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2GX5
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BU of 2gx5 by Molmil
N-terminal GAF domain of transcriptional pleiotropic repressor CodY
Descriptor: CYCLIC GUANOSINE MONOPHOSPHATE, GLYCEROL, GTP-sensing transcriptional pleiotropic repressor codY, ...
Authors:Wilkinson, A.J, Levdikov, V.M, Blagova, E.V.
Deposit date:2006-05-08
Release date:2007-04-17
Last modified:2023-08-30
Method:X-RAY DIFFRACTION (1.74 Å)
Cite:The structure of CodY, a GTP- and isoleucine-responsive regulator of stationary phase and virulence in gram-positive bacteria.
J.Biol.Chem., 281, 2006
5LOE
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BU of 5loe by Molmil
Structure of full length Cody from Bacillus subtilis in complex with Ile
Descriptor: GTP-sensing transcriptional pleiotropic repressor CodY, ISOLEUCINE
Authors:Wilkinson, A.J, Levdikov, V.M, Blagova, E.V.
Deposit date:2016-08-09
Release date:2017-01-11
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (3 Å)
Cite:Structure of the Branched-chain Amino Acid and GTP-sensing Global Regulator, CodY, from Bacillus subtilis.
J. Biol. Chem., 292, 2017
5LOJ
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BU of 5loj by Molmil
Structure of full length unliganded CodY from Bacillus subtilis
Descriptor: GTP-sensing transcriptional pleiotropic repressor CodY
Authors:Wilkinson, A.J, Levdikov, V.M, Blagova, E.V.
Deposit date:2016-08-09
Release date:2017-01-11
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (3.71 Å)
Cite:Structure of the Branched-chain Amino Acid and GTP-sensing Global Regulator, CodY, from Bacillus subtilis.
J. Biol. Chem., 292, 2017
5LNH
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BU of 5lnh by Molmil
Structure of full length Unliganded CodY from Bacillus subtilis
Descriptor: GTP-sensing transcriptional pleiotropic repressor CodY, SULFATE ION
Authors:Wilkinson, A.J, Levdikov, V.M, Blagova, E.V.
Deposit date:2016-08-04
Release date:2017-01-11
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (3 Å)
Cite:Structure of the Branched-chain Amino Acid and GTP-sensing Global Regulator, CodY, from Bacillus subtilis.
J. Biol. Chem., 292, 2017
5LOO
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BU of 5loo by Molmil
Structure of full length unliganded CodY from Bacillus subtilis
Descriptor: GTP-sensing transcriptional pleiotropic repressor CodY
Authors:Wilkinson, A.J, Levdikov, V.M, Blagova, E.V.
Deposit date:2016-08-09
Release date:2017-01-11
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (4.5 Å)
Cite:Structure of the Branched-chain Amino Acid and GTP-sensing Global Regulator, CodY, from Bacillus subtilis.
J. Biol. Chem., 292, 2017
8BPT
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BU of 8bpt by Molmil
Crystal structure of the second bromodomain of BRD5 from Leishmania donovani
Descriptor: Bromo domain-containing protein
Authors:Wilkinson, A.J, Dodson, E.J, Jones, N.G, Borgia, J.
Deposit date:2022-11-17
Release date:2023-09-27
Last modified:2023-11-22
Method:X-RAY DIFFRACTION (1.6 Å)
Cite:Bromodomain Factor 5 as a Target for Antileishmanial Drug Discovery.
Acs Infect Dis., 9, 2023
2HGV
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BU of 2hgv by Molmil
N-terminal GAF domain of transcriptional pleiotropic repressor CodY
Descriptor: GTP-sensing transcriptional pleiotropic repressor codY, VALINE
Authors:Wilkinson, A.J, Levdikov, V.M, Blagova, E.V.
Deposit date:2006-06-27
Release date:2006-08-15
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:The Structure of CodY, a GTP- and Isoleucine-responsive Regulator of Stationary Phase and Virulence in Gram-positive Bacteria
J.Biol.Chem., 281, 2006
1B3G
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BU of 1b3g by Molmil
OLIGO-PEPTIDE BINDING PROTEIN (OPPA) COMPLEXED WITH KIK
Descriptor: PROTEIN (LYS-ILE-LYS), PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN), URANYL (VI) ION
Authors:Tame, J.R.H, Wilkinson, A.J.
Deposit date:1998-12-14
Release date:1998-12-16
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (2 Å)
Cite:Crystallographic and calorimetric analysis of peptide binding to OppA protein.
J.Mol.Biol., 291, 1999
1B40
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BU of 1b40 by Molmil
OLIGO-PEPTIDE BINDING PROTEIN (OPPA) COMPLEXED WITH KFK
Descriptor: PROTEIN (LYS-PHE-LYS), PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN), URANYL (VI) ION
Authors:Tame, J.R.H, Wilkinson, A.J.
