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1SNT
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BU of 1snt by Molmil
Structure of the human cytosolic sialidase Neu2
Descriptor: Sialidase 2
Authors:Chavas, L.M.G, Fusi, P, Tringali, C, Venerando, B, Tettamanti, G, Kato, R, Monti, E, Wakatsuki, S.
Deposit date:2004-03-12
Release date:2004-11-02
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (1.75 Å)
Cite:Crystal Structure of the Human Cytosolic Sialidase Neu2: EVIDENCE FOR THE DYNAMIC NATURE OF SUBSTRATE RECOGNITION
J.Biol.Chem., 280, 2005
1SO7
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BU of 1so7 by Molmil
Maltose-induced structure of the human cytolsolic sialidase Neu2
Descriptor: CHLORIDE ION, Sialidase 2
Authors:Chavas, L.M.G, Fusi, P, Tringali, C, Venerando, B, Tettamanti, G, Kato, R, Monti, E, Wakatsuki, S.
Deposit date:2004-03-12
Release date:2004-11-02
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (1.49 Å)
Cite:Crystal Structure of the Human Cytosolic Sialidase Neu2: EVIDENCE FOR THE DYNAMIC NATURE OF SUBSTRATE RECOGNITION
J.Biol.Chem., 280, 2005
1VCU
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BU of 1vcu by Molmil
Structure of the human cytosolic sialidase Neu2 in complex with the inhibitor DANA
Descriptor: 2-DEOXY-2,3-DEHYDRO-N-ACETYL-NEURAMINIC ACID, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, Sialidase 2
Authors:Chavas, L.M.G, Fusi, P, Tringali, C, Venerando, B, Tettamanti, G, Kato, R, Monti, E, Wakatsuki, S.
Deposit date:2004-03-12
Release date:2004-11-02
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.85 Å)
Cite:Crystal Structure of the Human Cytosolic Sialidase Neu2: EVIDENCE FOR THE DYNAMIC NATURE OF SUBSTRATE RECOGNITION
J.Biol.Chem., 280, 2005
2F10
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BU of 2f10 by Molmil
Crystal Structure of the Human Sialidase Neu2 in Complex with Peramivir inhibitor
Descriptor: 3-(1-ACETYLAMINO-2-ETHYL-BUTYL)-4-GUANIDINO-2-HYDROXY-CYCLOPENTANECARBOXYLIC ACID, PHOSPHATE ION, Sialidase 2
Authors:Chavas, L.M.G, Kato, R, McKimm-Breschkin, J, Colman, P.M, Fusi, P, Tringali, C, Venerando, B, Tettamanti, G, Monti, E, Wakatsuki, S.
Deposit date:2005-11-14
Release date:2006-11-21
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.9 Å)
Cite:Crystal Structure of the Human Sialidase Neu2 in Complex with Peramivir inhibitor
To be Published
2F13
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BU of 2f13 by Molmil
Crystal Structure of the Human Sialidase Neu2 in Complex with 2',3'- dihydroxypropyl ether mimetic Inhibitor
Descriptor: (2R)-2,3-dihydroxypropyl 2-acetamido-2,4-dideoxy-alpha-L-threo-hex-4-enopyranosiduronic acid, PHOSPHATE ION, Sialidase 2
Authors:Chavas, L.M.G, Kato, R, Mann, M.C, Thomson, R.J, Dyason, J.C, von Itzstein, M, Fusi, P, Tringali, C, Venerando, B, Tettamanti, G, Monti, E, Wakatsuki, S.
Deposit date:2005-11-14
Release date:2006-11-21
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.26 Å)
Cite:Crystal Structure of the Human Sialidase Neu2 in Complex with 2',3'- dihydroxypropyl ether mimetic Inhibitor
To be Published
2F11
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BU of 2f11 by Molmil
Crystal Structure of the Human Sialidase Neu2 in Complex with isobutyl ether mimetic Inhibitor
Descriptor: 2-methylpropyl 2-acetamido-2,4-dideoxy-alpha-L-threo-hex-4-enopyranosiduronic acid, PHOSPHATE ION, Sialidase 2
Authors:Chavas, L.M.G, Kato, R, Mann, M.C, Thomson, R.J, Dyason, J.C, von Itzstein, M, Fusi, P, Tringali, C, Venerando, B, Tettamanti, G, Monti, E, Wakatsuki, S.
Deposit date:2005-11-14
Release date:2006-11-21
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.57 Å)
Cite:Crystal Structure of the Human Sialidase Neu2 in Complex with isobutyl ether mimetic Inhibitor
To be Published
2F26
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BU of 2f26 by Molmil
Crystal Structure of the Human Sialidase Neu2 E111Q-Q112E Double Mutant
Descriptor: CHLORIDE ION, Sialidase 2
Authors:Chavas, L.M.G, Kato, R, Fusi, P, Tringali, C, Venerando, B, Tettamanti, G, Monti, E, Wakatsuki, S.
