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5XY1

Crystal structure of Lyn kinase domain in complex with N-(1H-indazol-6-yl)-8-(piperidin-4-yloxy)-6-propylquinazolin-2-amine

Summary for 5XY1
Entry DOI10.2210/pdb5xy1/pdb
DescriptorTyrosine-protein kinase Lyn, N-(1H-indazol-6-yl)-8-piperidin-4-yloxy-6-propyl-quinazolin-2-amine (3 entities in total)
Functional Keywordskinase, transferase
Biological sourceHomo sapiens (Human)
Cellular locationCell membrane: P07948
Total number of polymer chains1
Total formula weight32200.03
Authors
Kim, H.T. (deposition date: 2017-07-05, release date: 2017-08-02, Last modification date: 2023-11-22)
Primary citationKim, H.T.
Crystal structure of Lyn kinase domain in complex with N-(1H-indazol-6-yl)-8-(piperidin-4-yloxy)-6-propylquinazolin-2-amine
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.7 Å)
Structure validation

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