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6GQ7
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BU of 6gq7 by Molmil
PI3Kg IN COMPLEX WITH INH
Descriptor: 3-methyl-1-(oxan-4-yl)-8-pyridin-3-yl-imidazo[4,5-c]quinolin-2-one, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Authors:Petersen, J.
Deposit date:2018-06-07
Release date:2018-06-20
Method:X-RAY DIFFRACTION (2.84 Å)
Cite:PI3Kg IN COMPLEX WITH INH
To Be Published
4Z7U
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BU of 4z7u by Molmil
S13 complex
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, MHC class II HLA-DQ-alpha chain, MHC class II HLA-DQ-beta-1, ...
Authors:Petersen, J, Rossjohn, J, Reid, H.H, Koning, F.
Deposit date:2015-04-08
Release date:2015-06-03
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.7 Å)
Cite:Determinants of Gliadin-Specific T Cell Selection in Celiac Disease.
J Immunol., 194, 2015
4Z7W
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BU of 4z7w by Molmil
T316 complex
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, DQ8-glia-alpha1, MHC class II HLA-DQ-alpha chain, ...
Authors:Petersen, J, Rossjohn, J, Reid, H.H, Koning, F.
Deposit date:2015-04-08
Release date:2015-06-03
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.89 Å)
Cite:Determinants of Gliadin-Specific T Cell Selection in Celiac Disease.
J Immunol., 194, 2015
4Z7V
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BU of 4z7v by Molmil
L3-12 complex
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, MHC class II HLA-DQ-alpha chain, MHC class II HLA-DQ-beta-1, ...
Authors:Petersen, J, Rossjohn, J, Reid, H.H, Koning, F.
Deposit date:2015-04-08
Release date:2015-06-03
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.65 Å)
Cite:Determinants of Gliadin-Specific T Cell Selection in Celiac Disease.
J Immunol., 194, 2015
5KSB
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BU of 5ksb by Molmil
T15-DQ8.5-glia-gamma1 complex
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, DQ8.5-glia-gamma1 peptide, ...
Authors:Petersen, J, Rossjohn, J, Reid, H.H.
Deposit date:2016-07-08
Release date:2016-09-21
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (2.9 Å)
Cite:Diverse T Cell Receptor Gene Usage in HLA-DQ8-Associated Celiac Disease Converges into a Consensus Binding Solution.
Structure, 24, 2016
5KS9
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BU of 5ks9 by Molmil
Bel502-DQ8-glia-alpha1 complex
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, Bel502 TCR alpha TRAV20*01, Bel502 TCR beta TRBV9*01, ...
Authors:Petersen, J, Rossjohn, J, Reid, H.H.
Deposit date:2016-07-08
Release date:2016-09-21
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (2.55 Å)
Cite:Diverse T Cell Receptor Gene Usage in HLA-DQ8-Associated Celiac Disease Converges into a Consensus Binding Solution.
Structure, 24, 2016
5KSA
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BU of 5ksa by Molmil
Bel602-DQ8.5-glia-gamma1 complex
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, Bel602 alpha TRAV20*01, Bel602 beta TRBV9*01, ...
Authors:Petersen, J, Rossjohn, J, Reid, H.H.
Deposit date:2016-07-08
Release date:2016-09-21
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (2 Å)
Cite:Diverse T Cell Receptor Gene Usage in HLA-DQ8-Associated Celiac Disease Converges into a Consensus Binding Solution.
Structure, 24, 2016
6U3O
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BU of 6u3o by Molmil
JR51 DQ2-p.aeru-alpha2a complex
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, MHC class II HLA-DQ-alpha chain, MHC class II HLA-DQ-beta-1, ...
Authors:Petersen, J, Rossjohn, J.
Deposit date:2019-08-22
Release date:2019-12-18
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (2.743 Å)
Cite:T cell receptor cross-reactivity between gliadin and bacterial peptides in celiac disease.
Nat.Struct.Mol.Biol., 27, 2020
6U3N
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BU of 6u3n by Molmil
LS2.8/3.15 - DQ2-P.fluor-alpha1a complex
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, MHC class II HLA-DQ-alpha chain, MHC class II HLA-DQ-beta-1, ...
Authors:Petersen, J, Rossjohn, J.
Deposit date:2019-08-22
Release date:2019-12-18
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (2.8 Å)
Cite:T cell receptor cross-reactivity between gliadin and bacterial peptides in celiac disease.
Nat.Struct.Mol.Biol., 27, 2020
6U3M
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BU of 6u3m by Molmil
DQ2-P.fluor-alpha1a
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Alpha1a peptide, ...