Deposit date:1998-11-23
Release date:1999-01-13
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Crystallographic and calorimetric analysis of peptide binding to OppA protein.
J.Mol.Biol., 291, 1999
1B05
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BU of 1b05 by Molmil
Structure of oligo-peptide binding protein complexed with LYS-CYS-LYS
Descriptor: PEPTIDE LYS-CYS-LYS, PERIPLASMIC OLIGOPEPTIDE-BINDING PROTEIN, URANIUM ATOM
Authors:Tame, J.R.H, Wilkinson, A.J.
Deposit date:1998-11-20
Release date:1998-11-25
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (2 Å)
Cite:Crystallographic and calorimetric analysis of peptide binding to OppA protein.
J.Mol.Biol., 291, 1999
1B4Z
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BU of 1b4z by Molmil
OLIGO-PEPTIDE BINDING PROTEIN (OPPA) COMPLEXED WITH KDK
Descriptor: ACETATE ION, PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN), PROTEIN (PEPTIDE LYS-ASP-LYS), ...
Authors:Tame, J.R.H, Sleigh, S.H, Wilkinson, A.J.
Deposit date:1999-01-04
Release date:1999-01-13
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (1.75 Å)
Cite:Crystallographic and calorimetric analysis of peptide binding to OppA protein.
J.Mol.Biol., 291, 1999
1B5J
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BU of 1b5j by Molmil
OLIGO-PEPTIDE BINDING PROTEIN (OPPA) COMPLEXED WITH KQK
Descriptor: PROTEIN (LYS-GLN-LYS), PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN), URANIUM ATOM
Authors:Tame, J.R.H, Wilkinson, A.J.
Deposit date:1999-01-06
Release date:1999-01-13
Last modified:2023-08-02
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Crystallographic and calorimetric analysis of peptide binding to OppA protein.
J.Mol.Biol., 291, 1999
1B51
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BU of 1b51 by Molmil
OLIGO-PEPTIDE BINDING PROTEIN (OPPA) COMPLEXED WITH KSK
Descriptor: PROTEIN (LYS-SER-LYS), PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN), URANYL (VI) ION
Authors:Tame, J.R.H, Wilkinson, A.J.
Deposit date:1999-01-11
Release date:1999-01-20
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Crystallographic and calorimetric analysis of peptide binding to OppA protein.
J.Mol.Biol., 291, 1999
1B9J
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BU of 1b9j by Molmil
OLIGO-PEPTIDE BINDING PROTEIN (OPPA) COMPLEXED WITH KLK
Descriptor: PROTEIN (LYS-LEU-LYS), PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN), URANYL (VI) ION
Authors:Tame, J.R.H, Wilkinson, A.J.
Deposit date:1999-02-11
Release date:1999-02-22
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Crystallographic and calorimetric analysis of peptide binding to OppA protein.
J.Mol.Biol., 291, 1999
1B58
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BU of 1b58 by Molmil
OLIGO-PEPTIDE BINDING PROTEIN (OPPA) COMPLEXED WITH KYK
Descriptor: PROTEIN (LYS-TYR-LYS), PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN), URANYL (VI) ION
Authors:Tame, J.R.H, Wilkinson, A.J.
Deposit date:1999-01-12
Release date:1999-01-20
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Crystallographic and calorimetric analysis of peptide binding to OppA protein.
J.Mol.Biol., 291, 1999
1B3L
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BU of 1b3l by Molmil
OLIGO-PEPTIDE BINDING PROTEIN (OPPA) COMPLEXED WITH KGK
Descriptor: PROTEIN (LYS-GLY-LYS), PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN), URANYL (VI) ION
Authors:Tame, J.R.H, Wilkinson, A.J.
Deposit date:1998-12-14
Release date:1998-12-16
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (2 Å)
Cite:Crystallographic and calorimetric analysis of peptide binding to OppA protein.
J.Mol.Biol., 291, 1999
1B46
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BU of 1b46 by Molmil
OLIGO-PEPTIDE BINDING PROTEIN (OPPA) COMPLEXED WITH KPK
Descriptor: ACETATE ION, PROTEIN (LYS-PRO-LYS), PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN), ...
Authors:Tame, J.R.H, Sleigh, S.H, Wilkinson, A.J.
Deposit date:1999-01-05
Release date:1999-01-13
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Crystallographic and calorimetric analysis of peptide binding to OppA protein.
J.Mol.Biol., 291, 1999
1B52
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BU of 1b52 by Molmil
OLIGO-PEPTIDE BINDING PROTEIN (OPPA) COMPLEXED WITH KTK
Descriptor: PROTEIN (LYS-THR-LYS), PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN), URANYL (VI) ION
Authors:Tame, J.R.H, Wilkinson, A.J.
