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1BV8
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BU of 1bv8 by Molmil
RECEPTOR DOMAIN FROM ALPHA-2-MACROGLOBULIN
Descriptor: ALPHA-2-MACROGLOBULIN
Authors:Huang, W, Dolmer, K, Liao, X, Gettins, P.G.W.
Deposit date:1998-09-22
Release date:2000-04-05
Last modified:2022-02-16
Method:SOLUTION NMR
Cite:NMR solution structure of complement-like repeat CR8 from the low density lipoprotein receptor-related protein.
J.Biol.Chem., 274, 1999
1AHJ
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BU of 1ahj by Molmil
NITRILE HYDRATASE
Descriptor: FE (III) ION, NITRILE HYDRATASE (SUBUNIT ALPHA), NITRILE HYDRATASE (SUBUNIT BETA)
Authors:Huang, W, Schneider, G, Lindqvist, Y.
Deposit date:1997-04-05
Release date:1998-04-08
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (2.65 Å)
Cite:Crystal structure of nitrile hydratase reveals a novel iron centre in a novel fold.
Structure, 5, 1997
1DAD
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BU of 1dad by Molmil
DETHIOBIOTIN SYNTHETASE COMPLEXED WITH ADP
Descriptor: ADENOSINE-5'-DIPHOSPHATE, DETHIOBIOTIN SYNTHETASE
Authors:Huang, W, Jia, J, Schneider, G, Lindqvist, Y.
Deposit date:1995-05-08
Release date:1996-06-20
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (1.6 Å)
Cite:Mechanism of an ATP-dependent carboxylase, dethiobiotin synthetase, based on crystallographic studies of complexes with substrates and a reaction intermediate.
Biochemistry, 34, 1995
8CWL
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BU of 8cwl by Molmil
Cryo-EM structure of Human 15-PGDH in complex with small molecule SW222746
Descriptor: 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, 15-hydroxyprostaglandin dehydrogenase [NAD(+)], 2-methyl-6-[7-(piperidine-1-carbonyl)quinoxalin-2-yl]isoquinolin-1(2H)-one
Authors:Huang, W, Taylor, D.J.
Deposit date:2022-05-19
Release date:2023-03-08
Method:ELECTRON MICROSCOPY (2.9 Å)
Cite:Small molecule inhibitors of 15-PGDH exploit a physiologic induced-fit closing system.
Nat Commun, 14, 2023
8CVN
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BU of 8cvn by Molmil
Cryo-EM Structure of Human 15-PGDH in Complex with Small Molecule SW209415
Descriptor: 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, 15-hydroxyprostaglandin dehydrogenase [NAD(+)], 2-[butyl(oxidanyl)-$l^{3}-sulfanyl]-4-(2,3-dimethylimidazol-4-yl)-6-(1,3-thiazol-2-yl)thieno[2,3-b]pyridin-3-amine
Authors:Huang, W, Taylor, D.J.
Deposit date:2022-05-18
Release date:2023-03-01
Last modified:2023-03-29
Method:ELECTRON MICROSCOPY (2.4 Å)
Cite:Small molecule inhibitors of 15-PGDH exploit a physiologic induced-fit closing system.
Nat Commun, 14, 2023
1DAG
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BU of 1dag by Molmil
DETHIOBIOTIN SYNTHETASE COMPLEXED WITH 7-(CARBOXYAMINO)-8-AMINO-NONANOIC ACID AND 5'-ADENOSYL-METHYLENE-TRIPHOSPHATE
Descriptor: 7-(CARBOXYAMINO)-8-AMINO-NONANOIC ACID, DETHIOBIOTIN SYNTHETASE, PHOSPHOMETHYLPHOSPHONIC ACID ADENYLATE ESTER
Authors:Huang, W, Jia, J, Schneider, G, Lindqvist, Y.
Deposit date:1995-05-08
Release date:1996-06-20
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (1.64 Å)
Cite:Mechanism of an ATP-dependent carboxylase, dethiobiotin synthetase, based on crystallographic studies of complexes with substrates and a reaction intermediate.
Biochemistry, 34, 1995
1DAE
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BU of 1dae by Molmil
DETHIOBIOTIN SYNTHETASE COMPLEXED WITH 3-(1-AMINOETHYL) NONANEDIOIC ACID
Descriptor: 3-(1-AMINOETHYL)NONANEDIOIC ACID, DETHIOBIOTIN SYNTHETASE
Authors:Huang, W, Jia, J, Schneider, G, Lindqvist, Y.
Deposit date:1995-05-08
Release date:1996-06-20
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (1.7 Å)
Cite:Mechanism of an ATP-dependent carboxylase, dethiobiotin synthetase, based on crystallographic studies of complexes with substrates and a reaction intermediate.
