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5UIG
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CRYSTAL STRUCTURE OF ADENOSINE A2A RECEPTOR BOUND TO A NOVEL TRIAZOLE-CARBOXIMIDAMIDE ANTAGONIST
Descriptor:Adenosine receptor A2a,Soluble cytochrome b562,Adenosine receptor A2a, {[-(BIS-CARBOXYMETHYL-AMINO)-ETHYL]-CARBOXYMETHYL-AMINO}-ACETIC ACID, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, ...
Authors:Sun, B., Bachhawat, P., Ling-Hon Chu, M., Ceska, T., Sands, Z., Lebon, F., Kobilka, T.S., Kobilka, B.
Deposit date:2017-01-13
Release date:2017-02-08
Last modified:2017-03-08
Method:X-RAY DIFFRACTION (3.5 Å)
Cite:Crystal structure of the adenosine A2A receptor bound to an antagonist reveals a potential allosteric pocket.
Proc. Natl. Acad. Sci. U.S.A., 114, 2017
5DSG
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STRUCTURE OF THE M4 MUSCARINIC ACETYLCHOLINE RECEPTOR (M4-MT4L) BOUND TO TIOTROPIUM
Descriptor:Muscarinic acetylcholine receptor M4,Endolysin,Endolysin,Muscarinic acetylcholine receptor M4, (1R,2R,4S,5S,7S)-7-{[hydroxy(dithiophen-2-yl)acetyl]oxy}-9,9-dimethyl-3-oxa-9-azoniatricyclo[3.3.1.0~2,4~]nonane, OLEIC ACID, ...
Authors:Thal, D.M., Kobilka, B.K., Sexton, P.M., Christopoulos, A.
Deposit date:2015-09-17
Release date:2016-03-16
Last modified:2017-10-11
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:Crystal structures of the M1 and M4 muscarinic acetylcholine receptors.
Nature, 531, 2016
5CXV
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STRUCTURE OF THE HUMAN M1 MUSCARINIC ACETYLCHOLINE RECEPTOR BOUND TO ANTAGONIST TIOTROPIUM
Descriptor:Muscarinic acetylcholine receptor M1,Endolysin,Muscarinic acetylcholine receptor M1, FLAG peptide, (1R,2R,4S,5S,7S)-7-{[hydroxy(dithiophen-2-yl)acetyl]oxy}-9,9-dimethyl-3-oxa-9-azoniatricyclo[3.3.1.0~2,4~]nonane, ...
Authors:Sun, B., Feng, D., Li, X., Kobilka, T.S., Kobilka, B.K.
Deposit date:2015-07-29
Release date:2016-03-09
Last modified:2016-03-30
Method:X-RAY DIFFRACTION (2.7 Å)
Cite:Crystal structures of the M1 and M4 muscarinic acetylcholine receptors.
Nature, 531, 2016
2PKX
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E.COLI RESPONSE REGULATOR PHOP RECEIVER DOMAIN
Descriptor:Transcriptional regulatory protein phoP
Authors:Bachhawat, P.
Deposit date:2007-04-18
Release date:2007-05-22
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (2.54 Å)
Cite:Crystal Structures of the Receiver Domain of the Response Regulator PhoP from Escherichia coli in the Absence and Presence of the Phosphoryl Analog Beryllofluoride.
J.Bacteriol., 189, 2007
2PL1
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BERRYLIUM FLUORIDE ACTIVATED RECEIVER DOMAIN OF E.COLI PHOP
Descriptor:Transcriptional regulatory protein phoP, PLATINUM (II) ION, MAGNESIUM ION, ...
Authors:Bachhawat, P.
Deposit date:2007-04-18
Release date:2007-05-22
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Crystal Structures of the Receiver Domain of the Response Regulator PhoP from Escherichia coli in the Absence and Presence of the Phosphoryl Analog Beryllofluoride.
J.Bacteriol., 189, 2007
1ZES
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BEF3- ACTIVATED PHOB RECEIVER DOMAIN
Descriptor:Phosphate regulon transcriptional regulatory protein phoB, MAGNESIUM ION, BERYLLIUM TRIFLUORIDE ION
Authors:Bachhawat, P., Montelione, G.T., Stock, A.M.
Deposit date:2005-04-19
Release date:2005-09-20
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Mechanism of Activation for Transcription Factor PhoB Suggested by Different Modes of Dimerization in the Inactive and Active States.
Structure, 13, 2005