Deposit date:2005-11-15
Release date:2006-11-21
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (1.58 Å)
Cite:Crystal Structure of the Human Sialidase Neu2 E111Q-Q112E Double Mutant
To be Published
2F0Z
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BU of 2f0z by Molmil
Crystal Structure of the Human Sialidase Neu2 in Complex with Zanamivir inhibitor
Descriptor: Sialidase 2, ZANAMIVIR
Authors:Chavas, L.M.G, Kato, R, McKimm-Breschkin, J, Colman, P.M, Fusi, P, Tringali, C, Venerando, B, Tettamanti, G, Monti, E, Wakatsuki, S.
Deposit date:2005-11-14
Release date:2006-11-21
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.8 Å)
Cite:Crystal Structure of the Human Sialidase Neu2 in Complex with Zanamivir inhibitor
To be Published
2F25
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BU of 2f25 by Molmil
Crystal Structure of the Human Sialidase Neu2 E111Q Mutant in Complex with DANA Inhibitor
Descriptor: 2-DEOXY-2,3-DEHYDRO-N-ACETYL-NEURAMINIC ACID, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, Sialidase 2
Authors:Chavas, L.M.G, Kato, R, Fusi, P, Tringali, C, Venerando, B, Tettamanti, G, Monti, E, Wakatsuki, S.
Deposit date:2005-11-15
Release date:2006-11-21
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (1.95 Å)
Cite:Crystal Structure of the Human Sialidase Neu2 E111Q Mutant in Complex with DANA Inhibitor
To be Published
2F24
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BU of 2f24 by Molmil
Crystal Structure of the Human Sialidase Neu2 E111Q Mutant
Descriptor: CHLORIDE ION, Sialidase 2
Authors:Chavas, L.M.G, Kato, R, Fusi, P, Tringali, C, Venerando, B, Tettamanti, G, Monti, E, Wakatsuki, S.
Deposit date:2005-11-15
Release date:2006-11-21
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (1.76 Å)
Cite:Crystal Structure of the Human Sialidase Neu2 E111Q Mutant
To be Published
2F29
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BU of 2f29 by Molmil
Crystal Structure of the Human Sialidase Neu2 Q116E Mutant in Complex with DANA Inhibitor
Descriptor: 2-DEOXY-2,3-DEHYDRO-N-ACETYL-NEURAMINIC ACID, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, Sialidase 2
Authors:Chavas, L.M.G, Kato, R, Fusi, P, Tringali, C, Venerando, B, Tettamanti, G, Monti, E, Wakatsuki, S.
Deposit date:2005-11-15
Release date:2006-11-21
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.921 Å)
Cite:Crystal Structure of the Human Sialidase Neu2 Q116E Mutant in Complex with DANA Inhibitor
To be Published
2F12
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BU of 2f12 by Molmil
Crystal Structure of the Human Sialidase Neu2 in Complex with 3- hydroxypropyl ether mimetic Inhibitor
Descriptor: 3-hydroxypropyl 2-acetamido-2,4-dideoxy-alpha-L-threo-hex-4-enopyranosiduronic acid, PHOSPHATE ION, Sialidase 2
Authors:Chavas, L.M.G, Kato, R, Mann, M.C, Thomson, R.J, Dyason, J.C, von Itzstein, M, Fusi, P, Tringali, C, Venerando, B, Tettamanti, G, Monti, E, Wakatsuki, S.
Deposit date:2005-11-14
Release date:2006-11-21
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.27 Å)
Cite:Crystal Structure of the Human Sialidase Neu2 in Complex with 3- hydroxypropyl ether mimetic Inhibitor
To be Published
2F28
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BU of 2f28 by Molmil
Crystal Structure of the Human Sialidase Neu2 Q116E Mutant
Descriptor: CHLORIDE ION, Sialidase 2
Authors:Chavas, L.M.G, Kato, R, Fusi, P, Tringali, C, Venerando, B, Tettamanti, G, Monti, E, Wakatsuki, S.
Deposit date:2005-11-15
Release date:2006-11-21
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (1.67 Å)
Cite:Crystal Structure of the Human Sialidase Neu2 Q116E Mutant
To be Published
2F27
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Crystal Structure of the Human Sialidase Neu2 E111Q-Q112E Double Mutant in Complex with DANA Inhibitor
Descriptor: 2-DEOXY-2,3-DEHYDRO-N-ACETYL-NEURAMINIC ACID, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, Sialidase 2
Authors:Chavas, L.M.G, Kato, R, Fusi, P, Tringali, C, Venerando, B, Tettamanti, G, Monti, E, Wakatsuki, S.
Deposit date:2005-11-15
Release date:2006-11-21
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.15 Å)
Cite:Crystal Structure of the Human Sialidase Neu2 E111Q-Q112E Double Mutant in Complex with DANA Inhibitor
To be Published

217705

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