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1FU3
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BU of 1fu3 by Molmil
THREE-DIMENSIONAL STRUCTURE IN SOLUTION OF THE SODIUM CHANNEL AGONIST/ANTAGONIST DELTA-CONOTOXIN TXVIA
Descriptor: DELTA-CONOTOXIN TXVIA
Authors:Kohno, T, Sasaki, T, Fainzilber, M, Sato, K.
Deposit date:2000-09-14
Release date:2002-09-20
Last modified:2022-02-23
Method:SOLUTION NMR
Cite:Three-dimensional solution structure of the sodium channel agonist/antagonist delta-conotoxin TxVIA.
J.Biol.Chem., 277, 2002
1OMG
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BU of 1omg by Molmil
NMR STUDY OF OMEGA-CONOTOXIN MVIIA
Descriptor: OMEGA-CONOTOXIN MVIIA
Authors:Kohno, T, Kim, J.-I, Kobayashi, K, Kodera, Y, Maeda, T, Sato, K.
Deposit date:1995-04-26
Release date:1996-04-03
Last modified:2022-02-23
Method:SOLUTION NMR
Cite:Three-dimensional structure in solution of the calcium channel blocker omega-conotoxin MVIIA.
Biochemistry, 34, 1995
1QCM
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BU of 1qcm by Molmil
AMYLOID BETA PEPTIDE (25-35), NMR, 20 STRUCTURES
Descriptor: AMYLOID BETA PEPTIDE
Authors:Kohno, T, Kobayashi, K, Maeda, T, Sato, K, Takashima, A.
Deposit date:1996-07-19
Release date:1997-07-07
Last modified:2022-03-02
Method:SOLUTION NMR
Cite:Three-dimensional structures of the amyloid beta peptide (25-35) in membrane-mimicking environment.
Biochemistry, 35, 1996
1V5A
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BU of 1v5a by Molmil
Solution Structure of Covalitoxin I
Descriptor: Covalitoxin-I
Authors:Kohno, T, Sasaki, T, Sato, K.
Deposit date:2003-11-21
Release date:2005-03-01
Last modified:2023-12-27
Method:SOLUTION NMR
Cite:Solution Structure of Covalitoxin I
To be Published
2D1O
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BU of 2d1o by Molmil
Stromelysin-1 (MMP-3) complexed to a hydroxamic acid inhibitor
Descriptor: CALCIUM ION, SM-25453, Stromelysin-1, ...
Authors:Kohno, T, Hochigai, H, Yamashita, E, Tsukihara, T, Kanaoka, M.
Deposit date:2005-08-30
Release date:2006-06-27
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.02 Å)
Cite:Crystal structures of the catalytic domain of human stromelysin-1 (MMP-3) and collagenase-3 (MMP-13) with a hydroxamic acid inhibitor SM-25453
Biochem.Biophys.Res.Commun., 344, 2006
2D1N
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BU of 2d1n by Molmil
Collagenase-3 (MMP-13) complexed to a hydroxamic acid inhibitor
Descriptor: CALCIUM ION, Collagenase 3, SM-25453, ...
Authors:Kohno, T, Hochigai, H, Yamashita, E, Tsukihara, T, Kanaoka, M.
Deposit date:2005-08-29
Release date:2006-06-27
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.37 Å)
Cite:Crystal structures of the catalytic domain of human stromelysin-1 (MMP-3) and collagenase-3 (MMP-13) with a hydroxamic acid inhibitor SM-25453
Biochem.Biophys.Res.Commun., 344, 2006
4PK5
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BU of 4pk5 by Molmil
Crystal structure of the indoleamine 2,3-dioxygenagse 1 (IDO1) complexed with Amg-1
Descriptor: Indoleamine 2,3-dioxygenase 1, N-(1,3-benzodioxol-5-yl)-2-{[5-(4-methylphenyl)[1,3]thiazolo[2,3-c][1,2,4]triazol-3-yl]sulfanyl}acetamide, PROTOPORPHYRIN IX CONTAINING FE
Authors:Kohno, T, Tojo, S, Ishii, T.
