Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
Search by PDB author
3BE8
DownloadVisualize
BU of 3be8 by Molmil
Crystal structure of the synaptic protein neuroligin 4
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, CHLORIDE ION, CITRATE ANION, ...
Authors:Fabrichny, I.P, Leone, P, Sulzenbacher, G, Comoletti, D, Miller, M.T, Taylor, P, Bourne, Y, Marchot, P.
Deposit date:2007-11-16
Release date:2008-01-29
Last modified:2023-11-01
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Structural Analysis of the Synaptic Protein Neuroligin and Its beta-Neurexin Complex: Determinants for Folding and Cell Adhesion
Neuron, 56, 2007
1C2B
DownloadVisualize
BU of 1c2b by Molmil
ELECTROPHORUS ELECTRICUS ACETYLCHOLINESTERASE
Descriptor: ACETYLCHOLINESTERASE
Authors:Bourne, Y, Marchot, P.
Deposit date:1999-07-26
Release date:1999-12-29
Last modified:2021-06-02
Method:X-RAY DIFFRACTION (4.5 Å)
Cite:Conformational flexibility of the acetylcholinesterase tetramer suggested by x-ray crystallography.
J.Biol.Chem., 274, 1999
1C2O
DownloadVisualize
BU of 1c2o by Molmil
ELECTROPHORUS ELECTRICUS ACETYLCHOLINESTERASE
Descriptor: ACETYLCHOLINESTERASE
Authors:Bourne, Y, Marchot, P.
Deposit date:1999-07-26
Release date:2000-01-19
Last modified:2021-06-02
Method:X-RAY DIFFRACTION (4.2 Å)
Cite:Conformational flexibility of the acetylcholinesterase tetramer suggested by x-ray crystallography.
J.Biol.Chem., 274, 1999
4QWW
DownloadVisualize
BU of 4qww by Molmil
Crystal structure of the Fab410-BfAChE complex
Descriptor: 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, Acetylcholinesterase, ...
Authors:Bourne, Y, Renault, L, Marchot, P.
Deposit date:2014-07-17
Release date:2014-11-26
Last modified:2023-09-20
Method:X-RAY DIFFRACTION (2.7 Å)
Cite:Crystal Structure of Snake Venom Acetylcholinesterase in Complex with Inhibitory Antibody Fragment Fab410 Bound at the Peripheral Site: EVIDENCE FOR OPEN AND CLOSED STATES OF A BACK DOOR CHANNEL.
J.Biol.Chem., 290, 2015
4XK9
DownloadVisualize
BU of 4xk9 by Molmil
Crystal structure of A-AChBP in complex with pinnatoxin G
Descriptor: CHLORIDE ION, Pinnatoxin G, Soluble acetylcholine receptor
Authors:Bourne, Y, Sulzenbacher, G, Marchot, P.
Deposit date:2015-01-10
Release date:2015-06-03
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Marine Macrocyclic Imines, Pinnatoxins A and G: Structural Determinants and Functional Properties to Distinguish Neuronal alpha 7 from Muscle alpha 12 beta gamma delta nAChRs.
Structure, 23, 2015
4XHE
DownloadVisualize
BU of 4xhe by Molmil
Crystal Structure of A-AChBP in complex with pinnatoxin A
Descriptor: CALCIUM ION, CHLORIDE ION, Pinnatoxin A, ...
Authors:Bourne, Y, Sulzenbacher, G, Marchot, P.
Deposit date:2015-01-05
Release date:2015-06-03
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Marine Macrocyclic Imines, Pinnatoxins A and G: Structural Determinants and Functional Properties to Distinguish Neuronal alpha 7 from Muscle alpha 12 beta gamma delta nAChRs.
Structure, 23, 2015
1YI5
DownloadVisualize
BU of 1yi5 by Molmil
Crystal structure of the a-cobratoxin-AChBP complex
Descriptor: Acetylcholine-binding protein, Long neurotoxin 1
Authors:Bourne, Y, Talley, T.T, Hansen, S.B, Taylor, P, Marchot, P.
