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6B0T
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BU of 6b0t by Molmil
Structural Insights into the Induced-fit Inhibition of Fascin by a Small Molecule
Descriptor: 4-methyl-N-(1-{[4-(trifluoromethyl)phenyl]methyl}-1H-indazol-3-yl)-1,2-oxazole-5-carboxamide, Fascin
Authors:Dey, R, Huang, X.Y.
Deposit date:2017-09-15
Release date:2018-04-18
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (2.8 Å)
Cite:Structural Insights into the Induced-fit Inhibition of Fascin by a Small-Molecule Inhibitor.
J. Mol. Biol., 430, 2018
7JJO
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BU of 7jjo by Molmil
Structural Basis of the Activation of Heterotrimeric Gs-protein by Isoproterenol-bound Beta1-Adrenergic Receptor
Descriptor: Beta1-Adrenergic Receptor, Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1, ...
Authors:Su, M, Zhu, L, Zhang, Y, Paknejad, N, Dey, R, Huang, J, Lee, M.Y, Williams, D, Jordan, K.D, Eng, E.T, Ernst, O.P, Meyerson, J.R, Hite, R.K, Walz, T, Liu, W, Huang, X.Y.
Deposit date:2020-07-27
Release date:2020-09-02
Last modified:2020-10-14
Method:ELECTRON MICROSCOPY (2.6 Å)
Cite:Structural Basis of the Activation of Heterotrimeric Gs-Protein by Isoproterenol-Bound beta 1 -Adrenergic Receptor.
Mol.Cell, 80, 2020
8U7E
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BU of 8u7e by Molmil
Structure of Sts-1 HP domain with rebamipide derivative
Descriptor: N-(4-ethylbenzoyl)-3-(2-oxo-1,2-dihydroquinolin-4-yl)-L-alanine, Ubiquitin-associated and SH3 domain-containing protein B
Authors:Aziz, F, Dey, R, French, J.B.
Deposit date:2023-09-15
Release date:2024-02-07
Last modified:2024-02-21
Method:X-RAY DIFFRACTION (2.63 Å)
Cite:Rebamipide and Derivatives are Potent, Selective Inhibitors of Histidine Phosphatase Activity of the Suppressor of T Cell Receptor Signaling Proteins.
J.Med.Chem., 67, 2024
8U5M
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BU of 8u5m by Molmil
Structure of Sts-1 HP domain with rebamipide
Descriptor: Rebamipide, Ubiquitin-associated and SH3 domain-containing protein B
Authors:Azia, F, Dey, R, French, J.B.
Deposit date:2023-09-12
Release date:2024-02-07
Last modified:2024-02-21
Method:X-RAY DIFFRACTION (2.46 Å)
Cite:Rebamipide and Derivatives are Potent, Selective Inhibitors of Histidine Phosphatase Activity of the Suppressor of T Cell Receptor Signaling Proteins.
J.Med.Chem., 67, 2024
7XUZ
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BU of 7xuz by Molmil
Crystal structure of a HDAC4-MEF2A-DNA ternary complex
Descriptor: DNA (5'-D(*TP*CP*TP*TP*AP*TP*AP*AP*AP*TP*AP*GP*T)-3'), DNA (5'-D(P*AP*CP*TP*AP*TP*TP*TP*AP*TP*AP*A)-3'), Histone deacetylase 4, ...
Authors:Dai, S.Y, Guo, L, Dey, R, Guo, M, Bates, D, Cayford, J, Chen, X.J, Wei, X.D, Chen, L, Chen, Y.H.
Deposit date:2022-05-20
Release date:2023-11-29
Method:X-RAY DIFFRACTION (3.591 Å)
Cite:Structural insights into transcription regulation by the higher-order HDAC4-MEF2-DNA complex
To Be Published
3KMD
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BU of 3kmd by Molmil
Crystal structure of the p53 core domain bound to a full consensus site as a self-assembled tetramer
Descriptor: 5'-D(*GP*GP*GP*CP*AP*TP*GP*CP*CP*TP*AP*GP*GP*CP*AP*TP*GP*CP*C)-3', Cellular tumor antigen p53, ZINC ION
Authors:Chen, Y, Dey, R, Chen, L.
Deposit date:2009-11-10
Release date:2010-02-23
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (2.15 Å)
Cite:Crystal structure of the p53 core domain bound to a full consensus site as a self-assembled tetramer.
Structure, 18, 2010
3KOV
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BU of 3kov by Molmil
Structure of MEF2A bound to DNA reveals a completely folded MADS-box/MEF2 domain that recognizes DNA and recruits transcription co-factors
Descriptor: DNA (5'-D(*AP*AP*CP*TP*AP*TP*TP*TP*AP*TP*AP*AP*G)-3'), DNA (5'-D(*TP*CP*TP*TP*AP*TP*AP*AP*AP*TP*AP*GP*T)-3'), Myocyte-specific enhancer factor 2A
Authors:Wu, Y, Dey, R, Han, A, Jayathilaka, N, Philips, M, Ye, J, Chen, L.
Deposit date:2009-11-14
Release date:2010-02-16
Last modified:2024-02-21
Method:X-RAY DIFFRACTION (2.9 Å)
Cite:Structure of the MADS-box/MEF2 Domain of MEF2A Bound to DNA and Its Implication for Myocardin Recruitment.
