Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
Search by PDB author
1AZE
DownloadVisualize
BU of 1aze by Molmil
NMR STRUCTURE OF THE COMPLEX BETWEEN THE C32S-Y7V MUTANT OF THE NSH3 DOMAIN OF GRB2 WITH A PEPTIDE FROM SOS, 10 STRUCTURES
Descriptor: GRB2, SOS
Authors:Vidal, M, Gincel, E, Goudreau, N, Cornille, F, Parker, F, Duchesne, M, Tocque, B, Garbay, C, Roques, B.P.
Deposit date:1997-11-17
Release date:1999-05-18
Last modified:2021-11-03
Method:SOLUTION NMR
Cite:Molecular and cellular analysis of Grb2 SH3 domain mutants: interaction with Sos and dynamin.
J.Mol.Biol., 290, 1999
1VZJ
DownloadVisualize
BU of 1vzj by Molmil
Structure of the tetramerization domain of acetylcholinesterase: four-fold interaction of a WWW motif with a left-handed polyproline helix
Descriptor: ACETYLCHOLINESTERASE, ACETYLCHOLINESTERASE COLLAGENIC TAIL PEPTIDE
Authors:Dvir, H, Harel, M, Bon, S, Liu, W.-Q, Vidal, M, Garbay, C, Sussman, J.L, Massoulie, J, Silman, I.
Deposit date:2004-05-20
Release date:2005-01-10
Last modified:2019-10-16
Method:X-RAY DIFFRACTION (2.35 Å)
Cite:The Synaptic Acetylcholinesterase Tetramer Assembles Around a Polyproline-II Helix
Embo J., 23, 2004
6GCW
DownloadVisualize
BU of 6gcw by Molmil
Focal Adhesion Kinase catalytic domain in complex with irreversible inhibitor
Descriptor: 2-[[5-chloranyl-2-[[4-[[[1-[2-(propanoylamino)ethyl]-1,2,3-triazol-4-yl]methylamino]methyl]phenyl]amino]pyrimidin-4-yl]amino]-~{N}-methyl-benzamide, Focal adhesion kinase 1, SULFATE ION
Authors:Yen-Pon, E, Li, B, Acebron-Garcia-de-Eulate, M, Tomkiewicz-Raulet, C, Dawson, J, Lietha, D, Frame, M.C, Coumoul, X, Garbay, C, Etheve-Quelquejeu, M, Chen, H.
Deposit date:2018-04-19
Release date:2019-05-01
Last modified:2019-10-02
Method:X-RAY DIFFRACTION (2 Å)
Cite:Structure-Based Design, Synthesis, and Characterization of the First Irreversible Inhibitor of Focal Adhesion Kinase.
Acs Chem.Biol., 13, 2018
6GCX
DownloadVisualize
BU of 6gcx by Molmil
Focal Adhesion Kinase catalytic domain in complex with irreversible inhibitor
Descriptor: 2-[[2-[[4-[[[3,4-bis(oxidanylidene)-2-[2-(propanoylamino)ethylamino]cyclobuten-1-yl]amino]methyl]phenyl]amino]-5-chloranyl-pyrimidin-4-yl]amino]-~{N}-methyl-benzamide, Focal adhesion kinase 1, SULFATE ION
Authors:Yen-Pon, E, Li, B, Acebron-Garcia de Eulate, M, Tomkiewicz-Raulet, C, Dawson, J, Lietha, D, Frame, M.C, Coumoul, X, Garbay, C, Etheve-Quelquejeu, M, Chen, H.
Deposit date:2018-04-19
Release date:2019-05-01
Last modified:2019-10-02
Method:X-RAY DIFFRACTION (1.553 Å)
Cite:Structure-Based Design, Synthesis, and Characterization of the First Irreversible Inhibitor of Focal Adhesion Kinase.
Acs Chem.Biol., 13, 2018
6GCR
DownloadVisualize
BU of 6gcr by Molmil
Focal Adhesion Kinase catalytic domain in complex with irreversible inhibitor
Descriptor: 2-[[2-[[4-[[[3,4-bis(oxidanylidene)-2-[2-(propanoylamino)ethylamino]cyclobuten-1-yl]amino]methyl]phenyl]amino]-5-chloranyl-pyrimidin-4-yl]amino]-~{N}-methyl-benzamide, Focal adhesion kinase 1
Authors:Yen-Pon, E, Li, B, Acebron-Garcia de Eulate, M, Tomkiewicz-Raulet, C, Dawson, J, Lietha, D, Frame, M.C, Coumoul, X, Garbay, C, Etheve-Quelquejeu, M, Chen, H.