Authors:Petersen, J, Rossjohn, J.
Deposit date:2019-08-22
Release date:2019-12-18
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:T cell receptor cross-reactivity between gliadin and bacterial peptides in celiac disease.
Nat.Struct.Mol.Biol., 27, 2020
1UIS
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BU of 1uis by Molmil
The 2.0 crystal structure of eqFP611, a far-red fluorescent protein from the sea anemone Entacmaea quadricolor
Descriptor: ACETIC ACID, CALCIUM ION, red fluorescent protein FP611
Authors:Petersen, J, Wilmann, P.G, Beddoe, T, Oakley, A.J, Devenish, R.J, Prescott, M, Rossjohn, J.
Deposit date:2003-07-21
Release date:2003-10-21
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (2 Å)
Cite:The 2.0A crystal structure of eqFP611, a far-red fluorescent protein from the sea anemone Entacmaea quadricolor
J.Biol.Chem., 278, 2003
3FQU
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BU of 3fqu by Molmil
Phosphorylation of self-peptides alters Human Leukocyte Antigen Class I-restricted antigen presentation and generates tumor specific epitopes
Descriptor: Beta-2-microglobulin, CADMIUM ION, GLYCEROL, ...
Authors:Petersen, J, Rossjohn, J.
Deposit date:2009-01-07
Release date:2009-03-03
Last modified:2023-11-01
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Phosphorylated self-peptides alter human leukocyte antigen class I-restricted antigen presentation and generate tumor-specific epitopes
Proc.Natl.Acad.Sci.Usa, 106, 2009
3FQR
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BU of 3fqr by Molmil
Phosphorylation of self-peptides alters Human Leukocyte Antigen Class I-restricted antigen presentation and generates tumor specific epitopes
Descriptor: Beta-2-microglobulin, CADMIUM ION, GLYCEROL, ...
Authors:Petersen, J, Rossjohn, J.
Deposit date:2009-01-07
Release date:2009-03-03
Last modified:2023-11-01
Method:X-RAY DIFFRACTION (1.7 Å)
Cite:Phosphorylated self-peptides alter human leukocyte antigen class I-restricted antigen presentation and generate tumor-specific epitopes
Proc.Natl.Acad.Sci.Usa, 106, 2009
3FQN
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BU of 3fqn by Molmil
Phosphorylation of self-peptides alters Human Leukocyte Antigen Class I-restricted antigen presentation and generates tumor specific epitopes
Descriptor: Beta-2-microglobulin, CADMIUM ION, GLYCEROL, ...
Authors:Petersen, J, Rossjohn, J.
Deposit date:2009-01-07
Release date:2009-03-03
Last modified:2023-11-01
Method:X-RAY DIFFRACTION (1.65 Å)
Cite:Phosphorylated self-peptides alter human leukocyte antigen class I-restricted antigen presentation and generate tumor-specific epitopes
Proc.Natl.Acad.Sci.Usa, 106, 2009
3FQX
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BU of 3fqx by Molmil
Phosphorylation of self-peptides alters Human Leukocyte Antigen Class I-restricted antigen presentation and generates tumor specific epitopes
Descriptor: Beta-2-microglobulin, CADMIUM ION, GLYCEROL, ...
Authors:Petersen, J, Rossjohn, J.
Deposit date:2009-01-07
Release date:2009-03-03
Last modified:2023-11-01
Method:X-RAY DIFFRACTION (1.7 Å)
Cite:Phosphorylated self-peptides alter human leukocyte antigen class I-restricted antigen presentation and generate tumor-specific epitopes
Proc.Natl.Acad.Sci.Usa, 106, 2009
3FQW
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BU of 3fqw by Molmil
Phosphorylation of self-peptides alters Human Leukocyte Antigen Class I-restricted antigen presentation and generates tumor specific epitopes
Descriptor: Beta-2-microglobulin, CADMIUM ION, COBALT (II) ION, ...
Authors:Petersen, J, Rossjohn, J.
Deposit date:2009-01-07
Release date:2009-03-03
Last modified:2023-11-01
Method:X-RAY DIFFRACTION (1.927 Å)
Cite:Phosphorylated self-peptides alter human leukocyte antigen class I-restricted antigen presentation and generate tumor-specific epitopes
Proc.Natl.Acad.Sci.Usa, 106, 2009
3FQT
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BU of 3fqt by Molmil
Phosphorylation of self-peptides alters Human Leukocyte Antigen Class I-restricted antigen presentation and generates tumor specific epitopes
Descriptor: Beta-2-microglobulin, CADMIUM ION, GLYCEROL, ...
