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5W9D

Estrogen Receptor Alpha Ligand Binding Domain C381S, C417S, C530S Mutant in Complex with Endoxifen

Summary for 5W9D
Entry DOI10.2210/pdb5w9d/pdb
DescriptorEstrogen receptor, Endoxifen (3 entities in total)
Functional Keywordsbreast cancer, selective estrogen receptor modulator, transcription
Biological sourceHomo sapiens (Human)
Total number of polymer chains2
Total formula weight57457.39
Authors
Fanning, S.W.,Greene, G.L. (deposition date: 2017-06-23, release date: 2017-10-11, Last modification date: 2023-10-04)
Primary citationMaximov, P.Y.,Abderrahman, B.,Fanning, S.W.,Sengupta, S.,Fan, P.,Curpan, R.F.,Rincon, D.M.Q.,Greenland, J.A.,Rajan, S.S.,Greene, G.L.,Jordan, V.C.
Endoxifen, 4-Hydroxytamoxifen and an Estrogenic Derivative Modulate Estrogen Receptor Complex Mediated Apoptosis in Breast Cancer.
Mol. Pharmacol., 94:812-822, 2018
Cited by
PubMed: 29739819
DOI: 10.1124/mol.117.111385
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.6464 Å)
Structure validation

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