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SOLUTION STRUCTURE OF THE N-TERMINAL 37 AMINO ACIDS OF THE MOUSE ARF TUMOR SUPPRESSOR PROTEIN
Descriptor:	P19 ARF PROTEIN
Authors:	DiGiammarino, E.L, Filippov, I, Weber, J.D, Bothner, B, Kriwacki, R.W.
Deposit date:	2000-12-05
Release date:	2001-12-05
Last modified:	2022-02-23
Method:	SOLUTION NMR
Cite:	Solution structure of the p53 regulatory domain of the p19Arf tumor suppressor protein. Biochemistry, 40, 2001

The novel p300/CBP inhibitor A-485 uncovers a unique mechanism of action to target AR in castrate resistant prostate cancer
Descriptor:	Histone acetyltransferase p300, N-[(4-fluorophenyl)methyl]-2-{(1R)-5-[(methylcarbamoyl)amino]-2',4'-dioxo-2,3-dihydro-3'H-spiro[indene-1,5'-[1,3]oxazolidin]-3'-yl}-N-[(2S)-1,1,1-trifluoropropan-2-yl]acetamide, SODIUM ION
Authors:	Jakob, C.G, Qiu, W, Edalji, R.P, Sun, C.
Deposit date:	2016-06-17
Release date:	2017-09-27
Last modified:	2023-09-27
Method:	X-RAY DIFFRACTION (1.95 Å)
Cite:	Discovery of a selective catalytic p300/CBP inhibitor that targets lineage-specific tumours. Nature, 550, 2017