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8FZ5
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BU of 8fz5 by Molmil
The PI31-free Bovine 20S proteasome
Descriptor: Proteasome subunit alpha type-1, Proteasome subunit alpha type-2, Proteasome subunit alpha type-3, ...
Authors:Hsu, H.-C, Li, H.
Deposit date:2023-01-27
Release date:2023-07-05
Method:ELECTRON MICROSCOPY (2.23 Å)
Cite:Eta igh-resolution structure of mammalian PI31-20S proteasome complex reveals mechanism of proteasome inhibition.
J.Biol.Chem., 299, 2023
8FZ6
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BU of 8fz6 by Molmil
The human PI31 complexed with bovine 20S proteasome
Descriptor: Proteasome inhibitor PI31 subunit, Proteasome subunit alpha type-1, Proteasome subunit alpha type-2, ...
Authors:Hsu, H.-C, Li, H.
Deposit date:2023-01-27
Release date:2023-07-05
Method:ELECTRON MICROSCOPY (2.54 Å)
Cite:Eta igh-resolution structure of mammalian PI31-20S proteasome complex reveals mechanism of proteasome inhibition.
J.Biol.Chem., 299, 2023
8G6E
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BU of 8g6e by Molmil
Structure of the Plasmodium falciparum 20S proteasome complexed with inhibitor TDI-8304
Descriptor: (7S,10S,13S)-N-cyclopentyl-10-[2-(morpholin-4-yl)ethyl]-9,12-dioxo-13-(2-oxopyrrolidin-1-yl)-2-oxa-8,11-diazabicyclo[13.3.1]nonadeca-1(19),15,17-triene-7-carboxamide, Proteasome subunit alpha type, Proteasome subunit alpha type-1, ...
Authors:Hsu, H.-C, Li, H.
Deposit date:2023-02-15
Release date:2023-12-20
Last modified:2024-01-03
Method:ELECTRON MICROSCOPY (2.18 Å)
Cite:Structures revealing mechanisms of resistance and collateral sensitivity of Plasmodium falciparum to proteasome inhibitors.
Nat Commun, 14, 2023
8G6F
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BU of 8g6f by Molmil
Structure of the Plasmodium falciparum 20S proteasome beta-6 A117D mutant complexed with inhibitor WLW-vs
Descriptor: (2S)-N-[(E,2S)-1-(1H-indol-3-yl)-4-methylsulfonyl-but-3-en-2-yl]-2-[[(2S)-3-(1H-indol-3-yl)-2-(2-morpholin-4-ylethanoylamino)propanoyl]amino]-4-methyl-pentanamide, Proteasome endopeptidase complex, Proteasome subunit alpha type-1, ...
Authors:Hsu, H.-C, Li, H.
Deposit date:2023-02-15
Release date:2023-12-20
Last modified:2024-01-03
Method:ELECTRON MICROSCOPY (2.58 Å)
Cite:Structures revealing mechanisms of resistance and collateral sensitivity of Plasmodium falciparum to proteasome inhibitors.
Nat Commun, 14, 2023
8SXF
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BU of 8sxf by Molmil
The C-terminal protease CtpA-LbcA complex of pseudomonas aeruginosa with the TPR at the high position
Descriptor: Probable carboxyl-terminal protease, TPR repeat-containing protein PA4667, polyA
Authors:Hsu, H.-C, Li, H.
Deposit date:2023-05-22
Release date:2024-03-06
Last modified:2024-03-27
Method:ELECTRON MICROSCOPY (3.92 Å)
Cite:P. aeruginosa CtpA protease adopts a novel activation mechanism to initiate the proteolytic process.
Embo J., 2024
8SXG
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BU of 8sxg by Molmil
The C-terminal protease CtpA-LbcA complex of pseudomonas aeruginosa with the TPR at the low position
Descriptor: Probable carboxyl-terminal protease, TPR repeat-containing protein PA4667, unidentified peptide
Authors:Hsu, H.-C, Li, H.
