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8U5G
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BU of 8u5g by Molmil
Crystal structure of the co-expressed SDS22:PP1:I3 complex
Descriptor: E3 ubiquitin-protein ligase PPP1R11, FE (III) ION, PHOSPHATE ION, ...
Authors:Choy, M.S, Peti, W, Page, R.
Deposit date:2023-09-12
Release date:2023-12-06
Last modified:2024-01-03
Method:X-RAY DIFFRACTION (3.2 Å)
Cite:The SDS22:PP1:I3 complex: SDS22 binding to PP1 loosens the active site metal to prime metal exchange.
J.Biol.Chem., 300, 2023
6OBS
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BU of 6obs by Molmil
PP1 Y134K
Descriptor: GLYCEROL, MANGANESE (II) ION, PHOSPHATE ION, ...
Authors:Choy, M.S, Moon, T.M, Bray, J.A, Archuleta, T.L, Shi, W, Peti, W, Page, R.
Deposit date:2019-03-21
Release date:2019-09-18
Last modified:2023-10-11
Method:X-RAY DIFFRACTION (1.803 Å)
Cite:SDS22 selectively recognizes and traps metal-deficient inactive PP1.
Proc.Natl.Acad.Sci.USA, 116, 2019
6ALZ
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BU of 6alz by Molmil
Crystal structure of Protein Phosphatase 1 bound to the natural inhibitor Tautomycetin
Descriptor: (2Z)-2-[(1R)-3-{[(2R,3S,4R,7S,8S,11S,13R,16E)-17-ethyl-4,8-dihydroxy-3,7,11,13-tetramethyl-6,15-dioxononadeca-16,18-dien-2-yl]oxy}-1-hydroxy-3-oxopropyl]-3-methylbut-2-enedioic acid, CHLORIDE ION, DIMETHYL SULFOXIDE, ...
Authors:Choy, M.S, Peti, W, Page, R.
Deposit date:2017-08-08
Release date:2017-11-29
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (2.208 Å)
Cite:PP1:Tautomycetin Complex Reveals a Path toward the Development of PP1-Specific Inhibitors.
J. Am. Chem. Soc., 139, 2017
4XPN
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BU of 4xpn by Molmil
Crystal Structure of Protein Phosphate 1 complexed with PP1 binding domain of GADD34
Descriptor: GLYCEROL, MANGANESE (II) ION, PHOSPHATE ION, ...
Authors:Choy, M.S, Peti, W, Page, R.
Deposit date:2015-01-17
Release date:2015-07-01
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.285 Å)
Cite:Structural and Functional Analysis of the GADD34:PP1 eIF2 alpha Phosphatase.
Cell Rep, 11, 2015
5KA2
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BU of 5ka2 by Molmil
Protein Tyrosine Phosphatase 1B YAYA (Y152A, Y153A) mutant, open state
Descriptor: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, GLYCEROL, ...
Authors:Choy, M.S, Peti, W, Page, R.
Deposit date:2016-06-01
Release date:2017-03-08
Last modified:2024-02-28
Method:X-RAY DIFFRACTION (2.071 Å)
Cite:Conformational Rigidity and Protein Dynamics at Distinct Timescales Regulate PTP1B Activity and Allostery.
Mol. Cell, 65, 2017
5KAC
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BU of 5kac by Molmil
Protein Tyrosine Phosphatase 1B P185G mutant, open state
Descriptor: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, GLYCEROL, ...
Authors:Choy, M.S, Machado, L.E.S.F, Peti, W, Page, R.
Deposit date:2016-06-01
Release date:2017-03-08
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Conformational Rigidity and Protein Dynamics at Distinct Timescales Regulate PTP1B Activity and Allostery.
Mol. Cell, 65, 2017
5KA3
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BU of 5ka3 by Molmil
Protein Tyrosine Phosphatase 1B YAYA (Y152A, Y153A) mutant in complex with TCS401, closed state
Descriptor: 2-(OXALYL-AMINO)-4,5,6,7-TETRAHYDRO-THIENO[2,3-C]PYRIDINE-3-CARBOXYLIC ACID, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, ...
Authors:Choy, M.S, Peti, W, Page, R.
Deposit date:2016-06-01
Release date:2017-03-08
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.141 Å)
Cite:Conformational Rigidity and Protein Dynamics at Distinct Timescales Regulate PTP1B Activity and Allostery.
Mol. Cell, 65, 2017
5KA1
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BU of 5ka1 by Molmil
Protein Tyrosine Phosphatase 1B Delta helix 7 mutant in complex with TCS401, closed state
Descriptor: 2-(OXALYL-AMINO)-4,5,6,7-TETRAHYDRO-THIENO[2,3-C]PYRIDINE-3-CARBOXYLIC ACID, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, ...
Authors:Choy, M.S, Peti, W, Page, R.
Deposit date:2016-06-01
Release date:2017-03-01
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (1.84 Å)
Cite:Conformational Rigidity and Protein Dynamics at Distinct Timescales Regulate PTP1B Activity and Allostery.
