eF-site ID 1h9u-A
PDB Code 1h9u
Chain A

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Title The structure of the human retinoid-X-receptor beta ligand binding domain in complex with the specific synthetic agonist LG100268
Classification NUCLEAR RECEPTOR
Compound RETINOID X RECEPTOR, BETA
Source Homo sapiens (Human) (RXRB_HUMAN)
Sequence A:  MPVDRILEAELAVPVTNICQAADKQLFTLVEWAKRIPHFS
SLPLDDQVILLRAGWNELLIASFSHRSIDVRDGILLATGL
HVHRNSAHSAGVGAIFDRVLTELVSKMRDMRMDKTELGCL
RAIILFNPDAKGLSNPSEVEVLREKVYASLETYCKQKYPE
QQGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTF
L
Description


Functional site

1) chain A
residue 402
type
sequence H
description BINDING SITE FOR RESIDUE NI A 2
source : AC1

2) chain A
residue 404
type
sequence H
description BINDING SITE FOR RESIDUE NI A 2
source : AC1

3) chain A
residue 404
type
sequence H
description BINDING SITE FOR RESIDUE CL A 3
source : AC2

4) chain A
residue 339
type
sequence I
description BINDING SITE FOR RESIDUE LG2 A 1
source : AC7

5) chain A
residue 342
type
sequence A
description BINDING SITE FOR RESIDUE LG2 A 1
source : AC7

6) chain A
residue 343
type
sequence A
description BINDING SITE FOR RESIDUE LG2 A 1
source : AC7

7) chain A
residue 346
type
sequence Q
description BINDING SITE FOR RESIDUE LG2 A 1
source : AC7

8) chain A
residue 376
type
sequence W
description BINDING SITE FOR RESIDUE LG2 A 1
source : AC7

9) chain A
residue 380
type
sequence L
description BINDING SITE FOR RESIDUE LG2 A 1
source : AC7

10) chain A
residue 381
type
sequence I
description BINDING SITE FOR RESIDUE LG2 A 1
source : AC7

11) chain A
residue 384
type
sequence F
description BINDING SITE FOR RESIDUE LG2 A 1
source : AC7

12) chain A
residue 387
type
sequence R
description BINDING SITE FOR RESIDUE LG2 A 1
source : AC7

13) chain A
residue 397
type
sequence L
description BINDING SITE FOR RESIDUE LG2 A 1
source : AC7

14) chain A
residue 398
type
sequence A
description BINDING SITE FOR RESIDUE LG2 A 1
source : AC7

15) chain A
residue 416
type
sequence I
description BINDING SITE FOR RESIDUE LG2 A 1
source : AC7

16) chain A
residue 503
type
sequence C
description BINDING SITE FOR RESIDUE LG2 A 1
source : AC7

17) chain A
residue 506
type
sequence H
description BINDING SITE FOR RESIDUE LG2 A 1
source : AC7


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