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1RMX
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BU of 1rmx by Molmil
A SHORT LEXITROPSIN THAT RECOGNIZES THE DNA MINOR GROOVE AT 5'-ACTAGT-3': UNDERSTANDING THE ROLE OF ISOPROPYL-THIAZOLE
Descriptor: 5'-D(*CP*GP*AP*CP*TP*AP*GP*TP*CP*G)-3', N-[3-(DIMETHYLAMINO)PROPYL]-2-({[4-({[4-(FORMYLAMINO)-1-METHYL-1H-PYRROL-2-YL]CARBONYL}AMINO)-1-METHYL-1H-PYRROL-2-YL]CARBONYL}AMINO)-5-ISOPROPYL-1,3-THIAZOLE-4-CARBOXAMIDE
Authors:Anthony, N.G, Johnston, B.F, Khalaf, A.I, Mackay, S.P, Parkinson, J.A, Suckling, C.J, Waigh, R.D.
Deposit date:2003-11-28
Release date:2004-08-24
Last modified:2022-03-02
Method:SOLUTION NMR
Cite:Short Lexitropsin that Recognizes the DNA Minor Groove at 5'-ACTAGT-3': Understanding the Role of Isopropyl-thiazole.
J.Am.Chem.Soc., 126, 2004
1RN9
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BU of 1rn9 by Molmil
A SHORT LEXITROPSIN THAT RECOGNIZES THE DNA MINOR GROOVE AT 5'-ACTAGT-3': UNDERSTANDING THE ROLE OF ISOPROPYL-THIAZOLE
Descriptor: 5'-D(*CP*GP*AP*CP*TP*AP*GP*TP*CP*G)-3'
Authors:Anthony, N.G, Johnston, B.F, Khalaf, A.I, Mackay, S.P, Parkinson, J.A, Suckling, C.J, Waigh, R.D.
Deposit date:2003-12-01
Release date:2004-08-24
Last modified:2022-03-02
Method:SOLUTION NMR
Cite:Short Lexitropsin that Recognizes the DNA Minor Groove at 5'-ACTAGT-3': Understanding the Role of Isopropyl-thiazole.
J.Am.Chem.Soc., 126, 2004
4V3L
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BU of 4v3l by Molmil
RNF38-UB-UbcH5B-Ub complex
Descriptor: 1,2-ETHANEDIOL, E3 UBIQUITIN-PROTEIN LIGASE RNF38, POLYUBIQUITIN-C, ...
Authors:Buetow, L, Gabrielsen, M, Anthony, N.G, Dou, H, Patel, A, Aitkenhead, H, Sibbet, G.J, Smith, B.O, Huang, D.T.
Deposit date:2014-10-20
Release date:2015-04-08
Last modified:2019-07-31
Method:X-RAY DIFFRACTION (1.53 Å)
Cite:Activation of a Primed Ring E3-E2-Ubiquitin Complex by Non-Covalent Ubiquitin.
Mol.Cell, 58, 2015
4V3K
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BU of 4v3k by Molmil
RNF38-UbcH5B-UB complex
Descriptor: 1,2-ETHANEDIOL, CHLORIDE ION, E3 UBIQUITIN-PROTEIN LIGASE RNF38, ...
Authors:Buetow, L, Gabrielsen, M, Anthony, N.G, Dou, H, Patel, A, Aitkenhead, H, Sibbet, G.J, Smith, B.O, Huang, D.T.
Deposit date:2014-10-20
Release date:2015-04-08
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (2.04 Å)
Cite:Activation of a Primed Ring E3-E2-Ubiquitin Complex by Non-Covalent Ubiquitin.
Mol.Cell, 58, 2015
4BXN
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BU of 4bxn by Molmil
Eg5(WT) complex
Descriptor: ADENOSINE-5'-DIPHOSPHATE, CADMIUM ION, CHLORIDE ION, ...
Authors:Talapatra, S.K, Anthony, N.G, Mackay, S.P, Kozielski, F.
Deposit date:2013-07-15
Release date:2013-07-31
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (2.793 Å)
Cite:The Mitotic Kinesin Eg5 Overcomes Inhibition to the Phase I/II Clinical Candidate Sb743921 by an Allosteric Resistance Mechanism.
J.Med.Chem., 56, 2013
2MNF
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BU of 2mnf by Molmil
AIK-18/51 DNA recognition sequence d(CGACTAGTCG)2
Descriptor: 5'-D(*CP*GP*AP*CP*TP*AP*GP*TP*CP*G)-3'
Authors:Alniss, H.Y, Salvia, M.-V, Sadikov, M, Golovchenko, I, Anthony, N.G, Khalaf, A.I, Mackay, S.P, Suckling, C.J, Parkinson, J.A.
