|
eF-site ID
|
1g65-T |
PDB Code
|
1g65 |
Chain
|
T |
|
click to enlarge
|
|
Title
|
Crystal structure of epoxomicin:20s proteasome reveals a molecular basis for selectivity of alpha,beta-epoxyketone proteasome inhibitors |
Classification
|
HYDROLASE/HYDROLASE inhibitor |
Compound
|
Proteasome component Y7 |
Source
|
ORGANISM_COMMON: Baker's yeast; ORGANISM_SCIENTIFIC: Saccharomyces cerevisiae; |
|
Sequence
|
T: |
GTGYDLSNSVFSPDGRNFQVEYAVKAVENGTTSIGIKCND
GVVFAVEKLITSKLLVPQKNVKIQVVDRHIGCVYSGLIPD
GRHLVNRGREEAASFKKLYKTPIPIPAFADRLGQYVQAHT
LYNSVRPFGVSTIFGGVDKNGAHLYMLEPSGSYWGYKGAA
TGKGRQSAKAELEKLVDHHPEGLSAREAVKQAAKIIYLAH
EDNKEKDFELEISWCSLSETNGLHKFVKGDLLQEAIDFAQ
KEIN
|
|
Description
|
|
|
|