J.Mol.Biol., 397, 2010
2FP2
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BU of 2fp2 by Molmil
Secreted Chorismate Mutase from Mycobacterium tuberculosis
Descriptor: 8-HYDROXY-2-OXA-BICYCLO[3.3.1]NON-6-ENE-3,5-DICARBOXYLIC ACID, Chorismate mutase
Authors:Okvist, M, Dey, R, Sasso, S, Grahn, E, Kast, P, Krengel, U.
Deposit date:2006-01-15
Release date:2006-03-28
Last modified:2023-08-30
Method:X-RAY DIFFRACTION (1.64 Å)
Cite:1.6A Crystal Structure of the Secreted Chorismate Mutase from Mycobacterium tuberculosis: Novel Fold Topology Revealed
J.Mol.Biol., 357, 2006
2FP1
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BU of 2fp1 by Molmil
Secreted Chorismate Mutase from Mycobacterium tuberculosis
Descriptor: Chorismate mutase, LEAD (II) ION
Authors:Okvist, M, Dey, R, Sasso, S, Grahn, E, Kast, P, Krengel, U.
Deposit date:2006-01-15
Release date:2006-03-28
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (1.55 Å)
Cite:1.6A Crystal Structure of the Secreted Chorismate Mutase from Mycobacterium tuberculosis: Novel Fold Topology Revealed
J.Mol.Biol., 357, 2006
4HCA
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BU of 4hca by Molmil
DNA binding by GATA transcription factor-complex 1
Descriptor: DNA (5'-D(*AP*AP*TP*GP*TP*CP*CP*AP*TP*CP*TP*GP*AP*TP*AP*AP*GP*AP*CP*G)-3'), DNA (5'-D(*TP*TP*CP*GP*TP*CP*TP*TP*AP*TP*CP*AP*GP*AP*TP*GP*GP*AP*CP*A)-3'), Trans-acting T-cell-specific transcription factor GATA-3, ...
Authors:Chen, Y, Bates, D.L, Dey, R, Chen, L.
Deposit date:2012-09-28
Release date:2012-12-05
Last modified:2024-02-28
Method:X-RAY DIFFRACTION (2.8 Å)
Cite:DNA Binding by GATA Transcription Factor Suggests Mechanisms of DNA Looping and Long-Range Gene Regulation.
Cell Rep, 2, 2012
4HC7
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BU of 4hc7 by Molmil
Crystal structure of the full DNA binding domain of GATA3-complex 2
Descriptor: DNA (5'-D(*AP*AP*GP*GP*TP*TP*AP*TP*CP*TP*CP*TP*GP*AP*TP*TP*TP*AP*GP*G)-3'), DNA (5'-D(*TP*TP*CP*CP*TP*AP*AP*AP*TP*CP*AP*GP*AP*GP*AP*TP*AP*AP*CP*C)-3'), Trans-acting T-cell-specific transcription factor GATA-3, ...
Authors:Chen, Y, Bates, D.L, Dey, R, Chen, L.
Deposit date:2012-09-28
Release date:2012-12-05
Last modified:2024-02-28
Method:X-RAY DIFFRACTION (2.65 Å)
Cite:DNA Binding by GATA Transcription Factor Suggests Mechanisms of DNA Looping and Long-Range Gene Regulation.
Cell Rep, 2, 2012
4HC9
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BU of 4hc9 by Molmil
DNA binding by GATA transcription factor-complex 3
Descriptor: DNA (5'-D(*AP*AP*GP*GP*TP*TP*AP*TP*CP*TP*CP*TP*GP*AP*TP*TP*TP*AP*GP*G)-3'), DNA (5'-D(*TP*TP*CP*CP*TP*AP*AP*AP*TP*CP*AP*GP*AP*GP*AP*TP*AP*AP*CP*C)-3'), Trans-acting T-cell-specific transcription factor GATA-3, ...
Authors:Chen, Y, Bates, D.L, Dey, R, Chen, L.
Deposit date:2012-09-28
Release date:2012-12-05
Last modified:2024-02-28
Method:X-RAY DIFFRACTION (1.6 Å)
Cite:DNA Binding by GATA Transcription Factor Suggests Mechanisms of DNA Looping and Long-Range Gene Regulation.
Cell Rep, 2, 2012
3MU6
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BU of 3mu6 by Molmil
Inhibiting the Binding of Class IIa Histone Deacetylases to Myocyte Enhancer Factor-2 by Small Molecules
Descriptor: (3E)-N~8~-(2-aminophenyl)-N~1~-phenyloct-3-enediamide, DNA (5'-D(*AP*AP*AP*GP*CP*TP*AP*TP*TP*AP*TP*TP*AP*GP*CP*TP*T)-3'), DNA (5'-D(*TP*AP*AP*GP*CP*TP*AP*AP*TP*AP*AP*TP*AP*GP*CP*TP*T)-3'), ...
Authors:Jayathilaka, N, Han, A, Gaffney, K, Dey, R, He, J, Ye, J, Gao, T, Petasis, N.A, Chen, L.
Deposit date:2010-05-01
Release date:2011-11-02
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (2.434 Å)
Cite:Inhibition of the function of class IIa HDACs by blocking their interaction with MEF2.
Nucleic Acids Res., 40, 2012

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PDB entries from 2024-03-27

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