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5JNA

Crystal structure for the complex of human carbonic anhydrase IV and topiramate

Summary for 5JNA
Entry DOI10.2210/pdb5jna/pdb
Related5JN8 5JN9 5JNC 5JND
DescriptorCarbonic anhydrase 4, ZINC ION, [(3aS,5aR,8aR,8bS)-2,2,7,7-tetramethyltetrahydro-3aH-bis[1,3]dioxolo[4,5-b:4',5'-d]pyran-3a-yl]methyl sulfamate, ... (7 entities in total)
Functional Keywordscarbonic anhydrase, lyase, zinc, inhibitor binding, lyase-lyase inhibitor complex, lyase/lyase inhibitor
Biological sourceHomo sapiens (Human)
Total number of polymer chains4
Total formula weight124298.89
Authors
Chen, Z.,Waheed, A.,Di Cera, E.,Sly, W.S. (deposition date: 2016-04-29, release date: 2017-05-03, Last modification date: 2023-09-27)
Primary citationMickeviciute, A.,Timm, D.D.,Gedgaudas, M.,Linkuviene, V.,Chen, Z.,Waheed, A.,Michailoviene, V.,Zubriene, A.,Smirnov, A.,Capkauskaite, E.,Baranauskiene, L.,Jachno, J.,Revuckiene, J.,Manakova, E.,Grazulis, S.,Matuliene, J.,Di Cera, E.,Sly, W.S.,Matulis, D.
Intrinsic thermodynamics of high affinity inhibitor binding to recombinant human carbonic anhydrase IV.
Eur. Biophys. J., 47:271-290, 2018
Cited by
PubMed: 28975383
DOI: 10.1007/s00249-017-1256-0
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2 Å)
Structure validation

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