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5LGS

Crystal structure of mouse CARM1 in complex with ligand P2C3u

Summary for 5LGS
Entry DOI10.2210/pdb5lgs/pdb
DescriptorHistone-arginine methyltransferase CARM1, Polyadenylate-binding protein 1, SULFATE ION, ... (9 entities in total)
Functional Keywordsprotein arginine methyltransferase, catalytic domain, chromatin regulator, mrna processing, mrna splicing, nucleus, s-adenosyl-l-methionine, transcription, transcription regulation, transferase
Biological sourceMus musculus (Mouse)
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Cellular locationNucleus: Q9WVG6
Cytoplasm: P11940
Total number of polymer chains8
Total formula weight169124.22
Authors
Marechal, N.,Troffer-Charlier, N.,Cura, V.,Bonnefond, L.,Cavarelli, J. (deposition date: 2016-07-08, release date: 2017-03-22, Last modification date: 2024-01-10)
Primary citationvan Haren, M.J.,Marechal, N.,Troffer-Charlier, N.,Cianciulli, A.,Sbardella, G.,Cavarelli, J.,Martin, N.I.
Transition state mimics are valuable mechanistic probes for structural studies with the arginine methyltransferase CARM1.
Proc. Natl. Acad. Sci. U.S.A., 114:3625-3630, 2017
Cited by
PubMed: 28330993
DOI: 10.1073/pnas.1618401114
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.1 Å)
Structure validation

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