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5JT2
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BU of 5jt2 by Molmil
BRAFV600E Kinase Domain In Complex with Chemically Linked Vemurafenib Inhibitor VEM-BISAMIDE
Descriptor: 2,2'-oxybis(N-{[4-(3-{2,6-difluoro-3-[(propane-1-sulfonyl)amino]benzoyl}-1H-pyrrolo[2,3-b]pyridin-5-yl)phenyl]methyl}acetamide), BENZAMIDINE, Serine/threonine-protein kinase B-raf
Authors:Grasso, M.J, Marmorstein, R.
Deposit date:2016-05-09
Release date:2016-09-14
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (2.702 Å)
Cite:Chemically Linked Vemurafenib Inhibitors Promote an Inactive BRAF(V600E) Conformation.
Acs Chem.Biol., 11, 2016
5JRQ
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BU of 5jrq by Molmil
BRAFV600E Kinase Domain In Complex with Chemically Linked Vemurafenib Inhibitor VEM-6-VEM
Descriptor: DIMETHYL SULFOXIDE, GLYCEROL, N-{2,4-difluoro-3-[5-(4-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]phenyl}propane-1-sulfonamide, ...
Authors:Grasso, M.J, Marmorstein, R.
Deposit date:2016-05-06
Release date:2016-09-14
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (2.287 Å)
Cite:Chemically Linked Vemurafenib Inhibitors Promote an Inactive BRAF(V600E) Conformation.
Acs Chem.Biol., 11, 2016
5JSM
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BU of 5jsm by Molmil
BRAFV600E Kinase Domain In Complex with Chemically Linked Vemurafenib Inhibitor VEM-3-VEM
Descriptor: BENZAMIDINE, CHLORIDE ION, DIMETHYL SULFOXIDE, ...
Authors:Grasso, M.J, Marmorstein, R.
Deposit date:2016-05-08
Release date:2016-09-14
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.19 Å)
Cite:Chemically Linked Vemurafenib Inhibitors Promote an Inactive BRAF(V600E) Conformation.
Acs Chem.Biol., 11, 2016
7L9X
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BU of 7l9x by Molmil
Structure of VPS4B in complex with an allele-specific covalent inhibitor
Descriptor: N-{3-[(8-phenyl[1,2,4]triazolo[1,5-a]pyridin-2-yl)amino]phenyl}propanamide, SULFATE ION, Vacuolar protein sorting-associated protein 4B
Authors:Grasso, M, Cupido, T, Kapoor, T.M.
Deposit date:2021-01-05
Release date:2021-04-14
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (2.81 Å)
Cite:A chemical genetics approach to examine the functions of AAA proteins.
Nat.Struct.Mol.Biol., 28, 2021

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PDB entries from 2024-03-27

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