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2VBA
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BU of 2vba by Molmil
beta-ketoacyl-ACP synthase I (KAS) from E. coli with bound amino- thiazole inhibitor
Descriptor: 2-PHENYLAMINO-4-METHYL-5-ACETYL THIAZOLE, 3-OXOACYL-[ACYL-CARRIER-PROTEIN] SYNTHASE 1
Authors:Pappenberger, G, Schulz-Gasch, T, Bailly, J, Hennig, M.
Deposit date:2007-09-06
Release date:2007-12-25
Last modified:2023-12-13
Method:X-RAY DIFFRACTION (1.36 Å)
Cite:Structure-Assisted Discovery of an Aminothiazole Derivative as a Lead Molecule for Inhibition of Bacterial Fatty-Acid Synthesis.
Acta Crystallogr.,Sect.D, 63, 2007
2VB7
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BU of 2vb7 by Molmil
beta-ketoacyl-ACP synthase I (KAS) from E. coli, apo structure after soak in PEG solution
Descriptor: 3-OXOACYL-[ACYL-CARRIER-PROTEIN] SYNTHASE 1
Authors:Pappenberger, G, Schulz-Gasch, T, Bailly, J, Hennig, M.
Deposit date:2007-09-06
Release date:2007-12-25
Last modified:2023-12-13
Method:X-RAY DIFFRACTION (1.6 Å)
Cite:Structure-Assisted Discovery of an Aminothiazole Derivative as a Lead Molecule for Inhibition of Bacterial Fatty-Acid Synthesis.
Acta Crystallogr.,Sect.D, 63, 2007
2VB8
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BU of 2vb8 by Molmil
beta-ketoacyl-ACP synthase I (KAS) from E. coli with bound inhibitor thiolactomycin
Descriptor: 3-OXOACYL-[ACYL-CARRIER-PROTEIN] SYNTHASE 1, CHLORIDE ION, THIOLACTOMYCIN
Authors:Pappenberger, G, Schulz-Gasch, T, Bailly, J, Hennig, M.
Deposit date:2007-09-06
Release date:2007-12-25
Last modified:2023-12-13
Method:X-RAY DIFFRACTION (1.52 Å)
Cite:Structure-Assisted Discovery of an Aminothiazole Derivative as a Lead Molecule for Inhibition of Bacterial Fatty-Acid Synthesis.
Acta Crystallogr.,Sect.D, 63, 2007
2VB9
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BU of 2vb9 by Molmil
beta-ketoacyl-ACP synthase I (KAS) from E. coli, apo structure
Descriptor: 3-OXOACYL-[ACYL-CARRIER-PROTEIN] SYNTHASE 1, CHLORIDE ION
Authors:Pappenberger, G, Schulz-Gasch, T, Bailly, J, Hennig, M.
Deposit date:2007-09-06
Release date:2007-12-25
Last modified:2023-12-13
Method:X-RAY DIFFRACTION (1.5 Å)
Cite:Structure-Assisted Discovery of an Aminothiazole Derivative as a Lead Molecule for Inhibition of Bacterial Fatty-Acid Synthesis.
Acta Crystallogr.,Sect.D, 63, 2007

217705

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