Deposit date:2014-04-03
Release date:2014-07-30
Last modified:2014-09-17
Method:SOLUTION NMR
Cite:Recognition of the DNA minor groove by thiazotropsin analogues.
Chembiochem, 15, 2014
2MND
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BU of 2mnd by Molmil
Recognition complex of DNA d(CGACGCGTCG)2 with thiazotropsin B
Descriptor: 5'-D(*CP*GP*AP*CP*GP*CP*GP*TP*CP*G)-3', thiazotropsin B
Authors:Alniss, H.Y, Salvia, M.-V, Sadikov, M, Golovchenko, I, Anthony, N.G, Khalaf, A.I, Mackay, S.P, Suckling, C.J, Parkinson, J.A.
Deposit date:2014-04-03
Release date:2014-07-30
Last modified:2014-09-17
Method:SOLUTION NMR
Cite:Recognition of the DNA minor groove by thiazotropsin analogues.
Chembiochem, 15, 2014
2MNB
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BU of 2mnb by Molmil
Thiazotropsin B DNA recognition sequence d(CGACGCGTCG)2
Descriptor: 5'-D(*CP*GP*AP*CP*GP*CP*GP*TP*CP*G)-3'
Authors:Alniss, H.Y, Salvia, M.-V, Sadikov, M, Golovchenko, I, Anthony, N.G, Khalaf, A.I, Mackay, S.P, Suckling, C.J, Parkinson, J.A.
Deposit date:2014-04-02
Release date:2014-09-17
Method:SOLUTION NMR
Cite:Recognition of the DNA minor groove by thiazotropsin analogues.
Chembiochem, 15, 2014
2MNE
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BU of 2mne by Molmil
Recognition complex of DNA d(CGACTAGTCG)2 with thiazotropsin analogue AIK-18/51
Descriptor: 5'-D(*CP*GP*AP*CP*TP*AP*GP*TP*CP*G)-3', AIK-18/51
Authors:Alniss, H.Y, Salvia, M.-V, Sadikov, M, Golovchenko, I, Anthony, N.G, Khalaf, A.I, Mackay, S.P, Suckling, C.J, Parkinson, J.A.
Deposit date:2014-04-03
Release date:2014-07-30
Last modified:2014-09-17
Method:SOLUTION NMR
Cite:Recognition of the DNA minor groove by thiazotropsin analogues.
Chembiochem, 15, 2014
4A1Z
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BU of 4a1z by Molmil
Eg5-1
Descriptor: ADENOSINE-5'-DIPHOSPHATE, KINESIN-LIKE PROTEIN KIF11, MAGNESIUM ION, ...
Authors:Talapatra, S.K, Kozielski, F.
Deposit date:2011-09-20
Release date:2012-10-31
Last modified:2023-12-20
Method:X-RAY DIFFRACTION (2.8 Å)
Cite:The Mitotic Kinesin Eg5 Overcomes Inhibition to the Phase I/II Clinical Candidate Sb743921 by an Allosteric Resistance Mechanism.
J.Med.Chem., 56, 2013
4A28
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BU of 4a28 by Molmil
Eg5-2
Descriptor: ADENOSINE-5'-DIPHOSPHATE, KINESIN-LIKE PROTEIN KIF11, MAGNESIUM ION
Authors:Talapatra, S.K, Kozielski, F.
Deposit date:2011-09-22
Release date:2012-10-31
Last modified:2023-12-20
Method:X-RAY DIFFRACTION (2.55 Å)
Cite:The Mitotic Kinesin Eg5 Overcomes Inhibition to the Phase I/II Clinical Candidate Sb743921 by an Allosteric Resistance Mechanism.
J.Med.Chem., 56, 2013
4AS7
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BU of 4as7 by Molmil
Eg5 complex 1
Descriptor: ADENOSINE-5'-DIPHOSPHATE, CADMIUM ION, CHLORIDE ION, ...
Authors:Talapatra, S.K, Kozielski, F.
Deposit date:2012-04-29
Release date:2013-05-15
Last modified:2023-12-20
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:The Mitotic Kinesin Eg5 Overcomes Inhibition to the Phase I/II Clinical Candidate Sb743921 by an Allosteric Resistance Mechanism.
J.Med.Chem., 56, 2013
4B7B
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BU of 4b7b by Molmil
Eg5-3
Descriptor: ADENOSINE-5'-DIPHOSPHATE, CADMIUM ION, CALCIUM ION, ...
Authors:Talapatra, S.K, Kozielski, F.
Deposit date:2012-08-17
Release date:2013-07-31
Last modified:2023-12-20
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:The Mitotic Kinesin Eg5 Overcomes Inhibition to the Phase I/II Clinical Candidate Sb743921 by an Allosteric Resistance Mechanism.
J.Med.Chem., 56, 2013

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