Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
Search by PDB author
1POI
DownloadVisualize
BU of 1poi by Molmil
CRYSTAL STRUCTURE OF GLUTACONATE COENZYME A-TRANSFERASE FROM ACIDAMINOCOCCUS FERMENTANS TO 2.55 ANGSTOMS RESOLUTION
Descriptor: COPPER (II) ION, GLUTACONATE COENZYME A-TRANSFERASE
Authors:Jacob, U, Mack, M, Clausen, T, Huber, R, Buckel, W, Messerschmidt, A.
Deposit date:1997-01-24
Release date:1998-03-18
Last modified:2024-02-14
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:Glutaconate CoA-transferase from Acidaminococcus fermentans: the crystal structure reveals homology with other CoA-transferases.
Structure, 5, 1997
1W12
DownloadVisualize
BU of 1w12 by Molmil
UROKINASE TYPE PLASMINOGEN ACTIVATOR
Descriptor: N-((1S)-4-{[AMINO(IMINO)METHYL]AMINO}-1-FORMYLBUTYL)-2-{(3R)-3-[(BENZYLSULFONYL)AMINO]-2-OXO-5-PHENYL-2,3-DIHYDRO-1H-1,4-BENZODIAZEPIN-1-YL}ACETAMIDE, UROKINASE-TYPE PLASMINOGEN ACTIVATOR
Authors:Jacob, U.
Deposit date:2004-06-15
Release date:2008-05-20
Last modified:2019-05-22
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:Crystals of Urokinase Type Plasminogen Activator Complexes Reveal the Binding Mode of Peptidomimetic Inhibitors.
J.Mol.Biol., 328, 2003
1W0Z
DownloadVisualize
BU of 1w0z by Molmil
Urokinase type plasminogen activator
Descriptor: N-(BUTYLSULFONYL)-D-SERYL-N-{4-[AMINO(IMINO)METHYL]BENZYL}-L-ALANINAMIDE, SULFATE ION, UROKINASE-TYPE PLASMINOGEN ACTIVATOR
Authors:Jacob, U.
Deposit date:2004-06-15
Release date:2008-05-20
Last modified:2019-09-18
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Crystals of urokinase type plasminogen activator complexes reveal the binding mode of peptidomimetic inhibitors.
J.Mol.Biol., 328, 2003
1W14
DownloadVisualize
BU of 1w14 by Molmil
UROKINASE TYPE PLASMINOGEN ACTIVATOR
Descriptor: N-[(2-PHENYLETHYL)SULFONYL]-D-SERYL-N-[(1S)-4-[(DIAMINOMETHYLENE)AMINO]-1-(HYDROXYMETHYL)BUTYL]-L-ALANINAMIDE, SULFATE ION, UROKINASE-TYPE PLASMINOGEN ACTIVATOR
Authors:Jacob, U.
Deposit date:2004-06-15
Release date:2008-05-20
Last modified:2019-05-22
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Crystals of Urokinase Type Plasminogen Activator Complexes Reveal the Binding Mode of Peptidomimetic Inhibitors.
J.Mol.Biol., 328, 2003
1W10
DownloadVisualize
BU of 1w10 by Molmil
Urokinase type plasminogen activator
Descriptor: N-(ISOBUTOXYCARBONYL)-D-SERYL-N-((1S)-4-{[AMINO(IMINO)METHYL]AMINO}-1-FORMYLBUTYL)-L-ALANINAMIDE, SULFATE ION, UROKINASE-TYPE PLASMINOGEN ACTIVATOR
Authors:Jacob, U.
Deposit date:2004-06-15
Release date:2008-05-20
Last modified:2019-09-18
Method:X-RAY DIFFRACTION (2 Å)
Cite:Crystals of urokinase type plasminogen activator complexes reveal the binding mode of peptidomimetic inhibitors.
J.Mol.Biol., 328, 2003
1W11
DownloadVisualize
BU of 1w11 by Molmil
UROKINASE TYPE PLASMINOGEN ACTIVATOR
Descriptor: N-(BENZYLSULFONYL)-D-SERYL-N-{4-[AMINO(IMINO)METHYL]BENZYL}-L-ALANINAMIDE, SULFATE ION, UROKINASE-TYPE PLASMINOGEN ACTIVATOR
Authors:Jacob, U.
Deposit date:2004-06-15
Release date:2008-05-20
Last modified:2019-10-09
Method:X-RAY DIFFRACTION (2 Å)
Cite:Crystals of Urokinase Type Plasminogen Activator Complexes Reveal the Binding Mode of Peptidomimetic Inhibitors.
