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1K8Q
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BU of 1k8q by Molmil
CRYSTAL STRUCTURE OF DOG GASTRIC LIPASE IN COMPLEX WITH A PHOSPHONATE INHIBITOR
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, Triacylglycerol lipase, gastric, ...
Authors:Roussel, A, Miled, N, Berti-Dupuis, L, Riviere, M, Spinelli, S, Berna, P, Gruber, V, Verger, R, Cambillau, C.
Deposit date:2001-10-25
Release date:2002-03-06
Last modified:2023-08-16
Method:X-RAY DIFFRACTION (2.7 Å)
Cite:Crystal structure of the open form of dog gastric lipase in complex with a phosphonate inhibitor.
J.Biol.Chem., 277, 2002
6ZCI
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BU of 6zci by Molmil
Crystal structure of BRD4-BD1 in complex with NVS-BET-1
Descriptor: (4~{R})-4-(4-chlorophenyl)-1-cyclopropyl-5-(1,5-dimethyl-6-oxidanylidene-pyridin-3-yl)-3-methyl-4~{H}-pyrrolo[3,4-c]pyrazol-6-one, Bromodomain-containing protein 4
Authors:Faller, M.
Deposit date:2020-06-11
Release date:2020-12-23
Last modified:2024-01-24
Method:X-RAY DIFFRACTION (1.976 Å)
Cite:BET bromodomain inhibitors regulate keratinocyte plasticity.
Nat.Chem.Biol., 17, 2021

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