Deposit date:2014-05-13
Release date:2014-09-03
Last modified:2020-01-29
Method:X-RAY DIFFRACTION (2.79 Å)
Cite:Crystal Structures and Structure-Activity Relationships of Imidazothiazole Derivatives as IDO1 Inhibitors.
Acs Med.Chem.Lett., 5, 2014
4PK6
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BU of 4pk6 by Molmil
Crystal structure of the indoleamine 2,3-dioxygenagse 1 (IDO1) complexed with imidazothiazole derivative
Descriptor: Indoleamine 2,3-dioxygenase 1, N-[2-(3-chlorophenyl)ethyl]-3-(4-methylphenyl)imidazo[2,1-b][1,3]thiazole-5-carboxamide, PROTOPORPHYRIN IX CONTAINING FE
Authors:Kohno, T, Tojo, S, Ishii, T, Kamioka, S.
Deposit date:2014-05-13
Release date:2014-09-03
Last modified:2017-10-04
Method:X-RAY DIFFRACTION (3.45 Å)
Cite:Crystal Structures and Structure-Activity Relationships of Imidazothiazole Derivatives as IDO1 Inhibitors.
Acs Med.Chem.Lett., 5, 2014
2D52
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BU of 2d52 by Molmil
Pentaketide chromone synthase (M207G mutant complexed with Coa)
Descriptor: COENZYME A, pentaketide chromone synthase
Authors:Kohno, T, Morita, H.
Deposit date:2005-10-27
Release date:2006-11-14
Last modified:2021-11-10
Method:X-RAY DIFFRACTION (1.6 Å)
Cite:Structural Insight into Chain-Length Control and Product Specificity of Pentaketide Chromone Synthase from Aloe arborescens
Chem.Biol., 14, 2007
2D51
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BU of 2d51 by Molmil
Pentaketide chromone synthase (M207G mutant)
Descriptor: pentaketide chromone synthase
Authors:Kohno, T, Morita, H.
Deposit date:2005-10-27
Release date:2006-11-14
Last modified:2021-11-10
Method:X-RAY DIFFRACTION (1.6 Å)
Cite:Structural Insight into Chain-Length Control and Product Specificity of Pentaketide Chromone Synthase from Aloe arborescens
Chem.Biol., 14, 2007
1A13
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BU of 1a13 by Molmil
G PROTEIN-BOUND CONFORMATION OF MASTOPARAN-X, NMR, 14 STRUCTURES
Descriptor: MASTOPARAN-X
Authors:Kusunoki, H, Wakamatsu, K, Sato, K, Miyazawa, T, Kohno, T.
Deposit date:1997-12-20
Release date:1999-01-13
Last modified:2022-02-16
Method:SOLUTION NMR
Cite:G protein-bound conformation of mastoparan-X: heteronuclear multidimensional transferred nuclear overhauser effect analysis of peptide uniformly enriched with 13C and 15N.
Biochemistry, 37, 1998
6FEK
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BU of 6fek by Molmil
Oncogenic point mutation of RET receptor tyrosine kinase
Descriptor: ADENOSINE, FORMIC ACID, Proto-oncogene tyrosine-protein kinase receptor Ret
Authors:McDonald, N.Q, Kohno, T.
Deposit date:2018-01-02
Release date:2018-02-28
Last modified:2018-05-02
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:A secondary RET mutation in the activation loop conferring resistance to vandetanib.
Nat Commun, 9, 2018
7EN4
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BU of 7en4 by Molmil
Multi-state structure determination and dynamics analysis elucidate a new ubiquitin-recognition mechanism of yeast ubiquitin C-terminal hydrolase.
Descriptor: Ubiquitin carboxyl-terminal hydrolase YUH1
Authors:Okada, M, Tateishi, Y, Nojiri, E, Mikawa, T, Rajesh, S, Ogasawa, H, Ueda, T, Yagi, H, Kohno, T, Kigawa, T, Shimada, I, Guentert, P, Yutaka, I, Ikeya, T.
