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3O9L
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BU of 3o9l by Molmil
Design and optimisation of new piperidines as renin inhibitors
Descriptor: (3R,4S)-N-[2-chloro-5-(3-methoxypropyl)benzyl]-N-cyclopropyl-4-{4-[2-(2,6-dichloro-4-methylphenoxy)ethoxy]phenyl}piperidine-3-carboxamide, 2-acetamido-2-deoxy-beta-D-glucopyranose, Renin
Authors:Corminboeuf, O, Bezencon, O, Grisostomi, C, Remen, L, Richard-Bildstein, S, Bur, D, Prade, L, Hess, P, Strickner, P, Treiber, A.
Deposit date:2010-08-04
Release date:2011-03-02
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:Design and optimization of new piperidines as renin inhibitors.
Bioorg.Med.Chem.Lett., 20, 2010
2QXG
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BU of 2qxg by Molmil
Crystal Structure of Human Kallikrein 7 in Complex with Ala-Ala-Phe-chloromethylketone
Descriptor: Kallikrein-7, L-alanyl-N-[(1S,2R)-1-benzyl-2-hydroxypropyl]-L-alaninamide
Authors:Debela, M, Hess, P, Magdolen, V, Bode, W, Steiner, T, Goettig, P.
Deposit date:2007-08-11
Release date:2008-01-08
Last modified:2023-08-30
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:Chymotryptic specificity determinants in the 1.0 A structure of the zinc-inhibited human tissue kallikrein 7.
Proc.Natl.Acad.Sci.Usa, 104, 2007
2QXH
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BU of 2qxh by Molmil
Crystal Structure of Human Kallikrein 7 in Complex with Suc-Ala-Ala-Pro-Phe-chloromethylketone
Descriptor: Kallikrein-7, N-(3-carboxypropanoyl)-L-alanyl-L-alanyl-N-[(2S,3S)-4-chloro-3-hydroxy-1-phenylbutan-2-yl]-L-prolinamide
Authors:Debela, M, Hess, P, Magdolen, V, Schechter, N.M, Bode, W, Goettig, P.
Deposit date:2007-08-11
Release date:2008-01-08
Last modified:2023-08-30
Method:X-RAY DIFFRACTION (2 Å)
Cite:Chymotryptic specificity determinants in the 1.0 A structure of the zinc-inhibited human tissue kallikrein 7.
Proc.Natl.Acad.Sci.Usa, 104, 2007
2QXJ
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BU of 2qxj by Molmil
Crystal Structure of Human Kallikrein 7 in Complex with Suc-Ala-Ala-Pro-Phe-chloromethylketone and Copper
Descriptor: COPPER (II) ION, Kallikrein-7, N-(3-carboxypropanoyl)-L-alanyl-L-alanyl-N-[(2S,3S)-4-chloro-3-hydroxy-1-phenylbutan-2-yl]-L-prolinamide
Authors:Debela, M, Hess, P, Magdolen, V, Schechter, N.M, Bode, W, Goettig, P.
Deposit date:2007-08-11
Release date:2008-01-08
Last modified:2023-08-30
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:Chymotryptic specificity determinants in the 1.0 A structure of the zinc-inhibited human tissue kallikrein 7.
Proc.Natl.Acad.Sci.Usa, 104, 2007
2QXI
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BU of 2qxi by Molmil
High resolution structure of Human Kallikrein 7 in Complex with Suc-Ala-Ala-Pro-Phe-chloromethylketone
Descriptor: Kallikrein-7, N-(3-carboxypropanoyl)-L-alanyl-L-alanyl-N-[(2S,3S)-4-chloro-3-hydroxy-1-phenylbutan-2-yl]-L-prolinamide
Authors:Debela, M, Hess, P, Magdolen, V, Schechter, N.M, Bode, W, Goettig, P.
Deposit date:2007-08-11
Release date:2008-01-08
Last modified:2023-08-30
Method:X-RAY DIFFRACTION (1 Å)
Cite:Chymotryptic specificity determinants in the 1.0 A structure of the zinc-inhibited human tissue kallikrein 7.
Proc.Natl.Acad.Sci.Usa, 104, 2007
2Q6P
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BU of 2q6p by Molmil
The Chemical Control of Protein Folding: Engineering a Superfolder Green Fluorescent Protein
Descriptor: Green fluorescent protein mutant 3
Authors:Steiner, T, Hess, P, Bae, J.H, Wiltschi, B, Moroder, L, Budisa, N.
Deposit date:2007-06-05
Release date:2007-06-19
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:Synthetic biology of proteins: tuning GFPs folding and stability with fluoroproline.
Plos One, 3, 2008
3G6Z
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BU of 3g6z by Molmil
Design and Preparation of Potent, Non-Peptidic, Bioavailable Renin Inhibitors
Descriptor: (1R,5S)-N-cyclopropyl-7-{4-[2-(2,6-dichloro-4-methylphenoxy)ethoxy]phenyl}-N-(2,3-dimethylbenzyl)-3,9-diazabicyclo[3.3.1]non-6-ene-6-carboxamide, 2-acetamido-2-deoxy-beta-D-glucopyranose, Renin
Authors:Bezencon, O, Bur, D, Prade, L, Weller, T, Boss, C, Fischli, W.