Deposit date:2018-04-19
Release date:2019-05-01
Last modified:2019-10-02
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Structure-Based Design, Synthesis, and Characterization of the First Irreversible Inhibitor of Focal Adhesion Kinase.
Acs Chem.Biol., 13, 2018
1JYR
DownloadVisualize
BU of 1jyr by Molmil
Xray Structure of Grb2 SH2 Domain Complexed with a Phosphorylated Peptide
Descriptor: GROWTH FACTOR RECEPTOR-BOUND PROTEIN 2, peptide: PSpYVNVQN
Authors:Nioche, P, Liu, W.-Q, Broutin, I, Charbonnier, F, Latreille, M.-T, Vidal, M, Roques, B, Garbay, C, Ducruix, A.
Deposit date:2001-09-13
Release date:2002-03-13
Last modified:2018-10-10
Method:X-RAY DIFFRACTION (1.55 Å)
Cite:Crystal structures of the SH2 domain of Grb2: highlight on the binding of a new high-affinity inhibitor.
J.Mol.Biol., 315, 2002
1JYU
DownloadVisualize
BU of 1jyu by Molmil
Xray Structure of Grb2 SH2 Domain
Descriptor: GROWTH FACTOR RECEPTOR-BOUND PROTEIN 2
Authors:Nioche, P, Liu, W.-Q, Broutin, I, Charbonnier, F, Latreille, M.-T, Vidal, M, Roques, B, Garbay, C, Ducruix, A.
Deposit date:2001-09-13
Release date:2002-03-13
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (2.75 Å)
Cite:Crystal structures of the SH2 domain of Grb2: highlight on the binding of a new high-affinity inhibitor.
J.Mol.Biol., 315, 2002
1JYQ
DownloadVisualize
BU of 1jyq by Molmil
Xray Structure of Grb2 SH2 Domain Complexed with a Highly Affine Phospho Peptide
Descriptor: GROWTH FACTOR RECEPTOR-BOUND PROTEIN 2, mAZ-pY-(alpha Me)pY-N-NH2 peptide inhibitor
Authors:Nioche, P, Liu, W.-Q, Broutin, I, Charbonnier, F, Latreille, M.-T, Vidal, M, Roques, B, Garbay, C, Ducruix, A.
Deposit date:2001-09-13
Release date:2002-03-13
Last modified:2018-04-04
Method:X-RAY DIFFRACTION (2 Å)
Cite:Crystal structures of the SH2 domain of Grb2: highlight on the binding of a new high-affinity inhibitor.
J.Mol.Biol., 315, 2002
4BRX
DownloadVisualize
BU of 4brx by Molmil
Focal Adhesion Kinase catalytic domain in complex with a diarylamino- 1,3,5-triazine inhibitor
Descriptor: 2-(4-(2-methoxy-4-morpholinophenylamino)-1,3,5-triazin-2-ylamino)-N-methylbenzamide, FOCAL ADHESION KINASE 1, SULFATE ION
Authors:Le Coq, J, Lietha, D.
Deposit date:2013-06-05
Release date:2013-07-24
Last modified:2023-12-20
Method:X-RAY DIFFRACTION (2.05 Å)
Cite:Synthesis of Novel Diarylamino-1,3,5-Triazine Derivatives as Fak Inhibitors with Anti-Angiogenic Activity.
Bioorg.Med.Chem.Lett., 23, 2013
4C7T
DownloadVisualize
BU of 4c7t by Molmil
Focal Adhesion Kinase catalytic domain in complex with a diarylamino- 1,3,5-triazine inhibitor
Descriptor: FOCAL ADHESION KINASE 1, N-methyl-2-[[4-[(3,4,5-trimethoxyphenyl)amino]-1,3,5-triazin-2-yl]amino]benzamide, SULFATE ION
Authors:Le Coq, J, Lietha, D.
Deposit date:2013-09-25
Release date:2014-04-02
Last modified:2023-12-20
Method:X-RAY DIFFRACTION (2.05 Å)
Cite:Inhibition of Both Focal Adhesion Kinase and Fibroblast Growth Factor Receptor 2 Pathways Induces Anti-Tumor and Anti-Angiogenic Activities.
Cancer Lett., 348, 2014

217705

PDB entries from 2024-03-27

PDB statisticsPDBj update infoContact PDBjnumon