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3F6X
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c-Src kinase domain in complex with small molecule inhibitor
Descriptor: Proto-oncogene tyrosine-protein kinase Src, [4-({4-[(5-cyclopropyl-1H-pyrazol-3-yl)amino]quinazolin-2-yl}amino)phenyl]acetonitrile
Authors:Seeliger, M.A, Statsuk, A.V, Maly, D.J, Patrick, P.Z, Kuriyan, J, Shokat, K.M.
Deposit date:2008-11-06
Release date:2008-12-09
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (2.35 Å)
Cite:Tuning a three-component reaction for trapping kinase substrate complexes.
J.Am.Chem.Soc., 130, 2008

217705

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