J.Mol.Biol., 328, 2003
1W13
DownloadVisualize
BU of 1w13 by Molmil
UROKINASE TYPE PLASMINOGEN ACTIVATOR
Descriptor: N-(BENZYLSULFONYL)-D-SERYL-N-(4-{[AMINO(IMINO)METHYL]AMINO}BENZYL)-L-ALANINAMIDE, SULFATE ION, UROKINASE-TYPE PLASMINOGEN ACTIVATOR
Authors:Jacob, U.
Deposit date:2004-06-15
Release date:2008-05-20
Last modified:2019-05-22
Method:X-RAY DIFFRACTION (2 Å)
Cite:Crystals of Urokinase Type Plasminogen Activator Complexes Reveal the Binding Mode of Peptidomimetic Inhibitors.
J.Mol.Biol., 328, 2003
1VPE
DownloadVisualize
BU of 1vpe by Molmil
CRYSTALLOGRAPHIC ANALYSIS OF PHOSPHOGLYCERATE KINASE FROM THE HYPERTHERMOPHILIC BACTERIUM THERMOTOGA MARITIMA
Descriptor: 3-PHOSPHOGLYCERIC ACID, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, ...
Authors:Auerbach, G, Huber, R, Graettinger, M, Zaiss, K, Schurig, H, Jaenicke, R, Jacob, U.
Deposit date:1997-05-06
Release date:1998-06-17
Last modified:2022-12-21
Method:X-RAY DIFFRACTION (2 Å)
Cite:Closed structure of phosphoglycerate kinase from Thermotoga maritima reveals the catalytic mechanism and determinants of thermal stability.
Structure, 5, 1997
3CSP
DownloadVisualize
BU of 3csp by Molmil
Crystal structure of the DM2 mutant of myelin oligodendrocyte glycoprotein
Descriptor: Myelin-oligodendrocyte glycoprotein
Authors:Breithaupt, C, Schafer, B, Pellkofer, H, Huber, R, Linington, C, Jacob, U.
Deposit date:2008-04-10
Release date:2008-10-21
Last modified:2021-10-20
Method:X-RAY DIFFRACTION (1.7 Å)
Cite:Demyelinating myelin oligodendrocyte glycoprotein-specific autoantibody response is focused on one dominant conformational epitope region in rodents
J.Immunol., 181, 2008
2FCB
DownloadVisualize
BU of 2fcb by Molmil
HUMAN FC GAMMA RECEPTOR IIB ECTODOMAIN (CD32)
Descriptor: PROTEIN (FC GAMMA RIIB)
Authors:Sondermann, P, Huber, R, Jacob, U.
Deposit date:1999-01-07
Release date:2000-03-01
Last modified:2024-02-21
Method:X-RAY DIFFRACTION (1.74 Å)
Cite:Crystal structure of the soluble form of the human fcgamma-receptor IIb: a new member of the immunoglobulin superfamily at 1.7 A resolution.
EMBO J., 18, 1999
1SEP
DownloadVisualize
BU of 1sep by Molmil
MOUSE SEPIAPTERIN REDUCTASE COMPLEXED WITH NADP AND SEPIAPTERIN
Descriptor: BIOPTERIN, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, SEPIAPTERIN REDUCTASE
Authors:Auerbach, G, Herrmann, A, Guetlich, M, Fischer, M, Jacob, U, Bacher, A, Huber, R.
Deposit date:1997-05-23
Release date:1999-01-13
Last modified:2024-02-14
Method:X-RAY DIFFRACTION (1.95 Å)
Cite:The 1.25 A crystal structure of sepiapterin reductase reveals its binding mode to pterins and brain neurotransmitters.
EMBO J., 16, 1997
1VJA
DownloadVisualize
BU of 1vja by Molmil
Urokinase Plasminogen Activator B-Chain-JT463 Complex
Descriptor: N-(BENZYLSULFONYL)SERYL-N~1~-{4-[(Z)-AMINO(IMINO)METHYL]BENZYL}SERINAMIDE, SULFATE ION, plasminogen activator, ...
Authors:Schweinitz, A, Steinmetzer, T, Banke, I.J, Arlt, M.J.E, Stuerzebecher, A, Schuster, O, Geissler, A, Giersiefen, H, Zeslawska, E, Jacob, U, Kruger, A, Stuerzebecher, J.
Deposit date:2004-02-03
Release date:2004-06-22
Last modified:2023-08-23
Method:X-RAY DIFFRACTION (2 Å)
Cite:Design of novel and selective inhibitors of urokinase-type plasminogen activator with improved pharmacokinetic properties for use as antimetastatic agents
J.Biol.Chem., 279, 2004
1VJ9
DownloadVisualize
BU of 1vj9 by Molmil
Urokinase Plasminogen Activator B-Chain-JT464 Complex
Descriptor: N-(BENZYLSULFONYL)-L-SERYL-N~1~-{4-[AMINO(IMINO)METHYL]BENZYL}-O-BENZYL-L-SERINAMIDE, SULFATE ION, plasminogen activator, ...