Mol. Cell, 65, 2017
5KA8
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BU of 5ka8 by Molmil
Protein Tyrosine Phosphatase 1B L192A mutant, open state
Descriptor: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, Tyrosine-protein phosphatase non-receptor type 1
Authors:Choy, M.S, Peti, W, Page, R.
Deposit date:2016-06-01
Release date:2017-03-01
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (1.971 Å)
Cite:Conformational Rigidity and Protein Dynamics at Distinct Timescales Regulate PTP1B Activity and Allostery.
Mol. Cell, 65, 2017
5KA9
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BU of 5ka9 by Molmil
Protein Tyrosine Phosphatase 1B L192A mutant in complex with TCS401, open state
Descriptor: 2-(OXALYL-AMINO)-4,5,6,7-TETRAHYDRO-THIENO[2,3-C]PYRIDINE-3-CARBOXYLIC ACID, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, ...
Authors:Choy, M.S, Peti, W, Page, R.
Deposit date:2016-06-01
Release date:2017-03-01
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.07 Å)
Cite:Conformational Rigidity and Protein Dynamics at Distinct Timescales Regulate PTP1B Activity and Allostery.
Mol. Cell, 65, 2017
5K9W
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BU of 5k9w by Molmil
Protein Tyrosine Phosphatase 1B (1-301) in complex with TCS401, closed state
Descriptor: 2-(OXALYL-AMINO)-4,5,6,7-TETRAHYDRO-THIENO[2,3-C]PYRIDINE-3-CARBOXYLIC ACID, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, ...
Authors:Choy, M.S, Peti, W, Page, R.
Deposit date:2016-06-01
Release date:2017-03-01
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.01 Å)
Cite:Conformational Rigidity and Protein Dynamics at Distinct Timescales Regulate PTP1B Activity and Allostery.
Mol. Cell, 65, 2017
5KA7
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BU of 5ka7 by Molmil
Protein Tyrosine Phosphatase 1B T178A mutant in complex with TCS401, closed state
Descriptor: 2-(OXALYL-AMINO)-4,5,6,7-TETRAHYDRO-THIENO[2,3-C]PYRIDINE-3-CARBOXYLIC ACID, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, ...
Authors:Choy, M.S, Peti, W, Page, R.
Deposit date:2016-06-01
Release date:2017-03-08
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.061 Å)
Cite:Conformational Rigidity and Protein Dynamics at Distinct Timescales Regulate PTP1B Activity and Allostery.
Mol. Cell, 65, 2017
5KA0
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BU of 5ka0 by Molmil
Protein Tyrosine Phosphatase 1B Delta helix 7, open state
Descriptor: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, GLYCEROL, ...
Authors:Choy, M.S, Peti, W, Page, R.
Deposit date:2016-06-01
Release date:2017-03-01
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (1.991 Å)
Cite:Conformational Rigidity and Protein Dynamics at Distinct Timescales Regulate PTP1B Activity and Allostery.
Mol. Cell, 65, 2017
5KAD
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BU of 5kad by Molmil
Protein Tyrosine Phosphatase 1B N193A mutant in complex with TCS401, closed state
Descriptor: 2-(OXALYL-AMINO)-4,5,6,7-TETRAHYDRO-THIENO[2,3-C]PYRIDINE-3-CARBOXYLIC ACID, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, ...
Authors:Choy, M.S, Peti, W, Page, R.
Deposit date:2016-06-01
Release date:2017-03-01
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Conformational Rigidity and Protein Dynamics at Distinct Timescales Regulate PTP1B Activity and Allostery.
Mol. Cell, 65, 2017
5K9V
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BU of 5k9v by Molmil
Protein Tyrosine Phosphatase 1B (1-301), open state
Descriptor: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, GLYCEROL, ...
Authors:Choy, M.S, Peti, W, Page, R.
Deposit date:2016-06-01
Release date:2017-03-01
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (1.898 Å)
Cite:Conformational Rigidity and Protein Dynamics at Distinct Timescales Regulate PTP1B Activity and Allostery.
Mol. Cell, 65, 2017
5KAA
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BU of 5kaa by Molmil
Protein Tyrosine Phosphatase 1B Delta helix 7, P185G mutant, open state
Descriptor: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, GLYCEROL, ...
Authors:Choy, M.S, Machado, L.E.S.F, Peti, W, Page, R.
Deposit date:2016-06-01
Release date:2017-03-08
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (1.968 Å)
Cite:Conformational Rigidity and Protein Dynamics at Distinct Timescales Regulate PTP1B Activity and Allostery.
Mol. Cell, 65, 2017
5KA4
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BU of 5ka4 by Molmil
Protein Tyrosine Phosphatase 1B T178A mutant, open state
Descriptor: Tyrosine-protein phosphatase non-receptor type 1
Authors:Choy, M.S, Peti, W, Page, R.
Deposit date:2016-06-01
Release date:2017-03-08
Last modified:2024-02-28
Method:X-RAY DIFFRACTION (2.185 Å)
Cite:Conformational Rigidity and Protein Dynamics at Distinct Timescales Regulate PTP1B Activity and Allostery.