Deposit date:2021-04-15
Release date:2022-04-20
Last modified:2023-06-14
Method:SOLUTION NMR
Cite:Multi-state structure determination and dynamics analysis elucidate a new ubiquitin-recognition mechanism of yeast ubiquitin C-terminal hydrolase.
To Be Published
4ZKF
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BU of 4zkf by Molmil
Crystal structure of human phosphodiesterase 12
Descriptor: 2',5'-phosphodiesterase 12, MAGNESIUM ION
Authors:Kim, S.Y, Kohno, T, Mori, T, Kitano, K, Hakoshima, T.
Deposit date:2015-04-30
Release date:2015-06-17
Last modified:2024-03-20
Method:X-RAY DIFFRACTION (1.82 Å)
Cite:Crystal structure of human phosphodiesterase
To Be Published
1NC8
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BU of 1nc8 by Molmil
HIGH-RESOLUTION SOLUTION NMR STRUCTURE OF THE MINIMAL ACTIVE DOMAIN OF THE HUMAN IMMUNODEFICIENCY VIRUS TYPE-2 NUCLEOCAPSID PROTEIN, 15 STRUCTURES
Descriptor: NUCLEOCAPSID PROTEIN, ZINC ION
Authors:Kodera, Y, Sato, K, Tsukahara, T, Komatsu, H, Maeda, T, Kohno, T.
Deposit date:1998-05-14
Release date:1999-05-25
Last modified:2022-02-23
Method:SOLUTION NMR
Cite:High-resolution solution NMR structure of the minimal active domain of the human immunodeficiency virus type-2 nucleocapsid protein.
Biochemistry, 37, 1998
1F3K
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BU of 1f3k by Molmil
THREE-DIMENSIONAL SOLUTION STRUCTURE OF OMEGA-CONOTOXIN TXVII, AN L-TYPE CALCIUM CHANNEL BLOCKER
Descriptor: OMEGA-CONOTOXIN TXVII
Authors:Kobayashi, K, Sasaki, T, Sato, K, Kohno, T.
Deposit date:2000-06-05
Release date:2000-12-13
Last modified:2022-02-16
Method:SOLUTION NMR
Cite:Three-dimensional solution structure of omega-conotoxin TxVII, an L-type calcium channel blocker.
Biochemistry, 39, 2000
1HD0
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BU of 1hd0 by Molmil
HETEROGENEOUS NUCLEAR RIBONUCLEOPROTEIN D0 (HNRNP D0 RBD1), NMR
Descriptor: PROTEIN (HETEROGENEOUS NUCLEAR RIBONUCLEOPROTEIN D0)
Authors:Nagata, T, Kurihara, Y, Matsuda, G, Saeki, J, Kohno, T, Yanagida, Y, Ishikawa, F, Uesugi, S, Katahira, M.
Deposit date:1999-05-18
Release date:2000-05-18
Last modified:2023-12-27
Method:SOLUTION NMR
Cite:Structure and interactions with RNA of the N-terminal UUAG-specific RNA-binding domain of hnRNP D0.
J.Mol.Biol., 287, 1999
1J1B
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BU of 1j1b by Molmil
Binary complex structure of human tau protein kinase I with AMPPNP
Descriptor: Glycogen synthase kinase-3 beta, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER
Authors:Aoki, M, Yokota, T, Sugiura, I, Sasaki, C, Hasegawa, T, Okumura, C, Kohno, T, Sugio, S, Matsuzaki, T.
Deposit date:2002-12-03
Release date:2003-12-03
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Structural insight into nucleotide recognition in tau-protein kinase I/glycogen synthase kinase 3 beta.
Acta Crystallogr.,Sect.D, 60, 2004
1J1C
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BU of 1j1c by Molmil
Binary complex structure of human tau protein kinase I with ADP
Descriptor: ADENOSINE-5'-DIPHOSPHATE, Glycogen synthase kinase-3 beta, MAGNESIUM ION
Authors:Aoki, M, Yokota, T, Sugiura, I, Sasaki, C, Hasegawa, T, Okumura, C, Kohno, T, Sugio, S, Matsuzaki, T.