Authors:Schweinitz, A, Steinmetzer, T, Banke, I.J, Arlt, M.J.E, Stuerzebecher, A, Schuster, O, Geissler, A, Giersiefen, H, Zeslawska, E, Jacob, U, Kruger, A, Stuerzebecher, J.
Deposit date:2004-02-03
Release date:2004-06-22
Last modified:2023-08-23
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:Design of novel and selective inhibitors of urokinase-type plasminogen activator with improved pharmacokinetic properties for use as antimetastatic agents
J.Biol.Chem., 279, 2004
1GV3
DownloadVisualize
BU of 1gv3 by Molmil
The 2.0 Angstrom resolution structure of the catalytic portion of a cyanobacterial membrane-bound manganese superoxide dismutase
Descriptor: MANGANESE (II) ION, MANGANESE SUPEROXIDE DISMUTASE
Authors:Atzenhofer, W, Regelsberger, G, Jacob, U, Huber, R, Peschek, G.A, Obinger, C.
Deposit date:2002-02-05
Release date:2002-08-08
Last modified:2023-12-13
Method:X-RAY DIFFRACTION (2 Å)
Cite:The 2.0A Resolution Structure of the Catalytic Portion of a Cyanobacterial Membrane-Bound Manganese Superoxide Dismutase
J.Mol.Biol., 321, 2002
1JHJ
DownloadVisualize
BU of 1jhj by Molmil
Crystal structure of the APC10/Doc1 subunit of the human anaphase-promoting complex
Descriptor: APC10, NICKEL (II) ION
Authors:Wendt, K.S, Vodermaier, H.C, Jacob, U, Gieffers, C, Gmachl, M, Peters, J.-M, Huber, R, Sondermann, P.
Deposit date:2001-06-28
Release date:2001-10-24
Last modified:2022-04-13
Method:X-RAY DIFFRACTION (1.6 Å)
Cite:Crystal structure of the APC10/DOC1 subunit of the human anaphase-promoting complex
Nat.Struct.Biol., 8, 2001
1PKQ
DownloadVisualize
BU of 1pkq by Molmil
Myelin Oligodendrocyte Glycoprotein-(8-18C5) Fab-complex
Descriptor: (8-18C5) chimeric Fab, heavy chain, light chain, ...
Authors:Breithaupt, C, Schubart, A, Zander, H, Skerra, A, Huber, R, Linington, C, Jacob, U.
Deposit date:2003-06-06
Release date:2003-07-15
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (3 Å)
Cite:Structural insights into the antigenicity of myelin oligodendrocyte glycoprotein
Proc.Natl.Acad.Sci.USA, 100, 2003
1PIX
DownloadVisualize
BU of 1pix by Molmil
Crystal structure of the carboxyltransferase subunit of the bacterial ion pump glutaconyl-coenzyme A decarboxylase
Descriptor: FORMIC ACID, Glutaconyl-CoA decarboxylase A subunit, SULFATE ION
Authors:Wendt, K.S, Schall, I, Huber, R, Buckel, W, Jacob, U.
Deposit date:2003-05-30
Release date:2003-08-05
Last modified:2024-02-14
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Crystal structure of the carboxyltransferase subunit of the bacterial sodium ion pump glutaconyl-coenzyme A decarboxylase
Embo J., 22, 2003
1PKO
DownloadVisualize
BU of 1pko by Molmil
Myelin Oligodendrocyte Glycoprotein (MOG)
Descriptor: Myelin Oligodendrocyte Glycoprotein
Authors:Breithaupt, C, Schubart, A, Zander, H, Skerra, A, Huber, R, Linington, C, Jacob, U.
Deposit date:2003-06-06
Release date:2003-07-15
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (1.45 Å)
Cite:Structural insights into the antigenicity of myelin oligodendrocyte glycoprotein
Proc.Natl.Acad.Sci.USA, 100, 2003
1QWJ
DownloadVisualize
BU of 1qwj by Molmil
The Crystal Structure of Murine CMP-5-N-Acetylneuraminic Acid Synthetase
Descriptor: CYTIDINE-5'-MONOPHOSPHATE-5-N-ACETYLNEURAMINIC ACID, cytidine monophospho-N-acetylneuraminic acid synthetase
Authors:Krapp, S, Muenster-Kuehnel, A.K, Kaiser, J.T, Huber, R, Tiralongo, J, Gerardy-Schahn, R, Jacob, U.
Deposit date:2003-09-02
Release date:2003-12-09
Last modified:2024-02-14
Method:X-RAY DIFFRACTION (2.8 Å)
Cite:The Crystal Structure of Murine CMP-5-N-acetylneuraminic Acid Synthetase
J.Mol.Biol., 334, 2003
1SC8
DownloadVisualize
BU of 1sc8 by Molmil
Urokinase Plasminogen Activator B-Chain-J435 Complex
Descriptor: N-(BENZYLSULFONYL)SERYL-N~1~-{4-[AMINO(IMINO)METHYL]BENZYL}GLYCINAMIDE, SULFATE ION, plasminogen activator, ...
