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2WPO
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BU of 2wpo by Molmil
HCMV protease inhibitor complex
Descriptor: (2S)-2-(3,3-dimethylbutanoylamino)-N-[(2S)-1-[[(2S,3S)-3-hydroxy-4-[(4-iodophenyl)methylamino]-4-oxo-butan-2-yl]amino]- 1,4-dioxo-4-pyrrol-1-yl-butan-2-yl]-3,3-dimethyl-butanamide, HUMAN CYTOMEGALOVIRUS PROTEASE
Authors:Tong, L, Qian, C, Massariol, M.-J, Deziel, R, Yoakim, C, Lagace, L.
Deposit date:1998-08-04
Release date:1999-08-04
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (2.7 Å)
Cite:Conserved mode of peptidomimetic inhibition and substrate recognition of human cytomegalovirus protease.
Nat.Struct.Biol., 5, 1998
1BFZ
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BU of 1bfz by Molmil
BOUND CONFORMATION OF N-TERMINAL CLEAVAGE PRODUCT PEPTIDE MIMIC (P1-P9 OF RELEASE SITE) WHILE BOUND TO HCMV PROTEASE AS DETERMINED BY TRANSFERRED NOESY EXPERIMENTS (P1-P5 SHOWN ONLY), NMR, 32 STRUCTURES
Descriptor: HCMV PROTEASE R-SITE N-TERMINAL CLEAVAGE PRODUCT
Authors:Laplante, S.R, Aubry, N, Bonneau, P.R, Cameron, D.R, Lagace, L, Massariol, M.-J, Montpetit, H, Ploufe, C, Kawai, S.H, Fulton, B.D, Chen, Z, Ni, F.
Deposit date:1998-05-25
Release date:1999-05-25
Last modified:2011-07-13
Method:SOLUTION NMR
Cite:Human cytomegalovirus protease complexes its substrate recognition sequences in an extended peptide conformation.
Biochemistry, 37, 1998
1ID4
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BU of 1id4 by Molmil
CRYSTAL STRUCTURE OF THE CATALYTIC SITE MUTANT (H157Q) OF THE HUMAN CYTOMEGALOVIRUS PROTEASE
Descriptor: CAPSID PROTEIN P40: ASSEMBLIN PROTEASE
Authors:Khayat, R, Batra, R, Massariol, M.J, Lagace, L, Tong, L.
Deposit date:2001-04-03
Release date:2001-06-06
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Investigating the role of histidine 157 in the catalytic activity of human cytomegalovirus protease.
Biochemistry, 40, 2001
1IEC
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BU of 1iec by Molmil
CRYSTAL STRUCTURE OF THE CATALYTIC SITE MUTANT (H157A) OF THE HUMAN CYTOMEGALOVIRUS PROTEASE
Descriptor: CAPSID PROTEIN P40: ASSEMBLIN PROTEASE
Authors:Khayat, R, Batra, R, Massariol, M.J, Lagace, L, Tong, L.
Deposit date:2001-04-09
Release date:2001-06-06
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Investigating the role of histidine 157 in the catalytic activity of human cytomegalovirus protease.
Biochemistry, 40, 2001
1IEG
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BU of 1ieg by Molmil
CRYSTAL STRUCTURE OF THE CATALYTIC SITE MUTANT S134A/H157A OF THE HUMAN CYTOMEGALOVIRUS PROTEASE
Descriptor: CAPSID PROTEIN P40: ASSEMBLIN PROTEASE
Authors:Khayat, R, Batra, R, Massariol, M.J, Lagace, L, Tong, L.
Deposit date:2001-04-09
Release date:2001-06-06
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (2 Å)
Cite:Investigating the role of histidine 157 in the catalytic activity of human cytomegalovirus protease.
Biochemistry, 40, 2001
1IEF
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BU of 1ief by Molmil
CRYSTAL STRUCTURE OF THE CATALYTIC SITE MUTANT S134A OF THE HUMAN CYTOMEGALOVIRUS PROTEASE
Descriptor: CAPSID PROTEIN P40: ASSEMBLIN PROTEASE
Authors:Khayat, R, Batra, R, Massariol, M.J, Lagace, L, Tong, L.
Deposit date:2001-04-09
Release date:2001-06-06
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Investigating the role of histidine 157 in the catalytic activity of human cytomegalovirus protease.
Biochemistry, 40, 2001
1IED
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BU of 1ied by Molmil
CRYSTAL STRUCTURE OF THE CATALYTIC SITE MUTANT (H157E) OF THE HUMAN CYTOMEGALOVIRUS PROTEASE
Descriptor: CAPSID PROTEIN P40: ASSEMBLIN PROTEASE
Authors:Khayat, R, Batra, R, Massariol, M.J, Lagace, L, Tong, L.
