |
B |
residue |
32 |
type |
ACT_SITE |
sequence |
D
|
description |
ACT_SITE => ECO:0000269|PubMed:20927107
|
source |
Swiss-Prot : SWS_FT_FI1
|
|
2)
|
chain |
B |
residue |
215 |
type |
ACT_SITE |
sequence |
D
|
description |
ACT_SITE => ECO:0000269|PubMed:20927107
|
source |
Swiss-Prot : SWS_FT_FI1
|
|
3)
|
chain |
B |
residue |
-1 |
type |
CARBOHYD |
sequence |
N
|
description |
N-linked (GlcNAc...) asparagine => ECO:0000269|PubMed:2493678
|
source |
Swiss-Prot : SWS_FT_FI2
|
|
4)
|
chain |
B |
residue |
67 |
type |
CARBOHYD |
sequence |
N
|
description |
N-linked (GlcNAc...) asparagine => ECO:0000269|PubMed:2493678
|
source |
Swiss-Prot : SWS_FT_FI2
|
|
|
|