Authors:Schweinitz, A, Steinmetzer, T, Banke, I.J, Arlt, M.J.E, Stuerzebecher, A, Schuster, O, Geissler, A, Giersiefen, H, Zeslawska, E, Jacob, U, Kruger, A, Stuerzebecher, J.
Deposit date:2004-02-12
Release date:2004-06-22
Last modified:2023-08-23
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:Design of novel and selective inhibitors of urokinase-type plasminogen activator with improved pharmacokinetic properties for use as antimetastatic agents
J.Biol.Chem., 279, 2004
1E4K
DownloadVisualize
BU of 1e4k by Molmil
CRYSTAL STRUCTURE OF SOLUBLE HUMAN IGG1 FC FRAGMENT-FC-GAMMA RECEPTOR III COMPLEX
Descriptor: FC FRAGMENT OF HUMAN IGG1, LOW AFFINITY IMMUNOGLOBULIN GAMMA FC RECEPTOR III, alpha-D-galactopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-6)-[2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-3)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Sondermann, P, Huber, R, Oosthuizen, V, Jacob, U.
Deposit date:2000-07-07
Release date:2000-08-06
Last modified:2023-12-13
Method:X-RAY DIFFRACTION (3.2 Å)
Cite:The 3.2A Crystal Structure of the Human Igg1 Fc Fragment-Fc-Gamma-Riii Complex
Nature, 406, 2000
1E4J
DownloadVisualize
BU of 1e4j by Molmil
Crystal structure of the soluble human Fc-gamma Receptor III
Descriptor: LOW AFFINITY IMMUNOGLOBULIN GAMMA FC RECEPTOR III
Authors:Sondermann, P, Huber, R, Jacob, U.
Deposit date:2000-07-07
Release date:2000-08-04
Last modified:2023-12-13
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:The 3.2-A Crystal Structure of the Human Igg1 Fc Fragment-Fc Gammariii Complex.
Nature, 406, 2000
1EJN
DownloadVisualize
BU of 1ejn by Molmil
UROKINASE PLASMINOGEN ACTIVATOR B-CHAIN INHIBITOR COMPLEX
Descriptor: N-(1-ADAMANTYL)-N'-(4-GUANIDINOBENZYL)UREA, SULFATE ION, UROKINASE-TYPE PLASMINOGEN ACTIVATOR
Authors:Sperl, S, Jacob, U, Arroyo de Prada, N, Stuerzebecher, J, Wilhelm, O.G, Bode, W, Magdolen, V, Huber, R, Moroder, L.
Deposit date:2000-04-22
Release date:2000-05-17
Last modified:2021-11-03
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:(4-aminomethyl)phenylguanidine derivatives as nonpeptidic highly selective inhibitors of human urokinase.
Proc.Natl.Acad.Sci.USA, 97, 2000
1F5L
DownloadVisualize
BU of 1f5l by Molmil
UROKINASE PLASMINOGEN ACTIVATOR B-CHAIN-AMILORIDE COMPLEX
Descriptor: 3,5-DIAMINO-N-(AMINOIMINOMETHYL)-6-CHLOROPYRAZINECARBOXAMIDE, SULFATE ION, UROKINASE-TYPE PLASMINOGEN ACTIVATOR
Authors:Zeslawska, E, Schweinitz, A, Karcher, A, Sondermann, P, Sperl, S, Sturzebecher, J, Jacob, U.
Deposit date:2000-06-15
Release date:2001-06-15
Last modified:2021-11-03
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:Crystals of the urokinase type plasminogen activator variant beta(c)-uPAin complex with small molecule inhibitors open the way towards structure-based drug design.
J.Mol.Biol., 301, 2000
1F5K
DownloadVisualize
BU of 1f5k by Molmil
UROKINASE PLASMINOGEN ACTIVATOR B-CHAIN-BENZAMIDINE COMPLEX
Descriptor: BENZAMIDINE, SULFATE ION, UROKINASE-TYPE PLASMINOGEN ACTIVATOR
Authors:Zeslawska, E, Schweinitz, A, Karcher, A, Sondermann, P, Sperl, S, Sturzebecher, J, Jacob, U.
Deposit date:2000-06-15
Release date:2001-06-15
Last modified:2021-11-03
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Crystals of the urokinase type plasminogen activator variant beta(c)-uPAin complex with small molecule inhibitors open the way towards structure-based drug design.
J.Mol.Biol., 301, 2000

 

12>

217705

PDB entries from 2024-03-27

PDB statisticsPDBj update infoContact PDBjnumon