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eF-site ID
|
1g65-A |
PDB Code
|
1g65 |
Chain
|
A |
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click to enlarge
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Title
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Crystal structure of epoxomicin:20s proteasome reveals a molecular basis for selectivity of alpha,beta-epoxyketone proteasome inhibitors |
Classification
|
HYDROLASE/HYDROLASE inhibitor |
Compound
|
Proteasome component Y7 |
Source
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ORGANISM_COMMON: Baker's yeast; ORGANISM_SCIENTIFIC: Saccharomyces cerevisiae; |
|
Sequence
|
A: |
MTDRYSFSLTTFSPSGKLGQIDYALTAVKQGVTSLGIKAT
NGVVIATEKKSSSPLAMSETLSKVSLLTPDIGAVYSGMGP
DYRVLVDKSRKVAHTSYKRIYGEYPPTKLLVSEVAKIMQE
ATQSGGVRPFGVSLLIAGHDEFNGFSLYQVDPSGSYFPWK
ATAIGKGSVAAKTFLEKRWNDELELEDAIHIALLTLKESV
EGEFNGDTIELAIIGDENPDLLGYTGIPTDKGPRFRKLTS
QEINDRLEAL
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Description
|
|
Functional site
|
|
1)
|
chain |
A |
residue |
8 |
type |
|
sequence |
Y
|
description |
BINDING SITE FOR RESIDUE MG F 302
|
source |
: AC3
|
|
2)
|
chain |
A |
residue |
8-30 |
type |
prosite |
sequence |
YSFSLTTFSPSGKLGQIDYALTA
|
description |
PROTEASOME_ALPHA_1 Proteasome alpha-type subunits signature. YdralSiFSPdGHifQVEYAleA
|
source |
prosite : PS00388
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