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5UVT

BRD4_BD2_A-1454056

Summary for 5UVT
Entry DOI10.2210/pdb5uvt/pdb
Related5UVS 5UVU 5UVV 5UVW 5UVX 5UVY 5UVZ
DescriptorBromodomain-containing protein 4, 7-(cyclopropylmethyl)-2-methyl-10-[(propan-2-yl)sulfonyl]-2,4,6,7-tetrahydro-3H-2,4,7-triazadibenzo[cd,f]azulen-3-one (3 entities in total)
Functional Keywordshelix bundle, signaling protein-inhibitor complex, signaling protein/inhibitor
Biological sourceHomo sapiens (Human)
Cellular locationNucleus: O60885
Total number of polymer chains1
Total formula weight13218.45
Authors
Park, C.H. (deposition date: 2017-02-20, release date: 2017-06-21, Last modification date: 2024-03-06)
Primary citationPark, C.H.
Complex structure of BRD4_BD2_A-1454056
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.67 Å)
Structure validation

217705

PDB entries from 2024-03-27

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