Deposit date:2002-12-03
Release date:2003-12-03
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:Structural insight into nucleotide recognition in tau-protein kinase I/glycogen synthase kinase 3 beta.
Acta Crystallogr.,Sect.D, 60, 2004
2EV8
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BU of 2ev8 by Molmil
Solution structure of the erythroid p55 PDZ domain
Descriptor: 55 kDa erythrocyte membrane protein
Authors:Kusunoki, H, Kohno, T.
Deposit date:2005-10-31
Release date:2006-10-10
Last modified:2022-03-09
Method:SOLUTION NMR
Cite:Solution structure of human erythroid p55 PDZ domain
Proteins, 64, 2006
2MLO
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BU of 2mlo by Molmil
Human CCR2 Membrane-Proximal C-Terminal Region (PRO-C) in a Membrane bound form
Descriptor: MCP-1 receptor
Authors:Esaki, K, Yoshinaga, S, Tsuji, T, Toda, E, Terashima, Y, Saitoh, T, Kohda, D, Kohno, T, Osawa, M, Ueda, T, Shimada, I, Matsushima, K, Terasawa, H.
Deposit date:2014-03-04
Release date:2014-10-08
Last modified:2023-06-14
Method:SOLUTION NMR
Cite:Structural basis for the binding of the membrane-proximal C-terminal region of chemokine receptor CCR2 with the cytosolic regulator FROUNT.
Febs J., 281, 2014
3AQP
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BU of 3aqp by Molmil
Crystal structure of SecDF, a translocon-associated membrane protein, from Thermus thrmophilus
Descriptor: Probable SecDF protein-export membrane protein
Authors:Tsukazaki, T, Mori, H, Echizen, Y, Ishitani, R, Fukai, S, Tanaka, T, Perederina, A, Vassylyev, D.G, Kohno, T, Ito, K, Nureki, O.
Deposit date:2010-11-16
Release date:2011-05-18
Last modified:2024-03-13
Method:X-RAY DIFFRACTION (3.3 Å)
Cite:Structure and function of a membrane component SecDF that enhances protein export
Nature, 474, 2011
2MLQ
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BU of 2mlq by Molmil
Human CCR2 Membrane-Proximal C-Terminal Region (PRO-C) in a frount bound form
Descriptor: MCP-1 receptor
Authors:Esaki, K, Yoshinaga, S, Tsuji, T, Toda, E, Terashima, Y, Saitoh, T, Kohda, D, Kohno, T, Osawa, M, Ueda, T, Shimada, I, Matsushima, K, Terasawa, H.
Deposit date:2014-03-04
Release date:2014-10-08
Last modified:2023-06-14
Method:SOLUTION NMR
Cite:Structural basis for the binding of the membrane-proximal C-terminal region of chemokine receptor CCR2 with the cytosolic regulator FROUNT.
Febs J., 281, 2014
2RRN
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BU of 2rrn by Molmil
Solution structure of SecDF periplasmic domain P4
Descriptor: Probable SecDF protein-export membrane protein
Authors:Tanaka, T, Tsukazaki, T, Echizen, Y, Nureki, O, Kohno, T.
Deposit date:2011-01-30
Release date:2011-05-18
Last modified:2011-12-28
Method:SOLUTION NMR
Cite:Structure and function of a membrane component SecDF that enhances protein export
Nature, 474, 2011
2ZJZ
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BU of 2zjz by Molmil
Structure of the K349P mutant of Gi alpha 1 subunit bound to GDP
Descriptor: GUANOSINE-5'-DIPHOSPHATE, Guanine nucleotide-binding protein G(i), alpha-1 subunit
Authors:Morikawa, T, Muroya, A, Sugio, S, Wakamatsu, K, Kohno, T.
Deposit date:2008-03-11
Release date:2009-03-24
Last modified:2023-11-01
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:How GPCRs activate G proteins: Structural changes from C-terminal tail to GDP binding pocket
To be Published

 

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