Deposit date:2023-05-22
Release date:2024-03-06
Last modified:2024-03-27
Method:ELECTRON MICROSCOPY (4.14 Å)
Cite:P. aeruginosa CtpA protease adopts a novel activation mechanism to initiate the proteolytic process.
Embo J., 2024
8SXH
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BU of 8sxh by Molmil
Structure of the C-terminal protease CtpA-LbcA complex of Pseudomonas aeruginosa
Descriptor: Carboxyl-terminal protease, TPR repeat-containing protein PA4667, unidentified peptide
Authors:Hsu, H.-C, Li, H.
Deposit date:2023-05-22
Release date:2024-03-06
Last modified:2024-03-27
Method:ELECTRON MICROSCOPY (3.94 Å)
Cite:P. aeruginosa CtpA protease adopts a novel activation mechanism to initiate the proteolytic process.
Embo J., 2024
8SXE
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BU of 8sxe by Molmil
Structure of the C-terminal protease CtpA-LbcA complex of Pseudomonas aeruginosa
Descriptor: Probable carboxyl-terminal protease, TPR repeat-containing protein PA4667, unidentified peptide
Authors:Hsu, H.-C, Li, H.
Deposit date:2023-05-22
Release date:2024-03-06
Last modified:2024-03-27
Method:ELECTRON MICROSCOPY (3.55 Å)
Cite:P. aeruginosa CtpA protease adopts a novel activation mechanism to initiate the proteolytic process.
Embo J., 2024
8UD9
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BU of 8ud9 by Molmil
Structure of human constitutive 20S proteasome complexed with the inhibitor TDI-8304
Descriptor: (7S,10S,13S)-N-cyclopentyl-10-[2-(morpholin-4-yl)ethyl]-9,12-dioxo-13-(2-oxopyrrolidin-1-yl)-2-oxa-8,11-diazabicyclo[13.3.1]nonadeca-1(19),15,17-triene-7-carboxamide, Proteasome subunit alpha type-1, Proteasome subunit alpha type-2, ...
Authors:Hsu, H.-C, Li, H.
Deposit date:2023-09-28
Release date:2023-12-20
Last modified:2024-01-03
Method:ELECTRON MICROSCOPY (2.04 Å)
Cite:Structures revealing mechanisms of resistance and collateral sensitivity of Plasmodium falciparum to proteasome inhibitors.
Nat Commun, 14, 2023
5TRR
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BU of 5trr by Molmil
Structure of Mycobacterium tuberculosis proteasome in complex with N,C-capped dipeptide PKS2169
Descriptor: N,N-diethyl-N~2~-(3-phenylpropanoyl)-L-asparaginyl-N-[(naphthalen-1-yl)methyl]-L-alaninamide, Proteasome subunit alpha, Proteasome subunit beta
Authors:Hsu, H.-C, Fan, H, Singh, P.K, Wang, R, Sukenick, G, Nathan, C, Lin, G, Li, H.
Deposit date:2016-10-27
Release date:2017-01-11
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (3.103 Å)
Cite:Structural Basis for the Species-Selective Binding of N,C-Capped Dipeptides to the Mycobacterium tuberculosis Proteasome.
Biochemistry, 56, 2017
5TRY
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BU of 5try by Molmil
Structure of Mycobacterium tuberculosis proteasome in complex with N,C-capped dipeptide PKS2206
Descriptor: (2~{S})-~{N}-[(2~{S})-3-methoxy-1-(naphthalen-1-ylmethylamino)-1-oxidanylidene-propan-2-yl]-4-oxidanylidene-2-(3-phenylpropanoylamino)-4-piperidin-1-yl-butanamide, Proteasome subunit alpha, Proteasome subunit beta
Authors:Hsu, H.-C, Fan, H, Singh, P.K, Wang, R, Sukenick, G, Nathan, C, Lin, G, Li, H.
Deposit date:2016-10-27
Release date:2017-01-11
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (3.000008 Å)
Cite:Structural Basis for the Species-Selective Binding of N,C-Capped Dipeptides to the Mycobacterium tuberculosis Proteasome.
