Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
Search by PDB author
3KMR
DownloadVisualize
BU of 3kmr by Molmil
Crystal structure of RARalpha ligand binding domain in complex with an agonist ligand (Am580) and a coactivator fragment
Descriptor: 4-{[(5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthalen-2-yl)carbonyl]amino}benzoic acid, Nuclear receptor coactivator 1, Retinoic acid receptor alpha
Authors:Bourguet, W, Teyssier, C.
Deposit date:2009-11-11
Release date:2010-06-02
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:A unique secondary-structure switch controls constitutive gene repression by retinoic acid receptor.
Nat.Struct.Mol.Biol., 17, 2010
6STI
DownloadVisualize
BU of 6sti by Molmil
Crystal structure of RXRalpha LBD in complex with LG 100754 and a coactivator peptide
Descriptor: (2E,4E,6Z)-3-methyl-7-(5,5,8,8-tetramethyl-3-propoxy-5,6,7,8-tetrahydronaphthalen-2-yl)octa-2,4,6-trienoic acid, ACETATE ION, Nuclear receptor coactivator 2, ...
Authors:le Maire, A, Teyssier, C, Germain, P, Bourguet, W.
Deposit date:2019-09-10
Release date:2019-11-20
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (1.892 Å)
Cite:Regulation of RXR-RAR Heterodimers by RXR- and RAR-Specific Ligands and Their Combinations.
Cells, 8, 2019
6SSQ
DownloadVisualize
BU of 6ssq by Molmil
Crystal structure of RARbeta LBD in complex with LG 100754
Descriptor: (2E,4E,6Z)-3-methyl-7-(5,5,8,8-tetramethyl-3-propoxy-5,6,7,8-tetrahydronaphthalen-2-yl)octa-2,4,6-trienoic acid, CITRATE ANION, GLYCEROL, ...
Authors:le Maire, A, Teyssier, C, Germain, P, Bourguet, W.
Deposit date:2019-09-09
Release date:2019-11-20
Last modified:2024-01-24
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Regulation of RXR-RAR Heterodimers by RXR- and RAR-Specific Ligands and Their Combinations.
Cells, 8, 2019
4JYI
DownloadVisualize
BU of 4jyi by Molmil
Crystal structure of RARbeta LBD in complex with selective partial agonist BMS641 [3-chloro-4-[(E)-2-(5,5-dimethyl-8-phenyl-5,6-dihydronaphthalen-2-yl)ethenyl]benzoic acid]
Descriptor: 3-chloro-4-[(E)-2-(5,5-dimethyl-8-phenyl-5,6-dihydronaphthalen-2-yl)ethenyl]benzoic acid, CITRATE ANION, Nuclear receptor coactivator 1, ...
Authors:Nadendla, E.K, Teyssier, C, Germain, P, Delfosse, V, Bourguet, W.
Deposit date:2013-03-29
Release date:2014-03-19
Last modified:2024-02-28
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:An Unexpected Mode Of Binding Defines BMS948 as A Full Retinoic Acid Receptor beta (RAR beta , NR1B2) Selective Agonist.
Plos One, 10, 2015
4JYH
DownloadVisualize
BU of 4jyh by Molmil
Crystal structure of RARbeta LBD in complex with selective agonist BMS948 [4-{[(8-phenylnaphthalen-2-yl)carbonyl]amino}benzoic acid]
Descriptor: 4-{[(8-phenylnaphthalen-2-yl)carbonyl]amino}benzoic acid, CITRATE ANION, Nuclear receptor coactivator 1, ...
Authors:Nadendla, E.K, Teyssier, C, Germain, P, Delfosse, V, Bourguet, W.
Deposit date:2013-03-29
Release date:2014-03-19
Last modified:2024-02-28
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:An Unexpected Mode Of Binding Defines BMS948 as A Full Retinoic Acid Receptor beta (RAR beta , NR1B2) Selective Agonist.
Plos One, 10, 2015
4JYG
DownloadVisualize
BU of 4jyg by Molmil
Crystal structure of RARbeta LBD in complex with agonist BMS411 [4-{[(5,5-dimethyl-8-phenyl-5,6-dihydronaphthalen-2-yl)carbonyl]amino}benzoic acid]
Descriptor: 2-{2-[2-(2-{2-[2-(2-ETHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHOXY]-ETHOXY}-ETHANOL, 4-{[(5,5-dimethyl-8-phenyl-5,6-dihydronaphthalen-2-yl)carbonyl]amino}benzoic acid, CITRATE ANION, ...
Authors:Nadendla, E.K, Teyssier, C, Germain, P, Delfosse, V, Bourguet, W.
Deposit date:2013-03-29
Release date:2014-03-19
Last modified:2024-02-28
Method:X-RAY DIFFRACTION (2.35 Å)
Cite:An Unexpected Mode Of Binding Defines BMS948 as A Full Retinoic Acid Receptor beta (RAR beta , NR1B2) Selective Agonist.
Plos One, 10, 2015
5HT6
DownloadVisualize
BU of 5ht6 by Molmil
Crystal structure of the SET domain of the human MLL5 methyltransferase
Descriptor: Histone-lysine N-methyltransferase 2E
Authors:le Maire, A, Mas-y-Mas, S, Dumas, C, Lebedev, A.
Deposit date:2016-01-26
Release date:2016-11-16
Method:X-RAY DIFFRACTION (2.093 Å)
Cite:The Human Mixed Lineage Leukemia 5 (MLL5), a Sequentially and Structurally Divergent SET Domain-Containing Protein with No Intrinsic Catalytic Activity.
Plos One, 11, 2016
3KMZ
DownloadVisualize
BU of 3kmz by Molmil
Crystal structure of RARalpha ligand binding domain in complex with the inverse agonist BMS493 and a corepressor fragment
Descriptor: 4-{(E)-2-[5,5-dimethyl-8-(phenylethynyl)-5,6-dihydronaphthalen-2-yl]ethenyl}benzoic acid, GLYCEROL, Nuclear receptor corepressor 1, ...
Authors:Bourguet, W, le Maire, A.
Deposit date:2009-11-11
Release date:2010-06-02
Last modified:2023-11-22
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:A unique secondary-structure switch controls constitutive gene repression by retinoic acid receptor.
Nat.Struct.Mol.Biol., 17, 2010

217705

PDB entries from 2024-03-27

PDB statisticsPDBj update infoContact PDBjnumon