Biochemistry, 34, 1995
1DAH
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BU of 1dah by Molmil
DETHIOBIOTIN SYNTHETASE COMPLEXED WITH 7,8-DIAMINO-NONANOIC ACID, 5'-ADENOSYL-METHYLENE-TRIPHOSPHATE, AND MANGANESE
Descriptor: 7,8-DIAMINO-NONANOIC ACID, DETHIOBIOTIN SYNTHETASE, MANGANESE (II) ION, ...
Authors:Huang, W, Jia, J, Schneider, G, Lindqvist, Y.
Deposit date:1995-05-08
Release date:1996-06-20
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (1.64 Å)
Cite:Mechanism of an ATP-dependent carboxylase, dethiobiotin synthetase, based on crystallographic studies of complexes with substrates and a reaction intermediate.
Biochemistry, 34, 1995
1DAI
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BU of 1dai by Molmil
DETHIOBIOTIN SYNTHETASE COMPLEXED WITH 7-(CARBOXYAMINO)-8-AMINO-NONANOIC ACID
Descriptor: 7-(CARBOXYAMINO)-8-AMINO-NONANOIC ACID, DETHIOBIOTIN SYNTHETASE
Authors:Huang, W, Jia, J, Schneider, G, Lindqvist, Y.
Deposit date:1995-05-08
Release date:1996-06-20
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (1.64 Å)
Cite:Mechanism of an ATP-dependent carboxylase, dethiobiotin synthetase, based on crystallographic studies of complexes with substrates and a reaction intermediate.
Biochemistry, 34, 1995
1DAF
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BU of 1daf by Molmil
DETHIOBIOTIN SYNTHETASE COMPLEXED WITH 7-(CARBOXYAMINO)-8-AMINO-NONANOIC ACID, ADP, AND CALCIUM
Descriptor: 7-(CARBOXYAMINO)-8-AMINO-NONANOIC ACID, ADENOSINE-5'-DIPHOSPHATE, CALCIUM ION, ...
Authors:Huang, W, Jia, J, Schneider, G, Lindqvist, Y.
Deposit date:1995-05-08
Release date:1996-06-20
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (1.7 Å)
Cite:Mechanism of an ATP-dependent carboxylase, dethiobiotin synthetase, based on crystallographic studies of complexes with substrates and a reaction intermediate.
Biochemistry, 34, 1995
8WRJ
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BU of 8wrj by Molmil
glycosyltransferase UGT74AN3
Descriptor: 5-[(1R,2S,4R,6R,7R,10S,11S,14S,16R)-14-hydroxy-7,11-dimethyl-3-oxapentacyclo[8.8.0.02,4.02,7.011,16]octadecan-6-yl]pyran-2-one, Glycosyltransferase, URIDINE-5'-DIPHOSPHATE
Authors:Huang, W, Long, F.
Deposit date:2023-10-15
Release date:2024-01-24
Method:X-RAY DIFFRACTION (1.85 Å)
Cite:Substrate Promiscuity, Crystal Structure, and Application of a Plant UDP-Glycosyltransferase UGT74AN3
Acs Catalysis, 14, 2024
8WRK
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BU of 8wrk by Molmil
glycosyltransferase UGT74AN3
Descriptor: Glycosyltransferase, PICEATANNOL, URIDINE-5'-DIPHOSPHATE
Authors:Huang, W, Long, F.
Deposit date:2023-10-15
Release date:2024-01-24
Method:X-RAY DIFFRACTION (2.03 Å)
Cite:Substrate Promiscuity, Crystal Structure, and Application of a Plant UDP-Glycosyltransferase UGT74AN3
Acs Catalysis, 14, 2024
1CR8
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BU of 1cr8 by Molmil
LOW DENSITY LIPOPROTEIN RECEPTOR-RELATED PROTEIN COMPLEMENT REPEAT 8
Descriptor: CALCIUM ION, PROTEIN (LOW DENSITY LIPOPROTEIN RECEPTOR RELATED PROTEIN)
Authors:Huang, W, Dolmer, K, Gettins, P.G.W.
Deposit date:1998-12-14
Release date:1998-12-23
Last modified:2023-12-27
Method:SOLUTION NMR
Cite:NMR solution structure of complement-like repeat CR8 from the low density lipoprotein receptor-related protein.