Deposit date:2005-01-11
Release date:2005-05-17
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (4.2 Å)
Cite:Crystal structure of a Cbtx-AChBP complex reveals essential interactions between snake alpha-neurotoxins and nicotinic receptors
Embo J., 24, 2005
1MAH
DownloadVisualize
BU of 1mah by Molmil
FASCICULIN2-MOUSE ACETYLCHOLINESTERASE COMPLEX
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, ACETYLCHOLINESTERASE, FASCICULIN 2
Authors:Bourne, Y, Taylor, P, Marchot, P.
Deposit date:1995-11-21
Release date:1996-04-03
Last modified:2021-03-31
Method:X-RAY DIFFRACTION (3.2 Å)
Cite:Acetylcholinesterase inhibition by fasciculin: crystal structure of the complex.
Cell(Cambridge,Mass.), 83, 1995
1FAS
DownloadVisualize
BU of 1fas by Molmil
1.9 ANGSTROM RESOLUTION STRUCTURE OF FASCICULIN 1, AN ANTI-ACETYLCHOLINESTERASE TOXIN FROM GREEN MAMBA SNAKE VENOM
Descriptor: FASCICULIN 1
Authors:Le Du, M.H, Marchot, P, Bougis, P.E, Fontecilla-Camps, J.C.
Deposit date:1992-08-07
Release date:1993-10-31
Last modified:2017-11-29
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:1.9-A resolution structure of fasciculin 1, an anti-acetylcholinesterase toxin from green mamba snake venom.
J.Biol.Chem., 267, 1992
4AEH
DownloadVisualize
BU of 4aeh by Molmil
Crystal structure of the anti-AaHI Fab9C2 antibody
Descriptor: FAB ANTIBODY, HEAVY CHAIN, LIGHT CHAIN
Authors:Fabrichny, I.P, Mondielli, G, Conrod, S, Martin-Eauclaire, M.F, Bourne, Y, Marchot, P.
Deposit date:2012-01-10
Release date:2012-03-07
Last modified:2012-05-02
Method:X-RAY DIFFRACTION (1.6 Å)
Cite:Structural Insights Into Antibody Sequestering and Neutralizing of Na+-Channel & [Alpha]-Type Modulator from Old-World Scorpion Venom
J.Biol.Chem., 287, 2012
1N5M
DownloadVisualize
BU of 1n5m by Molmil
Crystal structure of the mouse acetylcholinesterase-gallamine complex
Descriptor: 2,2',2"-[1,2,3-BENZENE-TRIYLTRIS(OXY)]TRIS[N,N,N-TRIETHYLETHANAMINIUM], 2-acetamido-2-deoxy-beta-D-glucopyranose, CARBONATE ION, ...
Authors:Bourne, Y, Taylor, P, Radic, Z, Marchot, P.
Deposit date:2002-11-06
Release date:2003-02-04
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Structural insights into ligand interactions at the acetylcholinesterase peripheral anionic site
EMBO J., 22, 2003
1N5R
DownloadVisualize
BU of 1n5r by Molmil
Crystal structure of the mouse acetylcholinesterase-propidium complex
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 3,8-DIAMINO-5[3-(DIETHYLMETHYLAMMONIO)PROPYL]-6-PHENYLPHENANTHRIDINIUM, ACETIC ACID, ...
Authors:Bourne, Y, Taylor, P, Radic, Z, Marchot, P.
Deposit date:2002-11-07
Release date:2003-02-04
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (2.25 Å)
Cite:Structural insights into ligand interactions at the acetylcholinesterase peripheral anionic site
EMBO J., 22, 2003
1Q83
DownloadVisualize
BU of 1q83 by Molmil
Crystal structure of the mouse acetylcholinesterase-TZ2PA6 syn complex
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 3,8-DIAMINO-6-PHENYL-5-[6-[1-[2-[(1,2,3,4-TETRAHYDRO-9-ACRIDINYL)AMINO]ETHYL]-1H-1,2,3-TRIAZOL-5-YL]HEXYL]-PHENANTHRIDINIUM, Acetylcholinesterase, ...
