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5JAO

Exploitation of a Novel Binding Pocket in Human Lipoprotein-Associated Phospholipase A2 (Lp-PLA2) Discovered Through X-Ray Fragment Screening

Summary for 5JAO
Entry DOI10.2210/pdb5jao/pdb
DescriptorPlatelet-activating factor acetylhydrolase, CALCIUM ION, CHLORIDE ION, ... (6 entities in total)
Functional Keywordsphospholipase, lipid metabolism, hydrolase
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight44574.49
Authors
Day, P.J. (deposition date: 2016-04-12, release date: 2016-05-25, Last modification date: 2019-10-16)
Primary citationWoolford, A.J.,Pero, J.E.,Aravapalli, S.,Berdini, V.,Coyle, J.E.,Day, P.J.,Dodson, A.M.,Grondin, P.,Holding, F.P.,Lee, L.Y.,Li, P.,Manas, E.S.,Marino, J.,Martin, A.C.,McCleland, B.W.,McMenamin, R.L.,Murray, C.W.,Neipp, C.E.,Page, L.W.,Patel, V.K.,Potvain, F.,Rich, S.,Rivero, R.A.,Smith, K.,Somers, D.O.,Trottet, L.,Velagaleti, R.,Williams, G.,Xie, R.
Exploitation of a Novel Binding Pocket in Human Lipoprotein-Associated Phospholipase A2 (Lp-PLA2) Discovered through X-ray Fragment Screening.
J.Med.Chem., 59:5356-5367, 2016
Cited by
PubMed: 27167608
DOI: 10.1021/acs.jmedchem.6b00212
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.06 Å)
Structure validation

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