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6BS0

JAK2 JH2 in complex with 63552444

Summary for 6BS0
Entry DOI10.2210/pdb6bs0/pdb
DescriptorTyrosine-protein kinase JAK2, 4-(5-aminopyrazin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine, GLYCEROL, ... (4 entities in total)
Functional Keywordspseudokinase domain, transferase-transferase inhibitor complex, transferase/transferase inhibitor
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight33623.48
Authors
Puleo, D.E.,Schlessinger, J. (deposition date: 2017-12-01, release date: 2018-08-22, Last modification date: 2023-10-04)
Primary citationPuleo, D.E.,Schlessinger, J.
JAK2 JH2 Binders
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.541 Å)
Structure validation

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