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3MO0
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BU of 3mo0 by Molmil
Human G9a-like (GLP, also known as EHMT1) in complex with inhibitor E11
Descriptor: 1,2-ETHANEDIOL, Histone-lysine N-methyltransferase, H3 lysine-9 specific 5, ...
Authors:Chang, Y, Horton, J.R, Cheng, X.
Deposit date:2010-04-22
Release date:2010-06-30
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (2.78 Å)
Cite:Adding a lysine mimic in the design of potent inhibitors of histone lysine methyltransferases.
J.Mol.Biol., 400, 2010
3MO5
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BU of 3mo5 by Molmil
Human G9a-like (GLP, also known as EHMT1) in complex with inhibitor E72
Descriptor: 7-[(5-aminopentyl)oxy]-N~4~-[1-(5-aminopentyl)piperidin-4-yl]-N~2~-[3-(dimethylamino)propyl]-6-methoxyquinazoline-2,4-diamine, Histone-lysine N-methyltransferase, H3 lysine-9 specific 5, ...
Authors:Chang, Y, Horton, J.R, Cheng, X.
Deposit date:2010-04-22
Release date:2010-06-30
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (2.14 Å)
Cite:Adding a lysine mimic in the design of potent inhibitors of histone lysine methyltransferases.
J.Mol.Biol., 400, 2010
3MO2
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BU of 3mo2 by Molmil
human G9a-like (GLP, also known as EHMT1) in complex with inhibitor E67
Descriptor: 7-[(5-aminopentyl)oxy]-N~4~-(1-benzylpiperidin-4-yl)-N~2~-[3-(dimethylamino)propyl]-6-methoxyquinazoline-2,4-diamine, Histone-lysine N-methyltransferase, H3 lysine-9 specific 5, ...
Authors:Chang, Y, Horton, J.R, Cheng, X.
Deposit date:2010-04-22
Release date:2010-06-30
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (2.49 Å)
Cite:Adding a lysine mimic in the design of potent inhibitors of histone lysine methyltransferases.
J.Mol.Biol., 400, 2010
3SW9
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BU of 3sw9 by Molmil
GLP (G9a-like protein) SET domain in complex with Dnmt3aK44me0 peptide
Descriptor: DNA (cytosine-5)-methyltransferase 3A, Histone-lysine N-methyltransferase EHMT1, SINEFUNGIN, ...
Authors:Chang, Y, Horton, J.R, Zhang, X, Cheng, X.
Deposit date:2011-07-13
Release date:2011-12-07
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (3.05 Å)
Cite:MPP8 mediates the interactions between DNA methyltransferase Dnmt3a and H3K9 methyltransferase GLP/G9a.
Nat Commun, 2, 2011
3SVM
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BU of 3svm by Molmil
Human MPP8 - human DNMT3AK47me2 peptide
Descriptor: DNA (cytosine-5)-methyltransferase 3A, M-phase phosphoprotein 8
Authors:Chang, Y, Horton, J.R, Zhang, X, Cheng, X.
Deposit date:2011-07-12
Release date:2011-11-30
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (2.31 Å)
Cite:MPP8 mediates the interactions between DNA methyltransferase Dnmt3a and H3K9 methyltransferase GLP/G9a.
Nat Commun, 2, 2011
3SWC
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BU of 3swc by Molmil
GLP (G9a-like protein) SET domain in complex with Dnmt3aK44me2 peptide
Descriptor: DNA (cytosine-5)-methyltransferase 3A, Histone-lysine N-methyltransferase EHMT1, S-ADENOSYL-L-HOMOCYSTEINE, ...
Authors:Chang, Y, Horton, J.R, Zhang, X, Cheng, X.
Deposit date:2011-07-13
Release date:2011-11-30
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (2.332 Å)
Cite:MPP8 mediates the interactions between DNA methyltransferase Dnmt3a and H3K9 methyltransferase GLP/G9a.
Nat Commun, 2, 2011
3OPW
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BU of 3opw by Molmil
Crystal Structure of the Rph1 catalytic core
Descriptor: DNA damage-responsive transcriptional repressor RPH1
Authors:Chang, Y, Wu, J, Tong, X, Zhou, J, Ding, J.
Deposit date:2010-09-02
Release date:2010-12-22
Last modified:2024-03-20
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:Crystal structure of the catalytic core of Saccharomyces cerevesiae histone demethylase Rph1: insights into the substrate specificity and catalytic mechanism
Biochem.J., 433, 2011
3OPT
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BU of 3opt by Molmil
Crystal structure of the Rph1 catalytic core with a-ketoglutarate
Descriptor: 2-OXOGLUTARIC ACID, DNA damage-responsive transcriptional repressor RPH1, NICKEL (II) ION
Authors:Chang, Y, Wu, J, Tong, X, Zhou, J, Ding, J.