Authors:Petersen, J, Rossjohn, J.
Deposit date:2009-01-07
Release date:2009-03-03
Last modified:2023-11-01
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Phosphorylated self-peptides alter human leukocyte antigen class I-restricted antigen presentation and generate tumor-specific epitopes
Proc.Natl.Acad.Sci.Usa, 106, 2009
4OZH
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BU of 4ozh by Molmil
S16 protein complex
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, Gliadin-alpha2 peptide, ...
Authors:Petersen, J, Reid, H.H, Rossjohn, J.
Deposit date:2014-02-16
Release date:2014-04-16
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (2.8 Å)
Cite:T-cell receptor recognition of HLA-DQ2-gliadin complexes associated with celiac disease.
Nat.Struct.Mol.Biol., 21, 2014
4OZF
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BU of 4ozf by Molmil
JR5.1 protein complex
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, HLA class II histocompatibility antigen, DQ alpha 1 chain, ...
Authors:Petersen, J, Reid, H.H, Rossjohn, J.
Deposit date:2014-02-15
Release date:2014-04-16
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (2.7 Å)
Cite:T-cell receptor recognition of HLA-DQ2-gliadin complexes associated with celiac disease.
Nat.Struct.Mol.Biol., 21, 2014
4OZI
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BU of 4ozi by Molmil
S2 protein complex
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, HLA class II histocompatibility antigen, ...
Authors:Petersen, J, Reid, H.H, Rossjohn, J.
Deposit date:2014-02-16
Release date:2014-04-16
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (3.2 Å)
Cite:T-cell receptor recognition of HLA-DQ2-gliadin complexes associated with celiac disease.
Nat.Struct.Mol.Biol., 21, 2014
4OZG
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BU of 4ozg by Molmil
D2 protein complex
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
Authors:Petersen, J, Reid, H.H, Rossjohn, J.
Deposit date:2014-02-16
Release date:2014-04-16
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (3 Å)
Cite:T-cell receptor recognition of HLA-DQ2-gliadin complexes associated with celiac disease.
Nat.Struct.Mol.Biol., 21, 2014
6XP6
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BU of 6xp6 by Molmil
3C11-DQ2-glia-a2 complex
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 3.C11 IgH Fab, ...
Authors:Petersen, J, Rossjohn, J.
Deposit date:2020-07-08
Release date:2021-07-28
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:A high-affinity human TCR-like antibody detects celiac disease gluten peptide-MHC complexes and inhibits T cell activation.
Sci Immunol, 6, 2021
6FTN
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BU of 6ftn by Molmil
mPI3Kd IN COMPLEX WITH AZ2
Descriptor: Phosphor inositol 3 kinase, ~{N}-[5-[2-[(1~{S})-1-cyclopropylethyl]-7-methyl-1-oxidanylidene-3~{H}-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]ethanamide
Authors:Petersen, J.
Deposit date:2018-02-22
Release date:2018-06-20
Last modified:2018-07-11
Method:X-RAY DIFFRACTION (2 Å)
Cite:Discovery of Highly Isoform Selective Orally Bioavailable Phosphoinositide 3-Kinase (PI3K)-gamma Inhibitors.
J. Med. Chem., 61, 2018
8QFZ
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BU of 8qfz by Molmil
TSLP-Bicycle complex
Descriptor: 1-[3,5-bis(3-bromanylpropanoyl)-1,3,5-triazinan-1-yl]-3-bromanyl-propan-1-one, CYS-HIS-TRP-LEU-GLU-ASN-CYS-TRP-ARG-GLY-PHE-CYS, Thymic stromal lymphopoietin
Authors:Petersen, J.
Deposit date:2023-09-05
Release date:2024-02-07
Last modified:2024-02-21
Method:X-RAY DIFFRACTION (1.65 Å)
Cite:Discovery and Characterization of a Bicyclic Peptide (Bicycle) Binder to Thymic Stromal Lymphopoietin.
J.Med.Chem., 67, 2024
6GY0
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BU of 6gy0 by Molmil
mPI3Kd IN COMPLEX WITH AZ3
Descriptor: Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform, ~{N}-[4-methyl-5-(1-oxidanylidene-7-sulfamoyl-isoindol-5-yl)-1,3-thiazol-2-yl]ethanamide
Authors:Petersen, J.
Deposit date:2018-06-27
Release date:2019-02-06
Last modified:2019-04-03
Method:X-RAY DIFFRACTION (2.55 Å)
Cite:A class of highly selective inhibitors bind to an active state of PI3K gamma.
Nat.Chem.Biol., 15, 2019

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PDB entries from 2024-03-27

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