Authors:Bourne, Y, Kolb, H.C, Radic, Z, Sharpless, K.B, Taylor, P, Marchot, P.
Deposit date:2003-08-20
Release date:2004-02-10
Last modified:2023-08-16
Method:X-RAY DIFFRACTION (2.65 Å)
Cite:Freeze-frame inhibitor captures acetylcholinesterase in a unique conformation.
Proc.Natl.Acad.Sci.Usa, 101, 2004
1Q84
DownloadVisualize
BU of 1q84 by Molmil
Crystal structure of the mouse acetylcholinesterase-TZ2PA6 anti complex
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 3,8-DIAMINO-6-PHENYL-5-[6-[1-[2-[(1,2,3,4-TETRAHYDRO-9-ACRIDINYL)AMINO]ETHYL]-1H-1,2,3-TRIAZOL-4-YL]HEXYL]-PHENANTHRIDINIUM, Acetylcholinesterase, ...
Authors:Bourne, Y, Kolb, H.C, Radic, Z, Sharpless, K.B, Taylor, P, Marchot, P.
Deposit date:2003-08-20
Release date:2004-02-10
Last modified:2023-08-16
Method:X-RAY DIFFRACTION (2.45 Å)
Cite:Freeze-frame inhibitor captures acetylcholinesterase in a unique conformation.
Proc.Natl.Acad.Sci.Usa, 101, 2004
4AEI
DownloadVisualize
BU of 4aei by Molmil
Crystal structure of the AaHII-Fab4C1 complex
Descriptor: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, ALPHA-MAMMAL TOXIN AAH2, CHLORIDE ION, ...
Authors:Fabrichny, I.P, Mondielli, G, Conrod, S, Martin-Eauclaire, M.F, Bourne, Y, Marchot, P.
Deposit date:2012-01-10
Release date:2012-03-07
Last modified:2023-12-20
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Structural Insights Into Antibody Sequestering and Neutralizing of Na+-Channel & [Alpha]-Type Modulator from Old-World Scorpion Venom
J.Biol.Chem., 287, 2012
1J07
DownloadVisualize
BU of 1j07 by Molmil
Crystal structure of the mouse acetylcholinesterase-decidium complex
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 3,8-DIAMINO-5,10'-(TRIMETHYLAMMONIUM)DECYL-6-PHENYL PHENANTHRIDINIUM, CARBONATE ION, ...
Authors:Bourne, Y, Taylor, P, Radic, Z, Marchot, P.
Deposit date:2002-11-07
Release date:2003-02-04
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (2.35 Å)
Cite:Structural insights into ligand interactions at the acetylcholinesterase peripheral anionic site
EMBO J., 22, 2003
1J06
DownloadVisualize
BU of 1j06 by Molmil
Crystal structure of mouse acetylcholinesterase in the apo form
Descriptor: 2-(2-ETHOXYETHOXY)ETHANOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, CARBONATE ION, ...
Authors:Bourne, Y, Taylor, P, Radic, Z, Marchot, P.
Deposit date:2002-11-07
Release date:2003-02-04
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.35 Å)
Cite:Structural insights into ligand interactions at the acetylcholinesterase peripheral anionic site
EMBO J., 22, 2003
1UKC
DownloadVisualize
BU of 1ukc by Molmil
Crystal Structure of Aspergillus niger EstA
Descriptor: 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Bourne, Y, Hasper, A.A, Chahinian, H, Juin, M, De Graaff, L.H, Marchot, P.
Deposit date:2003-08-19
Release date:2004-07-27
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:Aspergillus niger protein EstA defines a new class of fungal esterases within the alpha/beta hydrolase fold superfamily of proteins
STRUCTURE, 12, 2004
1KU6
DownloadVisualize
BU of 1ku6 by Molmil
Fasciculin 2-Mouse Acetylcholinesterase Complex
Descriptor: 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, ACETYLCHOLINESTERASE, ...
Authors:Bourne, Y, Burmeister, W, Taylor, P, Marchot, P.