Deposit date:2010-09-02
Release date:2010-12-22
Last modified:2024-03-20
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Crystal structure of the catalytic core of Saccharomyces cerevesiae histone demethylase Rph1: insights into the substrate specificity and catalytic mechanism
Biochem.J., 433, 2011
3QO2
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BU of 3qo2 by Molmil
Structural insights for MPP8 chromodomain interaction with histone H3 lysine 9
Descriptor: 1,2-ETHANEDIOL, Histone H3 peptide, M-phase phosphoprotein 8
Authors:Chang, Y, Horton, J.R, Bedford, M.T, Zhang, X, Cheng, X.
Deposit date:2011-02-09
Release date:2011-04-06
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (2.49 Å)
Cite:Structural insights for MPP8 chromodomain interaction with histone H3 lysine 9: potential effect of phosphorylation on methyl-lysine binding.
J.Mol.Biol., 408, 2011
3QXY
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BU of 3qxy by Molmil
Human SETD6 in complex with RelA Lys310
Descriptor: 1,2-ETHANEDIOL, N-lysine methyltransferase SETD6, S-ADENOSYLMETHIONINE, ...
Authors:Chang, Y, Levy, D, Horton, J.R, Peng, J, Zhang, X, Gozani, O, Cheng, X.
Deposit date:2011-03-02
Release date:2011-05-25
Last modified:2024-02-21
Method:X-RAY DIFFRACTION (2.09 Å)
Cite:Structural basis of SETD6-mediated regulation of the NF-kB network via methyl-lysine signaling.
Nucleic Acids Res., 39, 2011
3FPD
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BU of 3fpd by Molmil
G9a-like protein lysine methyltransferase inhibition by BIX-01294
Descriptor: Histone-lysine N-methyltransferase, H3 lysine-9 specific 5, N-(1-benzylpiperidin-4-yl)-6,7-dimethoxy-2-(4-methyl-1,4-diazepan-1-yl)quinazolin-4-amine, ...
Authors:Chang, Y, Zhang, X, Horton, J.R, Cheng, X.
Deposit date:2009-01-05
Release date:2009-02-17
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:Structural basis for G9a-like protein lysine methyltransferase inhibition by BIX-01294.
Nat.Struct.Mol.Biol., 16, 2009
3RC0
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BU of 3rc0 by Molmil
Human SETD6 in complex with RelA Lys310 peptide
Descriptor: 1,2-ETHANEDIOL, N-lysine methyltransferase SETD6, S-ADENOSYLMETHIONINE, ...
Authors:Chang, Y, Levy, D, Horton, J.R, Peng, J, Zhang, X, Gozani, O, Cheng, X.
Deposit date:2011-03-30
Release date:2011-05-25
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (2.19 Å)
Cite:Structural basis of SETD6-mediated regulation of the NF-kB network via methyl-lysine signaling.
Nucleic Acids Res., 39, 2011
4PGV
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BU of 4pgv by Molmil
Crystal structure of YetJ from Bacillus Subtilis at pH 8 by back soaking
Descriptor: Uncharacterized protein YetJ
Authors:Liu, Q, Chang, Y, Hendrickson, W.A, New York Consortium on Membrane Protein Structure (NYCOMPS)
Deposit date:2014-05-02
Release date:2014-06-04
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (2.61 Å)
Cite:Structural basis for a pH-sensitive calcium leak across membranes.
Science, 344, 2014
4PGW
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BU of 4pgw by Molmil
Crystal structure of YetJ from Bacillus Subtilis at pH 6 by Pt-SAD
Descriptor: PLATINUM (II) ION, Uncharacterized protein YetJ
Authors:Liu, Q, Chang, Y, Hendrickson, W.A, New York Consortium on Membrane Protein Structure (NYCOMPS)
Deposit date:2014-05-02
Release date:2014-06-04
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (3.6 Å)
Cite:Structural basis for a pH-sensitive calcium leak across membranes.
Science, 344, 2014
4PGS
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BU of 4pgs by Molmil
Crystal structure of YetJ from Bacillus Subtilis at pH 6 by soaking
Descriptor: Uncharacterized protein YetJ
Authors:Liu, Q, Chang, Y, Hendrickson, W.A, New York Consortium on Membrane Protein Structure (NYCOMPS)
Deposit date:2014-05-02
Release date:2014-06-04
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:Structural basis for a pH-sensitive calcium leak across membranes.
Science, 344, 2014
4PGU
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BU of 4pgu by Molmil
Crystal structure of YetJ from Bacillus Subtilis at pH 7 by soaking
Descriptor: Uncharacterized protein YetJ
Authors:Liu, Q, Chang, Y, Hendrickson, W.A, New York Consortium on Membrane Protein Structure (NYCOMPS)
Deposit date:2014-05-02
Release date:2014-06-04
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (3.401 Å)
Cite:Structural basis for a pH-sensitive calcium leak across membranes.
