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5TI3
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BU of 5ti3 by Molmil
CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX WITH INHIBITOR 17503468
Descriptor: 1,2-ETHANEDIOL, 2,5-dibromo-N-[3-(2-oxopyrrolidin-1-yl)phenyl]benzene-1-sulfonamide, Bromodomain-containing protein 4
Authors:Zhu, J.-Y, Ember, S.W.J, SCHONBRUNN, E.
Deposit date:2016-09-30
Release date:2017-08-09
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (1.703 Å)
Cite:Identification of a Novel Class of BRD4 Inhibitors by Computational Screening and Binding Simulations.
ACS Omega, 2, 2017
5TI6
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BU of 5ti6 by Molmil
CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX WITH INHIBITOR 8841881
Descriptor: 1,2-ETHANEDIOL, 2,6-difluoro-N-[3-(2-oxopyrrolidin-1-yl)phenyl]benzene-1-sulfonamide, Bromodomain-containing protein 4
Authors:Zhu, J.-Y, Ember, S.W.J, Schonbrunn, E.
Deposit date:2016-10-01
Release date:2017-08-09
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (1.704 Å)
Cite:Identification of a Novel Class of BRD4 Inhibitors by Computational Screening and Binding Simulations.
ACS Omega, 2, 2017
5TI2
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BU of 5ti2 by Molmil
CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX WITH INHIBITOR 7635936
Descriptor: 1,2-ETHANEDIOL, 3-fluoro-N-[3-(2-oxopyrrolidin-1-yl)phenyl]benzene-1-sulfonamide, Bromodomain-containing protein 4
Authors:Zhu, J.-Y, Ember, S.W.J, SCHONBRUNN, E.
Deposit date:2016-09-30
Release date:2017-08-09
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (1.65 Å)
Cite:Identification of a Novel Class of BRD4 Inhibitors by Computational Screening and Binding Simulations.
ACS Omega, 2, 2017
5TI7
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BU of 5ti7 by Molmil
CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX WITH INHIBITOR 17528462
Descriptor: 1,2-ETHANEDIOL, 5-bromo-2-methoxy-N-(3-(2-oxopyrrolidin-1-yl)phenyl)benzenesulfonamide, Bromodomain-containing protein 4
Authors:Zhu, J.-Y, Ember, S.W.J, Schonbrunn, E.
Deposit date:2016-10-01
Release date:2017-08-09
Last modified:2024-02-28
Method:X-RAY DIFFRACTION (1.65 Å)
Cite:Identification of a Novel Class of BRD4 Inhibitors by Computational Screening and Binding Simulations.
ACS Omega, 2, 2017
5TI5
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BU of 5ti5 by Molmil
CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX WITH INHIBITOR 8841880
Descriptor: 1,2-ETHANEDIOL, 3-bromo-N-[3-(2-oxo-2,3-dihydro-1H-pyrrol-1-yl)phenyl]benzene-1-sulfonamide, Bromodomain-containing protein 4
Authors:Zhu, J.-Y, Ember, S.W.J, Schonbrunn, E.
Deposit date:2016-10-01
Release date:2017-08-09
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.83 Å)
Cite:Identification of a Novel Class of BRD4 Inhibitors by Computational Screening and Binding Simulations.
ACS Omega, 2, 2017
5TI4
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BU of 5ti4 by Molmil
CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX WITH INHIBITOR 8841871
Descriptor: 1,2-ETHANEDIOL, 3-chloro-4-fluoro-N-[3-(2-oxopyrrolidin-1-yl)phenyl]benzene-1-sulfonamide, Bromodomain-containing protein 4
Authors:Zhu, J.-Y, Ember, S.W.J, SCHONBRUNN, E.
Deposit date:2016-09-30
Release date:2017-08-09
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (1.62 Å)
Cite:Identification of a Novel Class of BRD4 Inhibitors by Computational Screening and Binding Simulations.
ACS Omega, 2, 2017

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PDB entries from 2024-03-27

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