Biochemistry, 56, 2017
5TS0
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BU of 5ts0 by Molmil
Structure of Mycobacterium tuberculosis proteasome in complex with N,C-capped dipeptide PKS2208
Descriptor: (2S)-N-{(2S)-3-methoxy-1-[(naphthalen-1-ylmethyl)amino]-1-oxopropan-2-yl}-4-oxo-2-[(3-phenylpropanoyl)amino]-4-(1H-pyrrol-1-yl)butanamide (non-preferred name), Proteasome subunit alpha, Proteasome subunit beta
Authors:Hsu, H.-C, Fan, H, Singh, P.K, Wang, R, Sukenick, G, Nathan, C, Lin, G, Li, H.
Deposit date:2016-10-27
Release date:2017-01-11
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (2.84679747 Å)
Cite:Structural Basis for the Species-Selective Binding of N,C-Capped Dipeptides to the Mycobacterium tuberculosis Proteasome.
Biochemistry, 56, 2017
5TRS
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BU of 5trs by Molmil
Structure of Mycobacterium tuberculosis proteasome in complex with N,C-capped dipeptide PKS2144
Descriptor: N-tert-butoxy-N~2~-(5-methyl-1,2-oxazole-3-carbonyl)-L-asparaginyl-O-methyl-N-[(naphthalen-1-yl)methyl]-L-serinamide, Proteasome subunit alpha, Proteasome subunit beta
Authors:Hsu, H.-C, Fan, H, Singh, P.K, Wang, R, Sukenick, G, Nathan, C, Lin, G, Li, H.
Deposit date:2016-10-27
Release date:2017-01-11
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (3.083567 Å)
Cite:Structural Basis for the Species-Selective Binding of N,C-Capped Dipeptides to the Mycobacterium tuberculosis Proteasome.
Biochemistry, 56, 2017
5TRG
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BU of 5trg by Molmil
Structure of Mycobacterium tuberculosis proteasome in complex with N,C-capped dipeptide DPLG-2
Descriptor: N,N-diethyl-N~2~-[(2E)-3-phenylprop-2-enoyl]-L-asparaginyl-4-fluoro-N-[(naphthalen-1-yl)methyl]-L-phenylalaninamide, Proteasome subunit alpha, Proteasome subunit beta
Authors:Hsu, H.-C, Fan, H, Singh, R.K, Wang, R, Sukenick, G, Nathan, C, Lin, G, Li, H.
Deposit date:2016-10-26
Release date:2017-01-11
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (2.804 Å)
Cite:Structural Basis for the Species-Selective Binding of N,C-Capped Dipeptides to the Mycobacterium tuberculosis Proteasome.
Biochemistry, 56, 2017
5URA
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BU of 5ura by Molmil
Enantiomer-Specific Binding of the Potent Antinociceptive Agent SBFI-26 to Anandamide transporters FABP7
Descriptor: (1S,2S,3S,4S)-3-{[(naphthalen-1-yl)oxy]carbonyl}-2,4-diphenylcyclobutane-1-carboxylic acid, Fatty acid-binding protein, brain, ...
Authors:Hsu, H.-C, Li, H.
Deposit date:2017-02-09
Release date:2017-08-23
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (1.85002172 Å)
Cite:The Antinociceptive Agent SBFI-26 Binds to Anandamide Transporters FABP5 and FABP7 at Two Different Sites.
Biochemistry, 56, 2017
5UR9
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BU of 5ur9 by Molmil
Enantiomer-Specific Binding of the Potent Antinociceptive Agent SBFI-26 to Anandamide transporters FABP5
Descriptor: (1S,2S,3S,4S)-3-{[(naphthalen-1-yl)oxy]carbonyl}-2,4-diphenylcyclobutane-1-carboxylic acid, Fatty acid-binding protein, epidermal, ...
Authors:Hsu, H.-C, Li, H.
Deposit date:2017-02-09
Release date:2017-08-23
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (2.19800353 Å)
Cite:The Antinociceptive Agent SBFI-26 Binds to Anandamide Transporters FABP5 and FABP7 at Two Different Sites.
Biochemistry, 56, 2017

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PDB entries from 2024-03-27

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