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Cytochrome P411 P-4 A82L A78V F263L amination catalyst
Descriptor:	NADPH-cytochrome P450 reductase 102A1V3, PROTOPORPHYRIN IX CONTAINING FE
Authors:	Zhang, R.K, Buller, A.R, Arnold, F.H.
Deposit date:	2016-12-22
Release date:	2017-05-17
Last modified:	2023-10-04
Method:	X-RAY DIFFRACTION (1.7 Å)
Cite:	Enantioselective, intermolecular benzylic C-H amination catalysed by an engineered iron-haem enzyme. Nat Chem, 9, 2017

Crystal Structure of the first bromodomain of human BRD4 in complex with 5-((4-fluoro-1H-imidazol-1-yl)methyl)quinolin-8-ol
Descriptor:	5-[(4-fluoranylimidazol-1-yl)methyl]quinolin-8-ol, Bromodomain-containing protein 4
Authors:	Xing, J, Zhang, R.K, Zheng, M.Y, Luo, C, Jiang, X.R.
Deposit date:	2018-08-08
Release date:	2018-12-12
Last modified:	2024-03-27
Method:	X-RAY DIFFRACTION (1.998 Å)
Cite:	Rational design of 5-((1H-imidazol-1-yl)methyl)quinolin-8-ol derivatives as novel bromodomain-containing protein 4 inhibitors Eur J Med Chem, 163, 2018