Mol. Cell, 65, 2017
5KAB
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BU of 5kab by Molmil
Protein Tyrosine Phosphatase 1B Delta helix 7, P185G mutant in complex with TCS401, open state
Descriptor: 2-(OXALYL-AMINO)-4,5,6,7-TETRAHYDRO-THIENO[2,3-C]PYRIDINE-3-CARBOXYLIC ACID, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, ...
Authors:Choy, M.S, Machado, L.E.S.F, Peti, W, Page, R.
Deposit date:2016-06-01
Release date:2017-03-08
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (1.968 Å)
Cite:Conformational Rigidity and Protein Dynamics at Distinct Timescales Regulate PTP1B Activity and Allostery.
Mol. Cell, 65, 2017
6MKY
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BU of 6mky by Molmil
Human SDS22
Descriptor: Protein phosphatase 1 regulatory subunit 7, SULFATE ION
Authors:Choy, M.S, Bolik-Coulon, N, Page, R, Peti, W.
Deposit date:2018-09-26
Release date:2018-12-12
Last modified:2023-10-11
Method:X-RAY DIFFRACTION (2.9 Å)
Cite:The structure of SDS22 provides insights into the mechanism of heterodimer formation with PP1.
Acta Crystallogr F Struct Biol Commun, 74, 2018
6OBQ
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BU of 6obq by Molmil
PP1 H66K in complex with Microcystin LR
Descriptor: MANGANESE (II) ION, Microcystin LR, Serine/threonine-protein phosphatase PP1-alpha catalytic subunit
Authors:Choy, M.S, Moon, T.M, Bray, J.A, Archuleta, T.L, Shi, W, Peti, W, Page, R.
Deposit date:2019-03-21
Release date:2019-09-18
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (1.84 Å)
Cite:SDS22 selectively recognizes and traps metal-deficient inactive PP1.
Proc.Natl.Acad.Sci.USA, 116, 2019
6OBP
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BU of 6obp by Molmil
Reconstituted PP1 holoenzyme
Descriptor: CHLORIDE ION, MANGANESE (II) ION, PHOSPHATE ION, ...
Authors:Choy, M.S, Moon, T.M, Bray, J.A, Archuleta, T.L, Shi, W, Peti, W, Page, R.
Deposit date:2019-03-21
Release date:2019-09-18
Last modified:2023-10-11
Method:X-RAY DIFFRACTION (2.7 Å)
Cite:SDS22 selectively recognizes and traps metal-deficient inactive PP1.
Proc.Natl.Acad.Sci.USA, 116, 2019
6OBU
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BU of 6obu by Molmil
PP1 Y134K in complex with Microcystin LR
Descriptor: CHLORIDE ION, DIMETHYL SULFOXIDE, GLYCEROL, ...
Authors:Choy, M.S, Moon, T.M, Bray, J.A, Archuleta, T.L, Shi, W, Peti, W, Page, R.
Deposit date:2019-03-21
Release date:2019-09-18
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (1.95 Å)
Cite:SDS22 selectively recognizes and traps metal-deficient inactive PP1.
Proc.Natl.Acad.Sci.USA, 116, 2019
6OBN
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BU of 6obn by Molmil
The crystal structure of coexpressed SDS22:PP1 complex
Descriptor: (4S)-2-METHYL-2,4-PENTANEDIOL, CHLORIDE ION, FE (III) ION, ...
Authors:Choy, M.S, Moon, T.M, Bray, J.A, Archuleta, T.L, Shi, W, Peti, W, Page, R.
Deposit date:2019-03-21
Release date:2019-09-18
Last modified:2023-10-11
Method:X-RAY DIFFRACTION (2.7 Å)
Cite:SDS22 selectively recognizes and traps metal-deficient inactive PP1.
Proc.Natl.Acad.Sci.USA, 116, 2019
6OBR
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BU of 6obr by Molmil
PP1 Y134A in complex with Microcystin LR
Descriptor: CHLORIDE ION, MANGANESE (II) ION, Microcystin LR, ...
Authors:Choy, M.S, Moon, T.M, Bray, J.A, Archuleta, T.L, Shi, W, Peti, W, Page, R.
Deposit date:2019-03-21
Release date:2019-09-18
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (1.5 Å)
Cite:SDS22 selectively recognizes and traps metal-deficient inactive PP1.
Proc.Natl.Acad.Sci.USA, 116, 2019
4MOV
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BU of 4mov by Molmil
1.45 A Resolution Crystal Structure of Protein Phosphatase 1
Descriptor: CHLORIDE ION, MANGANESE (II) ION, PHOSPHATE ION, ...
Authors:Choy, M.S, Peti, W, Page, R.
Deposit date:2013-09-12
Release date:2014-03-26
Last modified:2023-09-20
Method:X-RAY DIFFRACTION (1.4503 Å)
Cite:Understanding the antagonism of retinoblastoma protein dephosphorylation by PNUTS provides insights into the PP1 regulatory code.
Proc.Natl.Acad.Sci.USA, 111, 2014

 

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