J.Biol.Chem., 274, 1999
1DBO
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BU of 1dbo by Molmil
CRYSTAL STRUCTURE OF CHONDROITINASE B
Descriptor: 4-deoxy-alpha-D-glucopyranose-(1-3)-[beta-D-glucopyranose-(1-4)]2-O-methyl-beta-L-fucopyranose-(1-4)-beta-D-xylopyranose-(1-4)-alpha-D-glucopyranuronic acid-(1-2)-[alpha-L-rhamnopyranose-(1-4)]alpha-D-mannopyranose, 4-deoxy-beta-D-glucopyranuronic acid-(1-3)-2-acetamido-2-deoxy-4-O-sulfo-beta-D-galactopyranose, CHONDROITINASE B
Authors:Huang, W, Matte, A, Li, Y, Kim, Y.S, Linhardt, R.J, Su, H, Cygler, M.
Deposit date:1999-11-03
Release date:2000-01-12
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (1.7 Å)
Cite:Crystal structure of chondroitinase B from Flavobacterium heparinum and its complex with a disaccharide product at 1.7 A resolution.
J.Mol.Biol., 294, 1999
1DBG
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BU of 1dbg by Molmil
CRYSTAL STRUCTURE OF CHONDROITINASE B
Descriptor: 4-deoxy-alpha-D-glucopyranose-(1-3)-[beta-D-glucopyranose-(1-4)]2-O-methyl-beta-L-fucopyranose-(1-4)-beta-D-xylopyranose-(1-4)-alpha-D-glucopyranuronic acid-(1-2)-[alpha-L-rhamnopyranose-(1-4)]alpha-D-mannopyranose, CHONDROITINASE B
Authors:Huang, W, Matte, A, Li, Y, Kim, Y.S, Linhardt, R.J, Su, H, Cygler, M.
Deposit date:1999-11-02
Release date:2000-01-12
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (1.7 Å)
Cite:Crystal structure of chondroitinase B from Flavobacterium heparinum and its complex with a disaccharide product at 1.7 A resolution.
J.Mol.Biol., 294, 1999
1DTS
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BU of 1dts by Molmil
CRYSTAL STRUCTURE OF AN ATP DEPENDENT CARBOXYLASE, DETHIOBIOTIN SYNTHASE, AT 1.65 ANGSTROMS RESOLUTION
Descriptor: DETHIOBIOTIN SYNTHETASE
Authors:Huang, W, Lindqvist, Y, Schneider, G.
Deposit date:1995-03-28
Release date:1995-04-20
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (1.65 Å)
Cite:Crystal structure of an ATP-dependent carboxylase, dethiobiotin synthetase, at 1.65 A resolution.
Structure, 2, 1994
1HN0
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BU of 1hn0 by Molmil
CRYSTAL STRUCTURE OF CHONDROITIN ABC LYASE I FROM PROTEUS VULGARIS AT 1.9 ANGSTROMS RESOLUTION
Descriptor: CHONDROITIN ABC LYASE I, SODIUM ION
Authors:Huang, W, Cygler, M.
Deposit date:2000-12-05
Release date:2003-04-08
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Crystal Structure of Proteus vulgaris Chondroitin Sulfate ABC Lyase I at 1.9 Angstroms Resolution
J.Mol.Biol., 328, 2003
1HMU
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BU of 1hmu by Molmil
ACTIVE SITE OF CHONDROITINASE AC LYASE REVEALED BY THE STRUCTURE OF ENZYME-OLIGOSACCHARIDE COMPLEXES AND MUTAGENESIS
Descriptor: 2-O-methyl-beta-L-fucopyranose-(1-4)-beta-D-xylopyranose-(1-4)-alpha-D-glucopyranuronic acid-(1-2)-[alpha-L-rhamnopyranose-(1-4)]alpha-D-mannopyranose, 4-deoxy-alpha-L-threo-hex-4-enopyranuronic acid-(1-3)-2-acetamido-2-deoxy-4-O-sulfo-beta-D-galactopyranose, CALCIUM ION, ...
Authors:Huang, W, Boju, L, Tkalec, L, Su, H, Yang, H.O, Gunay, N.S, Linhardt, R.J, Kim, Y.S, Matte, A, Cygler, M.
Deposit date:2000-12-05
Release date:2001-05-02
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (2 Å)
Cite:Active site of chondroitin AC lyase revealed by the structure of enzyme-oligosaccharide complexes and mutagenesis.
Biochemistry, 40, 2001
1HMW
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BU of 1hmw by Molmil
ACTIVE SITE OF CHONDROITINASE AC LYASE REVEALED BY THE STRUCTURE OF ENZYME-OLIGOSACCHARIDE COMPLEXES AND MUTAGENESIS
Descriptor: 2-O-methyl-beta-L-fucopyranose-(1-4)-beta-D-xylopyranose-(1-4)-alpha-D-glucopyranuronic acid-(1-2)-[alpha-L-rhamnopyranose-(1-4)]alpha-D-mannopyranose, 4-deoxy-alpha-L-threo-hex-4-enopyranuronic acid-(1-3)-2-acetamido-2-deoxy-4-O-sulfo-beta-D-galactopyranose-(1-4)-beta-D-glucopyranuronic acid-(1-3)-2-acetamido-2-deoxy-6-O-sulfo-beta-D-galactopyranose, CALCIUM ION, ...
