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5YAW
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BU of 5yaw by Molmil
Fragment-based Drug Discovery of inhibitors to block PDEdelta-RAS protein-protein interaction
Descriptor: 3-[(4-methoxyphenyl)methylsulfanyl]-5-(2-methylpropyl)-4-(phenylmethyl)-1,2,4-triazole, Retinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit delta
Authors:Bing, X, Yanlian, L, Danyan, C.
Deposit date:2017-09-01
Release date:2018-09-05
Last modified:2024-03-27
Method:X-RAY DIFFRACTION (2.027 Å)
Cite:Fragment-based Drug Discovery of inhibitors to block PDEdelta-RAS protein-protein interaction
To Be Published
5YAV
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BU of 5yav by Molmil
Fragment-based Drug Discovery of inhibitors to block PDEdelta-RAS protein-protein interaction
Descriptor: 1-phenyl-5-propan-2-ylsulfanyl-1,2,3,4-tetrazole, Retinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit delta
Authors:Bing, X, Yanlian, L, Danyan, C.
Deposit date:2017-09-01
Release date:2018-09-05
Last modified:2024-03-27
Method:X-RAY DIFFRACTION (1.989 Å)
Cite:Fragment-based Drug Discovery of inhibitors to block PDEdelta-RAS protein-protein interaction
To Be Published
5YOU
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BU of 5you by Molmil
Crystal structure of BRD4-BD1 bound with hjp64
Descriptor: (3~{R})-4-cyclopropyl-~{N},1,3-trimethyl-~{N}-(4-methylphenyl)-2-oxidanylidene-3~{H}-quinoxaline-6-carboxamide, Bromodomain-containing protein 4
Authors:Bing, X, Jianping, H, Yanlian, L, Danyan, C.
Deposit date:2017-10-31
Release date:2018-11-07
Last modified:2024-03-27
Method:X-RAY DIFFRACTION (1.503 Å)
Cite:Crystal structure of BRD4-BD1 bound with hjp64
To Be Published
6INS
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BU of 6ins by Molmil
X-RAY ANALYSIS OF THE SINGLE CHAIN B29-A1 PEPTIDE-LINKED INSULIN MOLECULE. A COMPLETELY INACTIVE ANALOGUE
Descriptor: INSULIN, ZINC ION
Authors:Derewenda, U, Derewenda, Z, Dodson, E.J, Dodson, G.G, Bing, X, Markussen, J.
Deposit date:1992-11-25
Release date:1994-01-31
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (2 Å)
Cite:X-ray analysis of the single chain B29-A1 peptide-linked insulin molecule. A completely inactive analogue.
J.Mol.Biol., 220, 1991
5XHY
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BU of 5xhy by Molmil
BRD4 bound with compound Bdi1
Descriptor: Bromodomain-containing protein 4, ~{N}-(4-cyclopropyl-1,3,3-trimethyl-2-oxidanylidene-quinoxalin-6-yl)-4-methyl-benzenesulfonamide
Authors:Xiong, B, Cao, D, Li, Y.
Deposit date:2017-04-25
Release date:2018-05-02
Last modified:2024-03-27
Method:X-RAY DIFFRACTION (1.976 Å)
Cite:BRD4 bound with compound Bdi1
To Be Published

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