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1H4W
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STRUCTURE OF HUMAN TRYPSIN IV (BRAIN TRYPSIN)
Descriptor:TRYPSIN IVA, BENZAMIDINE, CALCIUM ION
Authors:Katona, G., Berglund, G.I., Hajdu, J., Graf, L., Szilagyi, L.
Deposit date:2001-05-15
Release date:2002-02-11
Last modified:2019-02-27
Method:X-RAY DIFFRACTION (1.7 Å)
Cite:Crystal structure reveals basis for the inhibitor resistance of human brain trypsin.
J. Mol. Biol., 315, 2002
1HLF
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BINDING OF GLUCOPYRANOSYLIDENE-SPIRO-THIOHYDANTOIN TO GLYCOGEN PHOSPHORYLASE B: KINETIC AND CRYSTALLOGRAPHIC STUD
Descriptor:GLYCOGEN PHOSPHORYLASE, PYRIDOXAL-5'-PHOSPHATE, 8,9,10-TRIHYDROXY-7-HYDROXYMETHYL-2-THIOXO-6-OXA-1,3-DIAZA-SPIRO[4.5]DECAN-4-ONE
Authors:Oikonomakos, N.G., Skamnaki, V.T., Docsa, T., Toth, B., Gergely, P., Osz, E., Szilagyi, L., Somsak, L.
Deposit date:2000-12-01
Release date:2000-12-13
Last modified:2017-10-04
Method:X-RAY DIFFRACTION (2.26 Å)
Cite:Kinetic and crystallographic studies of glucopyranosylidene spirothiohydantoin binding to glycogen phosphorylase B
BIOORG.MED.CHEM., 10, 2002
2F91
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1.2A RESOLUTION STRUCTURE OF A CRAYFISH TRYPSIN COMPLEXED WITH A PEPTIDE INHIBITOR, SGTI
Descriptor:hepatopancreas trypsin, Serine protease inhibitor I/II, CADMIUM ION, ...
Authors:Fodor, K., Harmat, V., Hetenyi, C., Kardos, J., Antal, J., Perczel, A., Patthy, A., Katona, G., Graf, L.
Deposit date:2005-12-05
Release date:2006-04-18
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (1.2 Å)
Cite:Enzyme:Substrate Hydrogen Bond Shortening during the Acylation Phase of Serine Protease Catalysis.
Biochemistry, 45, 2006
1GGN
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STRUCTURES OF GLYCOGEN PHOSPHORYLASE-INHIBITOR COMPLEXES AND THE IMPLICATIONS FOR STRUCTURE-BASED DRUG DESIGN
Descriptor:PROTEIN (GLYCOGEN PHOSPHORYLASE), BETA-D-GLUCOPYRANOSE SPIROHYDANTOIN, PYRIDOXAL-5'-PHOSPHATE
Authors:Watson, K.A., Tsitsanou, K.E., Gregoriou, M., Zographos, S.E., Skamnaki, V.T., Oikonomakos, N.G., Fleet, G.W., Johnson, L.N.
Deposit date:2000-08-29
Release date:2000-09-13
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (2.36 Å)
Cite:Kinetic and crystallographic studies of glucopyranosylidene spirothiohydantoin binding to glycogen phosphorylase B.
Bioorg.Med.Chem., 10, 2002
1AMH
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UNCOMPLEXED RAT TRYPSIN MUTANT WITH ASP 189 REPLACED WITH SER (D189S)
Descriptor:ANIONIC TRYPSIN, CALCIUM ION
Authors:Szabo, E., Bocskei, Z.S., Naray-Szabo, G., Graf, L.
Deposit date:1997-06-17
Release date:1997-12-24
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:The three-dimensional structure of Asp189Ser trypsin provides evidence for an inherent structural plasticity of the protease.
Eur.J.Biochem., 263, 1999
1KTI
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BINDING OF 100 MM N-ACETYL-N'-BETA-D-GLUCOPYRANOSYL UREA TO GLYCOGEN PHOSPHORYLASE B: KINETIC AND CRYSTALLOGRAPHIC STUDIES
Descriptor:GLYCOGEN PHOSPHORYLASE, MUSCLE FORM, N-ACETYL-N'-BETA-D-GLUCOPYRANOSYL UREA, ...
Authors:Oikonomakos, N.G., Kosmopoulou, M., Zographos, S.E., Leonidas, D.D., Chrysina, E.D., Somsak, L., Nagy, V., Praly, J.P., Docsa, T., Toth, B., Gergely, P.
Deposit date:2002-01-16
Release date:2002-01-30
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (1.97 Å)
Cite:Binding of N-acetyl-N'-beta-D-glucopyranosyl urea and N-benzoyl-N'-beta-D-glucopyranosyl urea to glycogen phosphorylase b: kinetic and crystallographic studies.
Eur.J.Biochem., 269, 2002