Deposit date:2002-01-21
Release date:2003-12-23
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:Structural insights into ligand interactions at the acetylcholinesterase peripheral anionic site.
EMBO J., 22, 2003
1MAA
DownloadVisualize
BU of 1maa by Molmil
MOUSE ACETYLCHOLINESTERASE CATALYTIC DOMAIN, GLYCOSYLATED PROTEIN
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[beta-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ACETYLCHOLINESTERASE, ...
Authors:Bourne, Y, Taylor, P, Bougis, P.E, Marchot, P.
Deposit date:1998-11-04
Release date:1999-04-20
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (2.9 Å)
Cite:Crystal structure of mouse acetylcholinesterase. A peripheral site-occluding loop in a tetrameric assembly.
J.Biol.Chem., 274, 1999
5EHN
DownloadVisualize
BU of 5ehn by Molmil
mAChE-syn TZ2PA5 complex
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 6-phenyl-5-[5-[3-[2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethyl]-1,2,3-triazol-4-yl]pentyl]phenanthridin-5-ium-3,8-diamine, Acetylcholinesterase, ...
Authors:Bourne, Y, Marchot, P.
Deposit date:2015-10-28
Release date:2016-01-20
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:Steric and Dynamic Parameters Influencing In Situ Cycloadditions to Form Triazole Inhibitors with Crystalline Acetylcholinesterase.
J.Am.Chem.Soc., 138, 2016
5EIH
DownloadVisualize
BU of 5eih by Molmil
mAChE-TZ2/PA5 complex
Descriptor: 5-hept-6-ynyl-6-phenyl-phenanthridin-5-ium-3,8-diamine, ACETATE ION, Acetylcholinesterase, ...
Authors:Bourne, Y, Marchot, P.
Deposit date:2015-10-29
Release date:2016-01-20
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (2.7 Å)
Cite:Steric and Dynamic Parameters Influencing In Situ Cycloadditions to Form Triazole Inhibitors with Crystalline Acetylcholinesterase.
J.Am.Chem.Soc., 138, 2016
5EHZ
DownloadVisualize
BU of 5ehz by Molmil
mAChE-syn TZ2PA5 complex from an equimolar mixture of the syn/anti isomers
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 6-phenyl-5-[5-[3-[2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethyl]-1,2,3-triazol-4-yl]pentyl]phenanthridin-5-ium-3,8-diamine, Acetylcholinesterase, ...
Authors:Bourne, Y, Marchot, P.
Deposit date:2015-10-29
Release date:2016-01-20
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:Steric and Dynamic Parameters Influencing In Situ Cycloadditions to Form Triazole Inhibitors with Crystalline Acetylcholinesterase.
J.Am.Chem.Soc., 138, 2016
5EIA
DownloadVisualize
BU of 5eia by Molmil
mACHE-anti TZ2PA5 complex from a 1:6 mixture of the syn/anti isomers
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 6-phenyl-5-[5-[1-[2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethyl]-1,2,3-triazol-4-yl]pentyl]phenanthridin-5-ium-3,8-diamine, Acetylcholinesterase, ...
Authors:Bourne, Y, Marchot, P.
Deposit date:2015-10-29
Release date:2016-01-20
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (2.7 Å)
Cite:Steric and Dynamic Parameters Influencing In Situ Cycloadditions to Form Triazole Inhibitors with Crystalline Acetylcholinesterase.
J.Am.Chem.Soc., 138, 2016
5EIE
DownloadVisualize
BU of 5eie by Molmil
mAChE-TZ2 complex
Descriptor: 2,5,8,11,14,17,20,23-OCTAOXAPENTACOSAN-25-OL, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Bourne, Y, Marchot, P.
Deposit date:2015-10-29
Release date:2016-01-20
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:Steric and Dynamic Parameters Influencing In Situ Cycloadditions to Form Triazole Inhibitors with Crystalline Acetylcholinesterase.
J.Am.Chem.Soc., 138, 2016

 

123>

217705

PDB entries from 2024-03-27

PDB statisticsPDBj update infoContact PDBjnumon