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5BMM
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Src in complex with DNA-templated macrocyclic inhibitor MC25b
Descriptor: Proto-oncogene tyrosine-protein kinase Src, macrocyclic inhibitor MC25b
Authors:Georghiou, G, Guja, K.E, Aleem, S, Kleiner, R.E, Liu, D.R, Miller, W.T, Garcia-Diaz, M, Seeliger, M.A.
Deposit date:2015-05-22
Release date:2016-09-21
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:Structural and Biochemical Basis for Intracellular Kinase Inhibition by Src-specific Peptidic Macrocycles.
Cell Chem Biol, 23, 2016

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