Deposit date:2001-04-09
Release date:2001-06-06
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (2 Å)
Cite:Investigating the role of histidine 157 in the catalytic activity of human cytomegalovirus protease.
Biochemistry, 40, 2001
1WPO
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BU of 1wpo by Molmil
HYDROLYTIC ENZYME HUMAN CYTOMEGALOVIRUS PROTEASE
Descriptor: HUMAN CYTOMEGALOVIRUS PROTEASE, SULFATE ION
Authors:Tong, L.
Deposit date:1996-07-23
Release date:1997-10-15
Last modified:2021-11-03
Method:X-RAY DIFFRACTION (2 Å)
Cite:A new serine-protease fold revealed by the crystal structure of human cytomegalovirus protease.
Nature, 383, 1996
4I32
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BU of 4i32 by Molmil
Crystal structure of HCV NS3/4A D168V protease complexed with compound 4
Descriptor: (2R,6S,7E,10E,13aR,14aR,16aS)-2-{[7-methoxy-8-methyl-2-(propan-2-yloxy)quinolin-4-yl]oxy}-N-[(1-methylcyclopropyl)sulfonyl]-6-{[(1-methyl-1H-pyrazol-3-yl)carbonyl]amino}-5,16-dioxo-1,2,3,6,9,12,13,13a,14,15,16,16a-dodecahydrocyclopropa[e]pyrrolo[1,2-a][1,4]diazacyclopentadecine-14a(5H)-carboxamide, Genome polyprotein, HCV non-structural protein 4A, ...
Authors:Lemke, C.T.
Deposit date:2012-11-23
Release date:2013-01-02
Last modified:2013-03-13
Method:X-RAY DIFFRACTION (2.3001 Å)
Cite:Molecular Mechanism by Which a Potent Hepatitis C Virus NS3-NS4A Protease Inhibitor Overcomes Emergence of Resistance.
J.Biol.Chem., 288, 2013
4I33
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BU of 4i33 by Molmil
Crystal structure of HCV NS3/4A R155K protease complexed with compound 4
Descriptor: (2R,6S,7E,10E,13aR,14aR,16aS)-2-{[7-methoxy-8-methyl-2-(propan-2-yloxy)quinolin-4-yl]oxy}-N-[(1-methylcyclopropyl)sulfonyl]-6-{[(1-methyl-1H-pyrazol-3-yl)carbonyl]amino}-5,16-dioxo-1,2,3,6,9,12,13,13a,14,15,16,16a-dodecahydrocyclopropa[e]pyrrolo[1,2-a][1,4]diazacyclopentadecine-14a(5H)-carboxamide, Genome polyprotein, HCV non-structural protein 4A, ...
Authors:Lemke, C.T.
Deposit date:2012-11-23
Release date:2013-01-02
Last modified:2013-03-13
Method:X-RAY DIFFRACTION (1.9001 Å)
Cite:Molecular Mechanism by Which a Potent Hepatitis C Virus NS3-NS4A Protease Inhibitor Overcomes Emergence of Resistance.
J.Biol.Chem., 288, 2013
4I31
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BU of 4i31 by Molmil
Crystal structure of HCV NS3/NS4A protease complexed with compound 4
Descriptor: (2R,6S,7E,10E,13aR,14aR,16aS)-2-{[7-methoxy-8-methyl-2-(propan-2-yloxy)quinolin-4-yl]oxy}-N-[(1-methylcyclopropyl)sulfonyl]-6-{[(1-methyl-1H-pyrazol-3-yl)carbonyl]amino}-5,16-dioxo-1,2,3,6,9,12,13,13a,14,15,16,16a-dodecahydrocyclopropa[e]pyrrolo[1,2-a][1,4]diazacyclopentadecine-14a(5H)-carboxamide, Genome polyprotein, HCV non-structural protein 4A, ...
Authors:Lemke, C.T.
Deposit date:2012-11-23
Release date:2013-01-02
Last modified:2013-03-13
Method:X-RAY DIFFRACTION (1.9301 Å)
Cite:Molecular Mechanism by Which a Potent Hepatitis C Virus NS3-NS4A Protease Inhibitor Overcomes Emergence of Resistance.
J.Biol.Chem., 288, 2013
3CLN
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BU of 3cln by Molmil
STRUCTURE OF CALMODULIN REFINED AT 2.2 ANGSTROMS RESOLUTION
Descriptor: CALCIUM ION, CALMODULIN
Authors:Babu, Y.S, Bugg, C.E, Cook, W.J.
Deposit date:1988-05-11
Release date:1988-07-16
Last modified:2024-02-21
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Structure of calmodulin refined at 2.2 A resolution.
J.Mol.Biol., 204, 1988

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