Authors:Huang, W, Boju, L, Tkalec, L, Su, H, Yang, H.O, Gunay, N.S, Linhardt, R.J, Kim, Y.S, Matte, A, Cygler, M.
Deposit date:2000-12-05
Release date:2001-05-02
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Active site of chondroitin AC lyase revealed by the structure of enzyme-oligosaccharide complexes and mutagenesis.
Biochemistry, 40, 2001
1HM3
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BU of 1hm3 by Molmil
ACTIVE SITE OF CHONDROITINASE AC LYASE REVEALED BY THE STRUCTURE OF ENZYME-OLIGOSACCHARIDE COMPLEXES AND MUTAGENESIS
Descriptor: 2-O-methyl-beta-L-fucopyranose-(1-4)-beta-D-xylopyranose-(1-4)-alpha-D-glucopyranuronic acid-(1-2)-[alpha-L-rhamnopyranose-(1-4)]alpha-D-mannopyranose, CALCIUM ION, CHONDROITINASE AC, ...
Authors:Huang, W, Boju, L, Tkalec, L, Su, H, Yang, H.O, Gunay, N.S, Linhardt, R.J, Kim, Y.S, Matte, A, Cygler, M.
Deposit date:2000-12-04
Release date:2001-05-02
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:Active site of chondroitin AC lyase revealed by the structure of enzyme-oligosaccharide complexes and mutagenesis.
Biochemistry, 40, 2001
1HM2
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BU of 1hm2 by Molmil
ACTIVE SITE OF CHONDROITINASE AC LYASE REVEALED BY THE STRUCTURE OF ENZYME-OLIGOSACCHARIDE COMPLEXES AND MUTAGENESIS
Descriptor: 2-O-methyl-beta-L-fucopyranose-(1-4)-beta-D-xylopyranose-(1-4)-alpha-D-glucopyranuronic acid-(1-2)-[alpha-L-rhamnopyranose-(1-4)]alpha-D-mannopyranose, CALCIUM ION, CHONDROITINASE AC, ...
Authors:Huang, W, Boju, L, Tkalec, L, Su, H, Yang, H.O, Gunay, N.S, Linhardt, R.J, Kim, Y.S, Matte, A, Cygler, M.
Deposit date:2000-12-04
Release date:2001-05-02
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (2 Å)
Cite:Active site of chondroitin AC lyase revealed by the structure of enzyme-oligosaccharide complexes and mutagenesis.
Biochemistry, 40, 2001
1KAS
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BU of 1kas by Molmil
BETA-KETOACYL-ACP SYNTHASE II FROM ESCHERICHIA COLI
Descriptor: BETA-KETOACYL ACP SYNTHASE II
Authors:Huang, W, Jia, J, Edwards, P, Dehesh, K, Schneider, G, Lindqvist, Y.
Deposit date:1997-12-22
Release date:1999-03-02
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:Crystal structure of beta-ketoacyl-acyl carrier protein synthase II from E.coli reveals the molecular architecture of condensing enzymes.
EMBO J., 17, 1998
8FD8
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BU of 8fd8 by Molmil
human 15-PGDH with NADH bound
Descriptor: 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, 15-hydroxyprostaglandin dehydrogenase [NAD(+)]
Authors:Huang, W, Taylor, D.
Deposit date:2022-12-02
Release date:2023-03-08
Method:ELECTRON MICROSCOPY (3.3 Å)
Cite:Small molecule inhibitors of 15-PGDH exploit a physiologic induced-fit closing system.
Nat Commun, 14, 2023
2RG3
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BU of 2rg3 by Molmil
Covalent complex structure of elastase
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, Leukocyte elastase
Authors:Huang, W, Yamamoto, Y.
Deposit date:2007-10-02
Release date:2008-07-01
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:X-ray snapshot of the mechanism of inactivation of human neutrophil elastase by 1,2,5-thiadiazolidin-3-one 1,1-dioxide derivatives.
J.Med.Chem., 51, 2008
8H4J
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BU of 8h4j by Molmil
Crystal Structure of AzoR-FMN-Lyb24 complex
Descriptor: FLAVIN MONONUCLEOTIDE, FMN dependent NADH:quinone oxidoreductase, ~{N}-(3-methylsulfanylphenyl)-4~{H}-cyclopenta[b]quinolin-9-amine
Authors:Huang, W.
Deposit date:2022-10-10
Release date:2023-10-18
Method:X-RAY DIFFRACTION (2 Å)
Cite:Crystal Structure of AzoR-FMN-Lyb24 complex
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