Deposit date:1999-01-11
Release date:1999-01-20
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Crystallographic and calorimetric analysis of peptide binding to OppA protein.
J.Mol.Biol., 291, 1999
1B32
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BU of 1b32 by Molmil
OLIGO-PEPTIDE BINDING PROTEIN (OPPA) COMPLEXED WITH KMK
Descriptor: ACETATE ION, PROTEIN (LYS-MET-LYS), PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN), ...
Authors:Tame, J.R.H, Wilkinson, A.J.
Deposit date:1998-12-15
Release date:1998-12-23
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (1.75 Å)
Cite:Crystallographic and calorimetric analysis of peptide binding to OppA protein.
J.Mol.Biol., 291, 1999
1B3F
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BU of 1b3f by Molmil
OLIGO-PEPTIDE BINDING PROTEIN (OPPA) COMPLEXED WITH KHK
Descriptor: PROTEIN (LYS-HIS-LYS), PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN), URANYL (VI) ION
Authors:Tame, J.R.H, Wilkinson, A.J.
Deposit date:1998-12-14
Release date:1998-12-16
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Crystallographic and calorimetric analysis of peptide binding to OppA protein.
J.Mol.Biol., 291, 1999
1B5I
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BU of 1b5i by Molmil
OLIGO-PEPTIDE BINDING PROTEIN (OPPA) COMPLEXED WITH KNK
Descriptor: PROTEIN (LYS-ASN-LYS), PROTEIN (OLIGO-PEPTIDE BINDING PROTEIN), URANIUM ATOM
Authors:Tame, J.R.H, Wilkinson, A.J.
Deposit date:1999-01-06
Release date:1999-01-13
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Crystallographic and calorimetric analysis of peptide binding to OppA protein.
J.Mol.Biol., 291, 1999
2RKM
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BU of 2rkm by Molmil
STRUCTURE OF OPPA COMPLEXED WITH LYS-LYS
Descriptor: LYSINE, OLIGO-PEPTIDE BINDING PROTEIN, URANYL (VI) ION
Authors:Sleigh, S.H, Tame, J.R.H, Wilkinson, A.J.
Deposit date:1997-03-25
Release date:1997-07-29
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Peptide binding in OppA, the crystal structures of the periplasmic oligopeptide binding protein in the unliganded form and in complex with lysyllysine.
Biochemistry, 36, 1997
2OLB
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BU of 2olb by Molmil
OLIGOPEPTIDE BINDING PROTEIN (OPPA) COMPLEXED WITH TRI-LYSINE
Descriptor: ACETATE ION, OLIGO-PEPTIDE BINDING PROTEIN, TRIPEPTIDE LYS-LYS-LYS, ...
Authors:Tame, J, Wilkinson, A.J.
Deposit date:1995-09-10
Release date:1996-01-29
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (1.4 Å)
Cite:The crystal structures of the oligopeptide-binding protein OppA complexed with tripeptide and tetrapeptide ligands.
Structure, 3, 1995
5A28
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BU of 5a28 by Molmil
Leishmania major N-myristoyltransferase in complex with a chlorophenyl 1,3,4-oxadiazole inhibitor.
Descriptor: 4-(4-chloro-2-{5-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,3,4-oxadiazol-2-yl}phenoxy)piperidine, GLYCYLPEPTIDE N-TETRADECANOYLTRANSFERASE, MAGNESIUM ION, ...
Authors:Rackham, M.D, Yu, Z, Brannigan, J.A, Heal, W.P, Paape, D, Barker, K.V, Wilkinson, A.J, Smith, D.F, Tate, E.W, Leatherbarrow, R.J.
Deposit date:2015-05-15
Release date:2016-03-23
Method:X-RAY DIFFRACTION (1.48 Å)
Cite:Discovery of High Affinity Inhibitors of Leishmania Donovani N-Myristoyltransferase.
Medchemcomm, 6, 2015
5A27
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BU of 5a27 by Molmil
Leishmania major N-myristoyltransferase in complex with a chlorophenyl 1,2,4-oxadiazole inhibitor.
Descriptor: 5-chloranyl-N-[2-(3-methoxyphenyl)ethanimidoyl]-2-piperidin-4-yloxy-benzamide, GLYCYLPEPTIDE N-TETRADECANOYLTRANSFERASE, MAGNESIUM ION, ...
Authors:Rackham, M.D, Yu, Z, Brannigan, J.A, Heal, W.P, Paape, D, Barker, K.V, Wilkinson, A.J, Smith, D.F, Tate, E.W, Leatherbarrow, R.J.
Deposit date:2015-05-15
Release date:2016-03-23
Method:X-RAY DIFFRACTION (1.37 Å)
Cite:Discovery of High Affinity Inhibitors of Leishmania Donovani N-Myristoyltransferase.
Medchemcomm, 6, 2015

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