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3ZEB
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A COMPLEX OF GLPG WITH ISOCOUMARIN INHIBITOR COVALENTLY BONDED TO SERINE 201 AND HISTIDINE 150
Descriptor:RHOMBOID PROTEASE GLPG, 2-phenylethyl 2-(4-azanyl-2-methanoyl-phenyl)ethanoate, CHLORIDE ION, ...
Authors:Vinothkumar, K.R., voskya, O., Kuettler, E.V., Brouwer, A.J., Liskamp, R.M.J., Verhelst, S.H.L.
Deposit date:2012-12-04
Release date:2013-02-13
Last modified:2019-02-27
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Activity-Based Probes for Rhomboid Proteases Discovered in a Mass Spectrometry-Based Assay.
Proc.Natl.Acad.Sci.USA, 110, 2013
4R17
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LIGAND-INDUCED AZIRIDINE-FORMATION AT SUBUNIT BETA5 OF THE YEAST 20S PROTEASOME
Descriptor:Proteasome subunit alpha type-2, Proteasome subunit alpha type-3, Proteasome subunit alpha type-4, ...
Authors:Dubiella, C., Cui, H., Gersch, M., Brouwer, A.J., Sieber, S.A., Krueger, A., Liskamp, R., Groll, M.
Deposit date:2014-08-04
Release date:2014-10-15
Last modified:2014-11-05
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:Selective inhibition of the immunoproteasome by ligand-induced crosslinking of the active site.
Angew.Chem.Int.Ed.Engl., 53, 2014
4R18
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LIGAND-INDUCED LYS33-THR1 CROSSLINKING AT SUBUNIT BETA5 OF THE YEAST 20S PROTEASOME
Descriptor:PROTEASOME SUBUNIT ALPHA TYPE-2, PROTEASOME SUBUNIT ALPHA TYPE-3, PROTEASOME SUBUNIT ALPHA TYPE-4, ...
Authors:Dubiella, C., Cui, H., Gersch, M., Brouwer, A.J., Sieber, S.A., Krueger, A., Liskamp, R., Groll, M.
Deposit date:2014-08-04
Release date:2014-10-15
Last modified:2014-11-05
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:Selective inhibition of the immunoproteasome by ligand-induced crosslinking of the active site.
Angew.Chem.Int.Ed.Engl., 53, 2014