5UR9

Enantiomer-Specific Binding of the Potent Antinociceptive Agent SBFI-26 to Anandamide transporters FABP5

Summary for 5UR9

• Entry DOI: 10.2210/pdb5ur9/pdb
• Related: 5URA
• Descriptor: Fatty acid-binding protein, epidermal, (1S,2S,3S,4S)-3-{[(naphthalen-1-yl)oxy]carbonyl}-2,4-diphenylcyclobutane-1-carboxylic acid, SULFATE ION, ... (6 entities in total)
• Functional Keywords: inhibitor, lipid binding protein-inhibitor complex, lipid binding protein/inhibitor
• Biological source: Homo sapiens (Human)
• Total number of polymer chains: 8
• Total formula weight: 129952.62

Authors

Hsu, H.-C.,Li, H. (deposition date: 2017-02-09, release date: 2017-08-23, Last modification date: 2023-10-04)

• Primary citation: Hsu, H.C.,Tong, S.,Zhou, Y.,Elmes, M.W.,Yan, S.,Kaczocha, M.,Deutsch, D.G.,Rizzo, R.C.,Ojima, I.,Li, H.; The Antinociceptive Agent SBFI-26 Binds to Anandamide Transporters FABP5 and FABP7 at Two Different Sites.; Biochemistry, 56:3454-3462, 2017; PubMed: 28632393; DOI: 10.1021/acs.biochem.7b00194

Experimental method

X-RAY DIFFRACTION (2.19800343737 Å)