Science, 344, 2014
4PGR
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BU of 4pgr by Molmil
Crystal structure of YetJ from Bacillus Subtilis at pH 8
Descriptor: Uncharacterized protein YetJ
Authors:Liu, Q, Chang, Y, Hendrickson, W.A, New York Consortium on Membrane Protein Structure (NYCOMPS)
Deposit date:2014-05-02
Release date:2014-06-04
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (1.95 Å)
Cite:Structural basis for a pH-sensitive calcium leak across membranes.
Science, 344, 2014
4TKQ
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BU of 4tkq by Molmil
Native-SAD phasing for YetJ from Bacillus Subtilis
Descriptor: CALCIUM ION, CHLORIDE ION, Uncharacterized protein YetJ
Authors:Liu, Q, Chang, Y, Hendrickson, W.A, New York Consortium on Membrane Protein Structure (NYCOMPS)
Deposit date:2014-05-27
Release date:2014-06-18
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (2.8025 Å)
Cite:Multi-crystal native SAD analysis at 6 keV.
Acta Crystallogr.,Sect.D, 70, 2014
2LJV
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BU of 2ljv by Molmil
Solution structure of Rhodostomin G50L mutant
Descriptor: Disintegrin rhodostomin
Authors:Chuang, W, Shiu, J, Chen, C, Chen, Y, Chang, Y, Huang, C.
Deposit date:2011-09-29
Release date:2012-10-03
Last modified:2023-06-14
Method:SOLUTION NMR
Cite:Design of Integrin AlphaVbeta3-Specific Disintegrin for Cancer Therapy
To be Published
2M75
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BU of 2m75 by Molmil
The C-terminal Region of Disintegrin Modulate its 3D Conformation and Cooperate with RGD Loop in Regulating Recognitions of Integrins
Descriptor: Zinc metalloproteinase/disintegrin
Authors:Chuang, W, Chang, Y, Shiu, J.
Deposit date:2013-04-18
Release date:2013-05-22
Method:SOLUTION NMR
Cite:The C-terminal Region of Disintegrin Modulate its 3D Conformation and Cooperate with RGD Loop in Regulating Recognitions of Integrins
To be Published
2M7H
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BU of 2m7h by Molmil
The C-terminal Region of Disintegrin Modulate its 3D Conformation and Cooperate with RGD Loop in Regulating Integrin alpha-IIb beta-3 Recognition
Descriptor: Zinc metalloproteinase/disintegrin
Authors:Chuang, W, Chang, Y.
Deposit date:2013-04-22
Release date:2013-05-22
Method:SOLUTION NMR
Cite:The C-terminal Region of Disintegrin Modulate its 3D Conformation and Cooperate with RGD Loop in Regulating Recognitions of Integrins
To be Published
2M7F
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BU of 2m7f by Molmil
The C-terminal Region of Disintegrin Modulate its 3D Conformation and Cooperate with RGD Loop in Regulating Integrins Recognitions
Descriptor: Zinc metalloproteinase/disintegrin
Authors:Chuang, W, Chang, Y.
Deposit date:2013-04-22
Release date:2013-05-22
Method:SOLUTION NMR
Cite:The C-terminal Region of Disintegrin Modulate its 3D Conformation and Cooperate with RGD Loop in Regulating Recognitions of Integrins
To be Published
3OS5
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BU of 3os5 by Molmil
SET7/9-Dnmt1 K142me1 complex
Descriptor: 1,2-ETHANEDIOL, BETA-MERCAPTOETHANOL, Dnmt1, ...
Authors:Esteve, P.-O, Chang, Y, Samaranayake, M, Upadhyay, A.K, Horton, J.R, Feehery, G.R, Cheng, X, Pradhan, S.
Deposit date:2010-09-08
Release date:2010-12-15
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (1.69 Å)
Cite:A methylation and phosphorylation switch between an adjacent lysine and serine determines human DNMT1 stability.
Nat.Struct.Mol.Biol., 18, 2011
6NQ8
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BU of 6nq8 by Molmil
Crystal structure of YetJ mutant from Bacillus Subtilis - D171E
Descriptor: Uncharacterized protein YetJ
Authors:Guo, G, Chang, Y, Liu, Q.
Deposit date:2019-01-19
Release date:2019-04-17
Last modified:2023-10-11
Method:X-RAY DIFFRACTION (3.1 Å)
Cite:Ion and pH Sensitivity of a TMBIM Ca2+Channel.
Structure, 27, 2019
6NQ9
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BU of 6nq9 by Molmil
Crystal structure of YetJ mutant from Bacillus Subtilis - D195E
Descriptor: Uncharacterized protein YetJ
Authors:Guo, G, Chang, Y, Liu, Q.
Deposit date:2019-01-19
Release date:2019-04-17
Last modified:2023-10-11
Method:X-RAY DIFFRACTION (3.1 Å)
Cite:Ion and pH Sensitivity of a TMBIM Ca2+Channel.
Structure, 27, 2019

 

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