Deposit date:2009-02-09
Release date:2009-06-30
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (2 Å)
Cite:Design and Preparation of Potent, Nonpeptidic, Bioavailable Renin Inhibitors
J.Med.Chem., 52, 2009
3G70
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BU of 3g70 by Molmil
Design and Preparation of Potent, Non-Peptidic, Bioavailable Renin Inhibitors
Descriptor: (1R,5S)-7-{4-[3-(2-chloro-3,6-difluorophenoxy)propyl]phenyl}-N-cyclopropyl-N-(2,3-dichlorobenzyl)-3,9-diazabicyclo[3.3.1]non-6-ene-6-carboxamide, 2-acetamido-2-deoxy-beta-D-glucopyranose, DIMETHYL SULFOXIDE, ...
Authors:Bezencon, O, Bur, D, Prade, L, Weller, T, Boss, C, Fischli, W.
Deposit date:2009-02-09
Release date:2009-06-30
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (2 Å)
Cite:Design and Preparation of Potent, Nonpeptidic, Bioavailable Renin Inhibitors
J.Med.Chem., 52, 2009
3G72
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BU of 3g72 by Molmil
Design and Preparation of Potent, Non-Peptidic, Bioavailable Renin Inhibitors
Descriptor: (1S,5R)-7-{4-[3-(2-chloro-3,6-difluorophenoxy)propyl]phenyl}-N-cyclopropyl-N-(2,3-dichlorobenzyl)-3,9-diazabicyclo[3.3.1]non-6-ene-6-carboxamide, 2-acetamido-2-deoxy-beta-D-glucopyranose, DIMETHYL SULFOXIDE, ...
Authors:Bezencon, O, Bur, D, Prade, L, Weller, T, Boss, C, Fischli, W.
Deposit date:2009-02-09
Release date:2009-06-30
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Design and Preparation of Potent, Nonpeptidic, Bioavailable Renin Inhibitors
J.Med.Chem., 52, 2009
3K1W
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BU of 3k1w by Molmil
New Classes of Potent and Bioavailable Human Renin Inhibitors
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetylamino-2-deoxy-alpha-L-idopyranose, 4-{4-[3-(2-bromo-5-fluorophenoxy)propyl]phenyl}-N-(2-chlorobenzyl)-N-cyclopropyl-1,2,5,6-tetrahydropyridine-3-carboxamide, ...
Authors:Prade, L.
Deposit date:2009-09-29
Release date:2010-03-02
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (1.5 Å)
Cite:New classes of potent and bioavailable human renin inhibitors
Bioorg.Med.Chem.Lett., 19, 2009
3OAD
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BU of 3oad by Molmil
Design and optimization of new piperidines as renin inhibitors
Descriptor: (3S,4R)-N-[2-chloro-5-(2-methoxyethyl)benzyl]-N-cyclopropyl-4-{6-[2-(2,6-dichloro-4-methylphenoxy)ethoxy]pyridin-3-yl}-4-hydroxypiperidine-3-carboxamide, 2-acetamido-2-deoxy-beta-D-glucopyranose, Renin
Authors:Prade, L.
Deposit date:2010-08-05
Release date:2010-11-03
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (2.17 Å)
Cite:Design and optimization of new piperidines as renin inhibitors.
Bioorg.Med.Chem.Lett., 20, 2010
3OAG
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BU of 3oag by Molmil
Design and optimization of new piperidines as renin inhibitors
Descriptor: (3R,4S)-N-{2-chloro-5-[(cyclopropylamino)methyl]benzyl}-N-cyclopropyl-4-{6-[2-(2,6-dichloro-4-methylphenoxy)ethoxy]pyridin-3-yl}piperidine-3-carboxamide, 2-acetamido-2-deoxy-beta-D-glucopyranose, Renin
Authors:Prade, L.
Deposit date:2010-08-05
Release date:2010-11-03
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Design and optimization of new piperidines as renin inhibitors.
Bioorg.Med.Chem.Lett., 20, 2010
2OEF
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BU of 2oef by Molmil
Open and Closed Structures of the UDP-Glucose Pyrophosphorylase from Leishmania major
Descriptor: SULFATE ION, UTP-glucose-1-phosphate uridylyltransferase 2, putative
Authors:Steiner, T.
Deposit date:2006-12-29
Release date:2007-02-13
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:Open and Closed Structures of the UDP-glucose Pyrophosphorylase from Leishmania major.
J.Biol.Chem., 282, 2007
2OEG
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BU of 2oeg by Molmil
Open and Closed Structures of the UDP-Glucose Pyrophosphorylase from Leishmania major
Descriptor: URIDINE-5'-DIPHOSPHATE-GLUCOSE, UTP-glucose-1-phosphate uridylyltransferase 2, putative
Authors:Steiner, T.
Deposit date:2006-12-29
Release date:2007-02-13
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Open and Closed Structures of the UDP-glucose Pyrophosphorylase from Leishmania major.
J.Biol.Chem., 282, 2007

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